Zobrazeno 1 - 10
of 33
pro vyhledávání: '"Ranjan C. Khunt"'
Miscellaneous Passerini Reaction for α-Acyloxy Carboxamide: Synthesis and Process Optimization Study
Publikováno v:
Letters in Organic Chemistry. 19:326-332
An accelerating effect of “Phase Transfer Catalyst” as additive was exposed for the Passerini three-component reactions and the influence on the reaction rate was studied concerning direct involvement of reactant molecules. The most flexible reac
Autor:
Khushal M. Kapadiya, Kishor M. Kavadia, Vijay M. Khedkar, Piyush V. Dholaria, Amita J. Jivani, Ranjan C. Khunt
Publikováno v:
Heterocyclic Communications. 28:75-83
The purpose of this study was to prepare various derivatives of 4-amino-2-(3-fluoro-5-(trifluoromethyl)phenyl)-6-arylpyrimidine-5-carbonitrile (6a–6h) using a three-step procedure. The derivatives were screened in vitro for activity against Mycobac
Publikováno v:
Russian Journal of Organic Chemistry. 57:801-808
Two new pharmacologically active series of N-alkyne-substituted indole–thiazoles and C-alkyne-substituted benzylidene–thiazoles were synthesized by a two-step procedure involving initial reactions of thiosemicarbazide with, respectively, [1-(prop
Publikováno v:
Folia Medica, Vol 63, Iss 2, Pp 213-220 (2021)
Introduction: Due to the vast medicinal importance of purine nucleoside, a hybrid molecule of triazole with purine ring mightexplode a lead molecule in the pharma sector and based on the last decade’s studies suggested that the nitrogen-rich molecu
Publikováno v:
Asian Journal of Organic & Medicinal Chemistry. 6:92-101
Thiazole derivatives are potential candidates for drug development. They can be efficiently synthesized and are extremely active against several diseases, including antimicrobial screening. A series of 2-(2-(3-methoxy-4-(prop-2-yn-1-yloxy)benzylidene
Publikováno v:
Anti-Infective Agents. 18:135-143
Background: A 3D-QSAR study based on CoMFA and CoMSIA was performed on these pyrazole-pyrimidine derivatives to correlate their chemical structures with the observed activity against M. tuberculosis. Objective: The current research aimed to synthesiz
Autor:
Anamik Shah, Ranjan C. Khunt, Vijay M. Khedkar, Vijay D. Chodvadiya, Kaushik Pambhar, Ashish Dhamsaniya
Publikováno v:
Asian Journal of Organic & Medicinal Chemistry. 5:68-76
Herein, we report the synthesis methodology and anticancer evaluation of 15 compounds using copper(I)- catalyzed azide alkyne cycloaddition (CuAAC) to develop a library of saccharin-1,2,3-triazole hybrid molecules. All library compounds showed intera
The novel series of phthalimide-1H-1,2,3-triazole derivatives (6a–o) was created by combining various azide derivatives with an N-methylene bond using click chemistry. N-alkylation procedures using a base catalyst were used to make the initial alky
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::5ed514b11104af5d47ad7cbe9723b7d8
Thiazole is a well-established scaffold due to its wide range of therapeutic activities. Moreover, the chromane nucleus is also associated with various biological activities such as antibacterial, anticancer, anti-inflammatory, and anti-HIV. We have
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ce18771b932dc4a03a253a6a03323911
Autor:
Jagriti Behal, Ranjan C. Khunt
Introduction: In the preceding few years, nanotechnology attracts worldwide attention because it offers a huge range of uses and economical potential (1). Therefore, the synthesis of nanomaterials is an important area of research. The properties of i
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::667b9ae5d052f9e938bb2f9cca6e1830