Zobrazeno 1 - 5
of 5
pro vyhledávání: '"Robin Leguijt"'
Autor:
Bas Dros, Grietje Molema, Gabriela Leusink-Ionescu, Catherine Saccavini, Robin Leguijt, Jean-Paul G. Seerden, Richard M. Kellogg, Jan A. A. M. Kamps, Titia E. Woudenberg-Vrenken, Edith Gelens
Publikováno v:
Bioorganic & Medicinal Chemistry Letters, 24(5), 1352-1357. American Chemical Society
The design, synthesis and biological evaluation of novel triazolyl p38 alpha MAPK inhibitors with improved water solubility for formulation in cationic liposomes (SAINT-O-Somes) targeted at diseased endothelial cells is described. Water-solubilizing
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ca940e89d6bc5797224adde05e2c54e4
https://doi.org/10.1016/j.bmcl.2014.01.034
https://doi.org/10.1016/j.bmcl.2014.01.034
Publikováno v:
Journal of Carbohydrate Chemistry. 26:279-303
d‐glucosamine propane‐1,3‐diyl dithioacetal is a versatile synthetic building block, especially when being incorporated with the Corey‐Seebach method. Hence, exploring compatible protecting group patterns on this compound mainly for use with
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::cb002620982758b19f507aea340568ed
https://doi.org/10.1080/07328300701540183
https://doi.org/10.1080/07328300701540183
Publikováno v:
Synthesis. 2006:4212-4218
While 3,4;5,6-di-O-isopropylidene-N-phthaloyl-d-glucosamine propane-1,3-diyl dithioacetal (2) underwent fast β-elimination, the corresponding N-acetyl derivative 3 was easily deprotonated with butyllithium to form the dilithiated intermediate 7, whi
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::b672ef0b3f044256b81e7112ac675228
https://doi.org/10.1055/s-2006-950359
https://doi.org/10.1055/s-2006-950359
Publikováno v:
Synthesis. 2006:2242-2250
Versatile 3,4,5-tri-O-protected 2-acylamino-2-deoxy-6-O-tosyl-D-glucose propane-1,3-diyl dithioacetal intermediates were efficiently synthesized from D-glucosamine propane-1,3-diyl dithioacetal or its derivatives. Intramolecular cyclizations from the
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::0a98587bceaf654739bc20ac88da6610
https://doi.org/10.1055/s-2006-942430
https://doi.org/10.1055/s-2006-942430
Publikováno v:
XXIst International Carbohydrate Symposium 2002.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::28e690512217955b5f91031cad01bf30
https://doi.org/10.1100/tsw.2002.608
https://doi.org/10.1100/tsw.2002.608