Zobrazeno 1 - 6
of 6
pro vyhledávání: '"R. C. Haaseth"'
Publikováno v:
The Journal of pharmacology and experimental therapeutics. 275(3)
Antinociceptive effects of systemically or locally administered opioid mu, kappa and delta agonists were evaluated in a rat model of visceral pain. Resiniferatoxin (RTX, 3 nmol), a capsaicin-like mutant, produced abdominally directed grooming behavio
Autor:
Hitesh Shroff, Louis A. Carpino, Salvatore A. Triolo, R. C. Haaseth, Steven A. Kates, C. A. Minor, Ayman El-Faham, Fernando Albericio
Publikováno v:
Peptides 1994 ISBN: 9789072199218
Peptides 1994
Peptides 1994
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::1038127bfbf7569c85b13e3958dc079a
https://doi.org/10.1007/978-94-011-1468-4_106
https://doi.org/10.1007/978-94-011-1468-4_106
Autor:
L, Fang, R J, Knapp, R, Horvath, T O, Matsunaga, R C, Haaseth, V J, Hruby, F, Porreca, H I, Yamamura
Publikováno v:
The Journal of pharmacology and experimental therapeutics. 268(2)
Naltrindole (NTI) is a potent and selective nonpeptide delta opioid receptor antagonist. This study reports on the binding characteristics of [3H]NTI (specific activity = 30.5 Ci/mmole) for mouse brain and vas deferens (MVD) tissues. In brain, [3H]NT
Autor:
S J, Weber, T J, Abbruscato, E A, Brownson, A W, Lipkowski, R, Polt, A, Misicka, R C, Haaseth, H, Bartosz, V J, Hruby, T P, Davis
Publikováno v:
The Journal of pharmacology and experimental therapeutics. 266(3)
Confluent monolayers of primary and continuous passaged cultures of bovine brain microvessel endothelial cells (BMEC) have been suggested to model the blood-brain barrier (BBB). Increased lipophilicity has been previously suggested to increase BBB pe
Publikováno v:
The Journal of pharmacology and experimental therapeutics. 266(2)
In these studies, the antagonistic actions of (-)-1-Cyclopentyl-5-(1,2,3,4,5,-hexahydro-8-hydroxy-3,6,11-trimethyl-2,6 -methano-3-benzazocin-11-yl)-3-pentanone methanesulfonate (quadazocine) were evaluated against the kappa-receptor-mediated antinoci
Autor:
P J, Horan, K D, Wild, A, Misicka, A, Lipkowski, R C, Haaseth, V J, Hruby, S J, Weber, T P, Davis, H I, Yamamura, F, Porreca
Publikováno v:
The Journal of pharmacology and experimental therapeutics. 265(2)
Pharmacological evidence has suggested the presence of two supraspinal opioid delta receptor subtypes in the mouse, termed delta-1 and delta-2. [D-Pen2,D-Pen5]enkephalin (DPDPE) is thought to be primarily an agonist at the opioid delta-1 subtype, whe