Zobrazeno 1 - 6
of 6
pro vyhledávání: '"Radim Horák"'
Publikováno v:
Beilstein Journal of Organic Chemistry, Vol 11, Iss 1, Pp 884-892 (2015)
2-Aroylmethylidene-1,2,3,4-tetrahydroquinolines with the appropriate substituents can be suitable precursors for the synthesis of alkaloids from Galipea officinalis (cuspareine, galipeine, galipinine, angustureine). However, only two, rather low-yiel
Externí odkaz:
https://doaj.org/article/77b4c9c878db485491167a8cfa131ab5
Autor:
Lubomir Kvapil, Kamil Kořistek, Radim Horák, Pavel Hradil, Petr Funk, Martin Grepl, Veronika Šamšulová, Miroslav Soural, Ludmila Slaninová
Publikováno v:
Journal of Heterocyclic Chemistry. 57:1605-1615
Publikováno v:
Synlett. 31:911-915
In this work, we report the simple synthesis of furo[3,2-b]quinolin-4(1H)-ones from readily available 4-ethynyl-[1,3]dioxolo[4,5-c]quinolone as the key starting material. After Sonogashira (hetero)arylation, formation of the furoquinoline scaffold wa
Publikováno v:
Journal of Molecular Structure. 1177:16-25
A synthetic approach to novel 2-(1-glycosyl-1,2,3-triazol-4-yl)-3-hydroxyquinolone conjugates has been developed. The methodology involves preparation of a suitable quinoline intermediate and its subsequent conjugation with various acylated glycosyl
Autor:
Miroslav Urbasek, Pavel Hradil, Kamil Motyka, Miroslav Soural, Ludmila Slaninová, Martin Grepl, Lubomir Kvapil, Radim Horák, Kamil Kořistek
Publikováno v:
Tetrahedron. 74:366-374
2-Alkenyl-3-hydroxyquinolin-4(1H)-ones were prepared by the rearrangement of anthranilic acid esters synthesized by two alternative methods. The prepared derivatives were screened for their antimicrobial activities against representative Gram-positiv
Autor:
Tomáš Klunda, Alžzbeta Čížzová, Eva Machová, Slavomír Bystrický, Monika Poláková, Radim Horák
Publikováno v:
Chemical Papers. 70
Candida infections are becoming increasingly prevalent and many clinical isolates are resistant to common azole derivatives treatment. Accordingly, the capacity of a series of 19 alkyl glycosides, mainly mannosides and glucosides but also a cellobios