Zobrazeno 1 - 10 of 11 pro vyhledávání: '"R. C. MAKOFSKE"'
1
Synthesis of a potent enkephalin analog, Tyr-D-Thr-Gly-Phe-Δ3Pro-NH2, and some of its biological activities
Autor: Chryssa Tzougraki, Wallace M. Dairman, Johannes Meienhofer, Lislot Aeppli, R. C. Makofske
Publikováno v: International Journal of Peptide and Protein Research. 28:370-378
The enkephalin analog, H-Tyr-D-Thr-Gly-Phe-delta 3 Pro-NH2 X HCl (VI) ([D-Thr2, delta 3 Pro5]-enkephalinamide), has been synthesized by conventional methods in solution and purified to homogeneity by reversed phase HPLC. The analog is a potent analge
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::e07f71f27cbf4f8bf5e140340e64ce26
https://doi.org/10.1111/j.1399-3011.1986.tb03268.x
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2
Chimeric enkephalin-cystatins: opioid binding and structure-activity relationships of inhibitory domains
Autor: N, Marks, M J, Berg, R C, Makofske, J, Swistok, E J, Simon, D, Ofri, K, Del Compare, W, Danho
Publikováno v: Peptide research. 5(4)
A chimeric inhibitor of cysteine proteinases, YGGFLQVVAGK.amide, was synthesized for use in examining SAR of its cystatin and opioid domains. Analogs were prepared by solid-phase syntheses and evaluated for inhibition of rat brain cathepsin L (E.C. 3
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=pmid________::f1f919c6043a523f923e36c6e00cfb1e
https://pubmed.ncbi.nlm.nih.gov/1330108
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3
Synthesis and biological activity of novel, potent and long-acting analogs of AC-CCK-7 with high affinity for peripheral (type A) receptors
Autor: W, Danho, R C, Makofske, J, Swistok, J, Michalewsky, T, Gabriel, N, Marks, M J, Berg, L, Baird, V, Geiler, G, Mackie
Publikováno v: Peptide research. 4(2)
Analogs of cholecystokinin (CCK-7) in which the N-terminal Tyr(SO3H) was acetylated, Asp6 replaced with Thr(SO3H) and Phe7 replaced with N-methyl-Phe were prepared by solid-phase peptide synthesis and evaluated for their receptor-binding activity and
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=pmid________::7f4151144e3e883febe0bcc8a208d0de
https://pubmed.ncbi.nlm.nih.gov/1815779
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5
Solid phase synthesis without repetitive acidolysis. Preparation of leucyl-alanyl-glycyl-valine using 9-fluorenylmethyloxycarbonylamino acids
Autor: J, Meienhofer, M, Waki, E P, Heimer, T J, Lambros, R C, Makofske, C D, Chang
Publikováno v: International journal of peptide and protein research. 13(1)
The utility of repetitive nonhydrolytic base cleavage of alpha-amino protective groups in solid phase peptide synthesis is shown by a preparation of the model tetrapeptide leucyl-alanyl-glycyl-valine on a p-benzyloxybenzyl ester polystyrene--1% divin
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=pmid________::6d10184eb890205f79257946158c7c06
https://pubmed.ncbi.nlm.nih.gov/422322
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7
ChemInform Abstract: Synthesis of a Potent Enkephalin Analog, Tyr-D-Thr-Gly-Phe-δ3Pro-NH2, and Some of Its Biological Activities
Autor: Wallace M. Dairman, Johannes Meienhofer, Lislot Aeppli, R. C. Makofske, Chryssa Tzougraki
Publikováno v: ChemInform. 18
The enkephalin analog, H-Tyr-D-Thr-Gly-Phe-delta 3 Pro-NH2 X HCl (VI) ([D-Thr2, delta 3 Pro5]-enkephalinamide), has been synthesized by conventional methods in solution and purified to homogeneity by reversed phase HPLC. The analog is a potent analge
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::02da3ac9a5235cd366e7a79e1400125c
https://doi.org/10.1002/chin.198712332
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