Zobrazeno 1 - 4
of 4
pro vyhledávání: '"Richard Versace"'
Autor:
Stacy W. Remiszewski, Lidia C. Sambucetti, Kenneth W. Bair, John Bontempo, David Cesarz, Nagarajan Chandramouli, Ru Chen, Min Cheung, Susan Cornell-Kennon, Karl Dean, George Diamantidis, Dennis France, Michael A. Green, Kobporn Lulu Howell, Rina Kashi, Paul Kwon, Peter Lassota, Mary S. Martin, Yin Mou, Lawrence B. Perez, Sushil Sharma, Troy Smith, Eric Sorensen, Francis Taplin, Nancy Trogani, Richard Versace, Heather Walker, Susan Weltchek-Engler, Alexander Wood, Arthur Wu, Peter Atadja
Publikováno v:
Journal of Medicinal Chemistry. 46:4609-4624
A series of N-hydroxy-3-phenyl-2-propenamides were prepared as novel inhibitors of human histone deacetylase (HDAC). These compounds were potent enzyme inhibitors, having IC50s < 400 nM in a partially purified enzyme assay. However, potency in cell g
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::6e0206bc14fdb324b1acbdd17eeea9cc
https://doi.org/10.1021/jm030235w
https://doi.org/10.1021/jm030235w
Publikováno v:
Tetrahedron: Asymmetry. 7:2169-2172
HMQC correlation of diastereomeric salts obtained from complexes with quinine is described. The HMQC/quinine combination is a convenient and potentially general method for chiral purity determination. HMQC correlation of diastereomeric salts obtained
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::8f0592fc9310ae0a069585fb9c2a184c
https://doi.org/10.1016/0957-4166(96)00262-5
https://doi.org/10.1016/0957-4166(96)00262-5
Autor:
Roberto Mazzanti, Jan H.M. Schellens, Serena Marchetti, Olaf van Tellingen, Richard Versace, Dick Pluim, Monique van Eijndhoven, Roos L. Oostendorp, Alfred H. Schinkel, Jos H. Beijnen
Publikováno v:
Molecular cancer therapeutics. 6(12 Pt 1)
Lipophilic camptothecin derivatives are considered to have negligible affinity for breast cancer resistance protein (BCRP; ABCG2). Gimatecan, a new orally available 7-t-butoxyiminomethyl–substituted lipophilic camptothecin derivative, has been prev
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::637bf48dc3c04ff67d1e425312ab7d41
https://pubmed.ncbi.nlm.nih.gov/18089724
https://pubmed.ncbi.nlm.nih.gov/18089724
Autor:
Murugesan Gounder, Ahamed Nazar, Ahamed Saleem, Pooja Pungaliya, Diptee Kulkarni, Richard Versace
Publikováno v:
Investigational New Drugs; Jun2008, Vol. 26 Issue 3, p205-213, 9p, 6 Charts, 4 Graphs