Zobrazeno 1 - 4
of 4
pro vyhledávání: '"Robert Casella"'
Autor:
Tieguang Yao, Liangwei Wu, Craig S. Donald, Douglas Ferguson, Lei Wang, Andrew Pike, Jianyan Wang, Justin Cidado, Dedong Wu, Kurt Gordon Pike, Kumar Thakur, Chungang Gu, Calum Cook, James Horstick, Tyler Grebe, Theresa Proia, Darren Stead, Alexander Hird, Michelle Lamb, Wenlin Shao, Nichole O'Connell, Yun Jiang, Sudhir M. Hande, Bin Yang, Janet Hawkins, Barlaam Bernard Christophe, Neil Sumner, Melissa Vasbinder, Andrew D. Ferguson, Jane E. Moore, Jeffrey G. Varnes, Bryan Roberts, Maryann San Martin, Lisa Drew, Ujjal Sarkar, Allan Dishington, Chris De Savi, Robert Casella, Steve C. Glossop, Jane L. Holmes, Thomas M. McGuire
Publikováno v:
Journal of Medicinal Chemistry. 63:15564-15590
A CDK9 inhibitor having short target engagement would enable a reduction of Mcl-1 activity, resulting in apoptosis in cancer cells dependent on Mcl-1 for survival. We report the optimization of a series of amidopyridines (from compound 2), focusing o
Autor:
Graeme R. Robb, Lynsie Almeida, Rosemary A. Croft, Jian Huang, Haiyun Wang, Chungang Gu, Jane E. Moore, Steven L. Kazmirski, Michelle Lamb, Nancy Su, Timothy Pontz, Kurt Gordon Pike, Robert Casella, Hai-Jun Zhang, Xiaoyun Wu, Lakshmaiah Gingipalli, Derek Ogg, Barlaam Bernard Christophe, Janet Hawkins, Jeffrey W. Johannes, P. Ann Boriack-Sjodin, Allan Dishington, Yue Zhang, Stephanos Ioannidis, Tina Howard, Xiaolan Zheng, Tao Wang, Anil Patel, Jane L. Holmes, Thomas M. McGuire
Publikováno v:
ACS medicinal chemistry letters. 6(3)
The canonical Wnt pathway plays an important role in embryonic development, adult tissue homeostasis, and cancer. Germline mutations of several Wnt pathway components, such as Axin, APC, and ß-catenin, can lead to oncogenesis. Inhibition of the poly
Publikováno v:
Journal of Applied Polymer Science. 46:1369-1374
Splaying and curling of bristles is a very important performance characteristic of nylon toothbrushes. For this reason, analytical methods are needed that correlate fundamental physical–chemical properties with the eventural development of bristle
Autor:
Yair Lotan, Serge Benayoun, Pierre I. Karakiewicz, Frank Wians, K.-H. Felix Chun, Hans G. Boman, Michael Marberger, Craig D. Zippe, Shahrokh F. Shariat, Robert Casella, Hans Hedefin, Daniel J. Lewinshtein, Martin J. Friedrich, Hartwig Huland, Raina Rupesh, Paul Perrotte, Hideyuki Akaza, Arthur I. Sagalowsky, Ihor S. Sawczuk, Alberto Briganti, Sanaa Eissa, Claus G. Roehrborn, Gerson Lüdecke, Marta Sanchez-Carbayo, Naoto Miyanaga
Publikováno v:
Journal of Urology. 175:287-287