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of 10
pro vyhledávání: '"Ranjeet Bairwa"'
Publikováno v:
Monatshefte für Chemie - Chemical Monthly. 143:461-465
A wide variety of carbonyl compounds can be transformed to their corresponding cyanohydrins in a single step using a dimethyl sulfoxide (DMSO)–water system in excellent yields (75–94%). The major advantages of this system are that the reaction co
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 20:6175-6178
Based on stereoelectronic feature analysis using density functional theory (DFT) at B3LYP/3-21∗G level, a series of 4-(5-nitrofuran-2-yl)prop-2-en-1-one derivatives with low LUMO energies (-0.10eV); concentrated over the nitro group, furan moiety a
Autor:
Ranjeet Bairwa, Mariam S. Degani
Publikováno v:
Synthetic Communications. 38:943-952
The facile, regiospecific, one‐pot synthesis of 2‐(3,5‐diaryl‐4,5‐dihydro‐1H‐pyrazol‐1‐yl)‐4,6‐diarylpyrimidines derivatives has been described, involving a [3+2] and [3+3] cyclocondensation between the α,β‐unsaturated keton
Autor:
Nilesh R. Tawari, Mariam S. Degani, Dhiman Sarkar, Mukti Kanta Ray, Arundhati C. Lele, Ranjeet Bairwa, Archana Raju, Seema Bag, M. G. R. Rajan, Laxman Nawale
Publikováno v:
Future medicinal chemistry. 7(8)
Background: A series of 2,4-diamino-s-triazines was designed, with potential for activity against Mycobacterium tuberculosis (Mtb) dihydrofolate reductase enzyme, on the basis of virtual screening results and structure-based drug design. Results: The
Autor:
Ranjeet Bairwa, Amruta Alate, Muktikant Ray, Swapnil Anam, Ramakrishna M. G. Rajan, Mariam S. Degani, Nilesh R. Tawari
Publikováno v:
Medicinal chemistry (Shariqah (United Arab Emirates)). 9(1)
Siderophores are small molecules produced by bacteria under iron-scarcity conditions faced by bacteria inside host. Sideophores bind iron with high affinity (Kd < 10-25 M) and are required for iron transport into the bacterial cell. Small molecules i
Publikováno v:
ChemInform. 43
A wide variety of carbonyl compounds can be transformed to their corresponding cyanohydrins in a single step and without any catalyst using DMSO/water as reaction medium.
Publikováno v:
ChemInform. 41
Novel substituted 2-hydrazino-pyrimidin-4(3H)-one derivatives were synthesized and examined for their antifolate activity against DHFR from Pneumocystis carinii (pc), Toxoplasma gondii (tg), Mycobacterium avium (ma), and rat liver (rl). A novel, simp
Autor:
Manoj D. Kakwani, Nilesh R. Tawari, Jaya Lalchandani, M. K. Ray, M. G. R. Rajan, Mariam S. Degani, Ranjeet Bairwa
Publikováno v:
ChemInform. 41
In an attempt to identify potential new agents active against tuberculosis, 20 novel phenylacrylamide derivatives incorporating cinnamic acids and guanylhydrazones were synthesized using microwave assisted synthesis. Activity of the synthesized compo
Publikováno v:
Journal of Heterocyclic Chemistry.
Novel substituted 2-hydrazino-pyrimidin-4(3H)-one derivatives were synthesized and examined for their antifolate activity against DHFR from Pneumocystis carinii (pc), Toxoplasma gondii (tg), Mycobacterium avium (ma), and rat liver (rl). A novel, simp
Autor:
Mariam S. Degani, Ranjeet Bairwa
Publikováno v:
ChemInform. 39
The facile, regiospecific, one‐pot synthesis of 2‐(3,5‐diaryl‐4,5‐dihydro‐1H‐pyrazol‐1‐yl)‐4,6‐diarylpyrimidines derivatives has been described, involving a [3+2] and [3+3] cyclocondensation between the α,β‐unsaturated keton