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Cocaine receptors labeled by [3H]2 beta-carbomethoxy-3 beta-(4-fluorophenyl)tropane

Autor: Bk, Madras, Rd, Spealman, Ma, Fahey, John Neumeyer, Jk, Saha, Ra, Milius

Publikováno v: Europe PubMed Central

The potent cocaine analog 2 beta-carbomethoxy-3 beta-(4-fluorophenyl)-tropane (CFT, also designated WIN 35,428) was tritiated and evaluated as a molecular probe for cocaine receptors in caudate putamen membranes of cynomolgus monkeys. Kinetic, satura

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=pmid_dedup__::20dadb36d54d5adedc53eee2b6850980
https://pubmed.ncbi.nlm.nih.gov/2811854

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Akademický článek

N-substituted analogs of 2 beta-carbomethoxy-3 beta- (4'-iodophenyl)tropane (beta-CIT) with selective affinity to dopamine or serotonin transporters in rat forebrain.

Autor: Neumeyer JL; Research Biochemicals International (RBI), Natick, Massachusetts 01760, USA., Tamagnan G, Wang S, Gao Y, Milius RA, Kula NS, Baldessarini RJ

Publikováno v: Journal of medicinal chemistry [J Med Chem] 1996 Jan 19; Vol. 39 (2), pp. 543-8.

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Akademický článek

[O-methyl-11C]beta-CIT-FP, a potential radioligand for quantitation of the dopamine transporter: preparation, autoradiography, metabolite studies, and positron emission tomography examinations.

Autor: Lundkvist C; Karolinska Institutet, Department of Clinical Neuroscience, Stockholm, Sweden., Halldin C, Swahn CG, Hall H, Karlsson P, Nakashima Y, Wang S, Milius RA, Neumeyer JL, Farde L

Publikováno v: Nuclear medicine and biology [Nucl Med Biol] 1995 Oct; Vol. 22 (7), pp. 905-13.

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Akademický článek

Regional brain uptake and pharmacokinetics of [123I]N-omega-fluoroalkyl-2 beta-carboxy-3 beta-(4-iodophenyl)nortropane esters in baboons.

Autor: Baldwin RM; Department of Psychiatry, Yale University School of Medicine, West Haven, CT, USA., Zea-Ponce Y, al-Tikriti MS, Zoghbi SS, Seibyl JP, Charney DS, Hoffer PB, Wang S, Milius RA, Neumeyer JL, et. al.

Publikováno v: Nuclear medicine and biology [Nucl Med Biol] 1995 Feb; Vol. 22 (2), pp. 211-9.

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Akademický článek

N-omega-fluoroalkyl analogs of (1R)-2 beta-carbomethoxy-3 beta-(4-iodophenyl)-tropane (beta-CIT): radiotracers for positron emission tomography and single photon emission computed tomography imaging of dopamine transporters.

Autor: Neumeyer JL; Research Biochemicals International, Natick, Massachusetts 01760., Wang S, Gao Y, Milius RA, Kula NS, Campbell A, Baldessarini RJ, Zea-Ponce Y, Baldwin RM, Innis RB

Publikováno v: Journal of medicinal chemistry [J Med Chem] 1994 May 27; Vol. 37 (11), pp. 1558-61.

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Akademický článek

Evaluation of the monoamine uptake site ligand [123I]methyl 3 beta-(4-iodophenyl)-tropane-2 beta-carboxylate ([123I]beta-CIT) in non-human primates: pharmacokinetics, biodistribution and SPECT brain imaging coregistered with MRI.

Autor: Baldwin RM; Department of Psychiatry, Yale University School of Medicine, West Haven, CT 06516., Zea-Ponce Y, Zoghbi SS, Laurelle M, al-Tikriti MS, Sybirska EH, Malison RT, Neumeyer JL, Milius RA, Wang S, et. al.

Publikováno v: Nuclear medicine and biology [Nucl Med Biol] 1993 Jul; Vol. 20 (5), pp. 597-606.

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Akademický článek

[123I]-2 beta-carbomethoxy-3 beta-(4-iodophenyl)tropane: high-affinity SPECT radiotracer of monoamine reuptake sites in brain.

Autor: Neumeyer JL; Research Biochemicals Inc., Natick, Massachusetts 01760., Wang SY, Milius RA, Baldwin RM, Zea-Ponce Y, Hoffer PB, Sybirska E, al-Tikriti M, Charney DS, Malison RT, et. al.

Publikováno v: Journal of medicinal chemistry [J Med Chem] 1991 Oct; Vol. 34 (10), pp. 3144-6.

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Akademický článek

Synthesis and receptor binding of N-substituted tropane derivatives. High-affinity ligands for the cocaine receptor.

Autor: Milius RA; Research Biochemicals Inc., Natick, Massachusetts 01760., Saha JK, Madras BK, Neumeyer JL

Publikováno v: Journal of medicinal chemistry [J Med Chem] 1991 May; Vol. 34 (5), pp. 1728-31.

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Akademický článek

N-modified fluorophenyltropane analogs of cocaine with high affinity for cocaine receptors.

Autor: Madras BK; Harvard Medical School, New England Regional Primate Research Center, Southborough, MA 01772., Kamien JB, Fahey MA, Canfield DR, Milius RA, Saha JK, Neumeyer JL, Spealman RD

Publikováno v: Pharmacology, biochemistry, and behavior [Pharmacol Biochem Behav] 1990 Apr; Vol. 35 (4), pp. 949-53.

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Akademický článek

Estrogen receptor-mediated cytotoxicity using iodine-125.

Autor: Bloomer WD, McLaughlin WH, Milius RA, Weichselbaum RR, Adelstein SJ

Publikováno v: Journal of cellular biochemistry [J Cell Biochem] 1983; Vol. 21 (1), pp. 39-45.

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