Zobrazeno 1 - 10
of 26
pro vyhledávání: '"Ramesh S. Yamgar"'
Autor:
Mustapha C. Mandewale, Udaysinha C. Patil, Supriya V. Shedge, Uttam R. Dappadwad, Ramesh S. Yamgar
Publikováno v:
Beni-Suef University Journal of Basic and Applied Sciences, Vol 6, Iss 4, Pp 354-361 (2017)
Tuberculosis (TB) and Cancer remains a global public health problem in recent years. There is an urgent need for the screening of new bioactive molecules with new targets and with a different mechanism of action. Among heterocyclic compounds, compoun
Externí odkaz:
https://doaj.org/article/9e2fe91766fb4b4aae5b5581611b051e
Autor:
Ramesh S. Yamgar, Y. Nivid, Satish Nalawade, Mustapha Mandewale, R. G. Atram, Sudhir S. Sawant
Publikováno v:
Bioinorganic Chemistry and Applications, Vol 2014 (2014)
The synthesis and antimicrobial activity of novel Zn(II) metal complexes derived from three novel heterocyclic Schiff base ligands 8-[(Z)-{[3-(N-methylamino)propyl]imino}methyl]-7-hydroxy-4-methyl-2H-chromen-2-one, 2-[(E)-{[4-(1H-1,2,4-triazol-1-ylme
Externí odkaz:
https://doaj.org/article/0d5373cc4d274f6ab8cb449b74a9aad8
Publikováno v:
Current Computer-Aided Drug Design. 18:247-257
Background: Hydrazide-hydrazone based compounds are reported for their wider pharmacological potentials. Methods: In present work, we synthesized 10 new Schiff based-aryl-carbohydrazide (3a-3e) and (4a-4e), analogues and characterized further using s
Publikováno v:
Current Computer-Aided Drug Design. 17:493-503
Background: For the past several decades, the presence of tuberculosis (TB) is being remarked as the most common infectious disease leading to mortality. Objective: Hydrazone containing azometine group (-NHN=CH-) compounds have been reported for a br
Autor:
Bapu R. Thorat, Suraj N. Mali, Vijay J. Desale, Ramesh S. Yamgar, Swapnali V. Dharanguttikar, Vyankatesh R. Dharanguttikar, Samir Chtita, Mozaniel Oliveira, Jorddy Neves Cruz
Publikováno v:
Current computer-aided drug design.
Background: Hydrazide-hydrazone derivatives have shown diverse biological activities, such as antitubercular (anti-TB), antibacterial, antifungal, anticancer, anti-inflammatory, antiviral, and antiprotozoal actions. Objectives: Hydrazide–hydrazones
Publikováno v:
Current Computer-Aided Drug Design. 16:802-813
Background: Antimicrobial resistance is a major global health problem, which is being rapidly deteriorating the quality of human health. Series of substituted N-(benzo[d]thiazol-2-yl)-2- (4-(6-fluorobenzo[d]isoxazol-3-yl) piperidin-1-yl)acetamide (3a
Publikováno v:
JOURNAL OF SCIENTIFIC RESEARCH. 65:66-71
Publikováno v:
Recent advances in anti-infective drug discovery.
Background: The human respiratory syncytial virus (RSV) is responsible for causing upper and lower respiratory tract infections in young children. RSV Fusion (F) protein is a surface glycoprotein that facilitates virus entry into host cells. Thus, ne
Autor:
Suraj N. Mali, Rajesh S. Kenny, Bhagwat S. Jadhav, Mustapha Mandewale, Hemchandra K. Chaudhari, Ramesh S. Yamgar
Publikováno v:
Current Computer-Aided Drug Design. 16:511-522
Background: A series of new six thiazolyl-2-amine-based Schiff base derivatives (4a-4f) were synthesized by a sequential multistep reaction starting with Salicylaldehyde. Methods: All the Schiff base derivatives were screened in-vitro for their antib
Autor:
Suraj N. Mali, Devidas G. Anuse, Hemchandra K. Chaudhari, Ramesh S. Yamgar, Sudhir Sawant, Bapu R. Thorat
Publikováno v:
Current Computer-Aided Drug Design. 16:530-540
Background: Benzothiazoles are reported to have bioorganic and pharmaceutical chemistry applications. Introduction: A series of substituted N-bromoamido-2-aminobenzothiazoles was synthesized from substituted anilines via 2-aminobenzothiazoles and it