Zobrazeno 1 - 10
of 24
pro vyhledávání: '"Riviello Christopher"'
Publikováno v:
In Visual Journal of Emergency Medicine July 2024 36
Autor:
Andrew G. Cole, Douglas S. Auld, Riviello Christopher, Hema Desai, Hong Li, Heather A. Zanetakos, Fiona Thomson, J. Richard Morphy, Jiuqiao Zhao, Susan Elizabeth Napier, Michael Ohlmeyer, Katharine A. Goan, Koc-Kan Ho, Maria L. Webb, Jeffrey J. Letourneau
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 20:5394-5397
The discovery, synthesis, and preliminary structure–activity relationship (SAR) of a novel class of vasopressin V3 (V1b) receptor antagonists is described. Compound 1, identified by high throughput screening of a diverse, three million-member compo
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::af9cd65c56eed38d36dbec9326862276
https://doi.org/10.1016/j.bmcl.2010.07.118
https://doi.org/10.1016/j.bmcl.2010.07.118
Autor:
Celia Kingsbury, Irina Neagu, Ming You, Haengsoon Park, Tsung H. Lin, Koc-Kan Ho, Elizabeth Quadros, Maria L. Webb, Michael Ohlmeyer, Yuefei Shao, Matthew Sills, Jeffrey J. Letourneau, Andrew G. Cole, Yingchun Lu, Earl F. Kimble, Jorge Quintero, Riviello Christopher, Ray Anthony James, Bojing Wang, Vidyadhar M. Paradkar, Adolph Bohnstedt, Kenneth C. Appell, David J. Diller
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 19:6788-6792
A novel class of Janus tyrosine kinase 3 (JAK3) inhibitors based on a 2-benzimidazoylpurinone core structure is described. Through substitution of the benzimidazoyl moiety and optimization of the N-9 substituent of the purinone, compound 24 was ident
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::3dd21d26420d59e8a1c379ce66894ef1
https://doi.org/10.1016/j.bmcl.2009.09.080
https://doi.org/10.1016/j.bmcl.2009.09.080
Publikováno v:
Tetrahedron Letters. 48:1739-1743
A novel synthesis of 5-aryl-4-bromo-3-carboxyisoxazoles employing a [3+2] cycloaddition of a nitrile N-oxide with 2-aryl-1-bromoalkynes as the key step is described. The utility of these 5-aryl-4-bromo-3-carboxyisoxazoles in the solid-phase synthesis
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::2638a411ae8f0ea852ff1d0fbc4629a4
https://doi.org/10.1016/j.tetlet.2007.01.040
https://doi.org/10.1016/j.tetlet.2007.01.040
Autor:
Jingchun Yang, Robert Swanson, Maria L. Webb, Koc-Kan Ho, Olson John T, Lihong McAleer, Phillip M. Cowley, Jokiel Patrick, Darren Edwards, Michael Ohlmeyer, James R. Baker, Riviello Christopher, Nick Ward, Jeffrey J. Letourneau
Publikováno v:
Bioorganicmedicinal chemistry letters. 20(18)
The discovery, synthesis and preliminary structure-activity relationships (SARs) of a novel class of CB1 antagonists is described. Initial optimization of benzimidazole-based screening hit 4 led to the identification of 'inverted' indole-based lead c
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ce2b8e4693c7824e759fa9bc312f5738
https://pubmed.ncbi.nlm.nih.gov/20719511
https://pubmed.ncbi.nlm.nih.gov/20719511
Autor:
Letourneau, Jeffrey J., Riviello, Christopher M., Li, Hong, Cole, Andrew G., Ho, Koc-Kan, Zanetakos, Heather A., Desai, Hema, Zhao, Jiuqiao, Auld, Douglas S., Napier, Susan E., Thomson, Fiona J., Goan, Katharine A., Morphy, J. Richard, Ohlmeyer, Michael H.J., Webb, Maria L.
Publikováno v:
In Bioorganic & Medicinal Chemistry Letters 2010 20(18):5394-5397
Autor:
Letourneau, Jeffrey J., Jokiel, Patrick, Olson, John, Riviello, Christopher M., Ho, Koc-Kan, McAleer, Lihong, Yang, Jingchun, Swanson, Robert N., Baker, James, Cowley, Phillip, Edwards, Darren, Ward, Nick, Ohlmeyer, Michael H.J., Webb, Maria L.
Publikováno v:
In Bioorganic & Medicinal Chemistry Letters 2010 20(18):5449-5453
Autor:
Cole, Andrew G., Bohnstedt, Adolph C., Paradkar, Vidyadhar, Kingsbury, Celia, Quintero, Jorge G., Park, Haengsoon, Lu, Yingchun, You, Ming, Neagu, Irina, Diller, David J., Letourneau, Jeffrey J., Shao, Yuefei, James, Ray A., Riviello, Christopher M., Ho, Koc-Kan, Lin, Tsung H., Wang, Bojing, Appell, Kenneth C., Sills, Matthew, Quadros, Elizabeth, Kimble, Earl F., Ohlmeyer, Michael H.J., Webb, Maria L.
Publikováno v:
In Bioorganic & Medicinal Chemistry Letters 2009 19(23):6788-6792
Autor:
Megan B Thorn, Barbara Strohl, Robert A. Horlick, Roland E. Dolle, Bassam Damaj, Gonghua Pan, Nolan H. Sigal, Baldwin John J, Riviello Christopher, Adriane E. Schilling, V.Danial Fitzpatrick, Jorge Quintero, Ilana L. Stroke, Ming You, Maria L. Webb, Ohlmeyer Michael, Vidyadhar M. Paradkar
Publikováno v:
Immunopharmacology. 43(2-3)
Screening Pharmacopeia's encoded combinatorial libraries has led to the identification of potent, selective, competitive antagonists at the bradykinin Bl receptor. Libraries were screened using a displacement assay of [ 3 H]-des-Arg 10 -kallidir ([ 3
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7a1d19dda9301b4d7abb21754a6c0b41
https://pubmed.ncbi.nlm.nih.gov/10596850
https://pubmed.ncbi.nlm.nih.gov/10596850
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