Zobrazeno 1 - 10
of 53
pro vyhledávání: '"R. Jasztold‐Howorko"'
Publikováno v:
Letters in Drug Design & Discovery. 3:192-199
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::97c867890e1418f8356d798ac4a8c4ea
https://doi.org/10.2174/157018006776286961
https://doi.org/10.2174/157018006776286961
Publikováno v:
Acta Crystallographica Section C Crystal Structure Communications. 52:2106-2111
2-Chloro-5-p-toluoylamino-N-p-tolyl-4-p-tolylamino-6-pyrimidinecarboxamide, C 27 H 24 ClN 5 O 2 , crystallizes in two forms: orthorhombic (I) and triclinic (Ia). The orthorhombic form is almost isomorphous with the crystals of N-p-tolyl-5-benzoylamin
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::c04c75742687a29e250b795023cc19aa
https://doi.org/10.1107/s0108270196005616
https://doi.org/10.1107/s0108270196005616
Autor:
Alain Pierré, C. Landras, Ghanem Atassi, Laurence Kraus-Berthier, Yves Rolland, R. Jasztold‐Howorko, Stéphane Léonce, Claude Guillonneau, Emile Bisagni, Nicolas Guilbaud
Publikováno v:
Chemical and Pharmaceutical Bulletin. 44:2169-2172
Starting from 2-(6-methoxy-1-methylcarbazol-2-yl)ethylamine and diethyl-2, 6-pyridine dicarboxylate, the title compounds were obtained through five or six steps. The new compounds retained significant cytotoxicity towards various tumor cell lines, bu
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::03727c92430d4dd60688ed895c1ea40a
https://doi.org/10.1248/cpb.44.2169
https://doi.org/10.1248/cpb.44.2169
Autor:
Nicolas Guilbaud, Prost Jf, Laurence Kraus-Berthier, Stéphane Léonce, Alain Pierre, Ghanem Atassi, R. Jasztold‐Howorko, Yves Rolland, C. Landras, Emile Bisagni
Publikováno v:
ChemInform. 25
Starting from 2-(2-aminoethyl)-6-methoxy-1-methylcarbazole, ethyl 9-methoxy-5-methyl-6H-pyrido[4,3-b]carbazole-1-carboxylate was obtained through a three-step sequence. This compound and its 6-methyl derivative react with (dialkylamino)alkylamines to
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::5391db19edb19ee58e15198488eac9c0
https://doi.org/10.1002/chin.199452170
https://doi.org/10.1002/chin.199452170
Autor:
Claude Guillonneau, Laurence Kraus-Berthier, R. Jasztold‐Howorko, Emile Bisagni, C. Landras, Alain Pierré, Ghanem Atassi, Yves Rolland, Stéphane Léonce, Nicolas Guilbaud
Publikováno v:
ChemInform. 28
Starting from 2-(6-methoxy-1-methylcarbazol-2-yl)ethylamine and diethyl-2, 6-pyridine dicarboxylate, the title compounds were obtained through five or six steps. The new compounds retained significant cytotoxicity towards various tumor cell lines, bu
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::1e16117b4d1fad56ed2267244ac9ed5b
https://doi.org/10.1002/chin.199721158
https://doi.org/10.1002/chin.199721158
Autor:
R, Jasztold-Howorko, Z, Machoń, M, Wilimowski, W, Wojewódzki, J, Barczyńska, L, Kedzierska, K, Orzechowska-Juzwenko, E, Duś, M, Rutkowska, A, Szelag
Publikováno v:
Polish journal of pharmacology. 47(5)
2,4-Disubstituted 5-amino-6-pyrimidinecarboxylic acid derivatives 5-20 were synthesized and evaluated for their pharmacological activity. Compounds 11-14, 17-19 showed antiaggressive effect, compounds 5, 8, 9, 11, 12 and 19 displayed antiserotonin ac
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=pmid_dedup__::165bf8f2eaa2754ae1fd5e3c9e851890
https://pubmed.ncbi.nlm.nih.gov/8868136
https://pubmed.ncbi.nlm.nih.gov/8868136
Autor:
R. Jasztold‐Howorko, Prost Jf, Yves Rolland, Emile Bisagni, Stéphane Léonce, Alain Pierre, C. Landras, Laurence Kraus-Berthier, Ghanem Atassi, Nicolas Guilbaud
Publikováno v:
Journal of medicinal chemistry. 37(15)
Starting from 2-(2-aminoethyl)-6-methoxy-1-methylcarbazole, ethyl 9-methoxy-5-methyl-6H-pyrido[4,3-b]carbazole-1-carboxylate was obtained through a three-step sequence. This compound and its 6-methyl derivative react with (dialkylamino)alkylamines to
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::e8fc91e9ed7b1eb2dd4dce6085b51601
https://pubmed.ncbi.nlm.nih.gov/8057291
https://pubmed.ncbi.nlm.nih.gov/8057291
Publikováno v:
ChemInform. 21
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::fe790409048720d01e8ace942805c39c
https://doi.org/10.1002/chin.199012216
https://doi.org/10.1002/chin.199012216
Akademický článek
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Autor:
Z, Machoń, R, Jasztold-Howorko
Publikováno v:
Polish journal of pharmacology and pharmacy. 28(1)
5-Benzoyloaminoorotic acid in a reaction with POCl3 forms 2,4-dichloro-5-benzylo-aminopyrimidine-6-carboxylic acid lactam 3, which heated with aliphatic and aromatic amines gives corresponding amides 6-11. These compounds don't show any antiinflammat
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=pmid________::f543005f87ca1540162d680243f051a3
https://pubmed.ncbi.nlm.nih.gov/1264859
https://pubmed.ncbi.nlm.nih.gov/1264859