Zobrazeno 1 - 10
of 33
pro vyhledávání: '"R G, Ball"'
Autor:
P D, Williams, P S, Anderson, R G, Ball, M G, Bock, L, Carroll, S H, Chiu, B V, Clineschmidt, J C, Culberson, J M, Erb, B E, Evans
Publikováno v:
Journal of Medicinal Chemistry. 37:565-571
Modifications to the previously reported spiroindenylpiperidine camphor-sulfonamide oxytocin (OT) antagonist L-366,509 have produced a new series of o-tolylpiperazine (TP) camphor-sulfonamides. A number of analogues in the TP series that incorporate
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::cbee35be16d415185dfe2956648b8b43
https://doi.org/10.1021/jm00031a004
https://doi.org/10.1021/jm00031a004
Publikováno v:
ChemInform. 22
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::f65ccf6a468c17a26172461821ea56ca
https://doi.org/10.1002/chin.199146172
https://doi.org/10.1002/chin.199146172
Autor:
K. Cheng, M. H. Fisher, R. G. Ball, B. Butler, R. G. Smith, M. J. Jun. Wyvratt, W. W.-S. Chan, J. M. Pisano, K. Prendergast, W. R. Schoen
Publikováno v:
ChemInform. 25
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::bb708ab4c43e9528d6988d82e3e5823e
https://doi.org/10.1002/chin.199434184
https://doi.org/10.1002/chin.199434184
Autor:
A E, Weber, M G, Steiner, P A, Krieter, A E, Colletti, J R, Tata, T A, Halgren, R G, Ball, J J, Doyle, T W, Schorn, R A, Stearns
Publikováno v:
Journal of Medicinal Chemistry. 35:3755-3773
Replacing one amide bond in macrocyclic renin inhibitors of the general structure 1 and 2 with an ester linkage gave glutamate-derived inhibitors 3 and serine-derived inhibitors 4. While this oxygen-for-nitrogen exchange had little effect on potency
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ef15bd203b00d1c5841faf09f5e4fbfc
https://doi.org/10.1021/jm00099a004
https://doi.org/10.1021/jm00099a004
Publikováno v:
Journal of the American Chemical Society. 123(46)
The stereospecific total synthesis of (+/-)-thielocin A1beta has been achieved from the common intermediate ethyl 5-formyl-2,4-dihydroxy-3,6-dimethyl benzoate (8). The racemic synthesis was achieved based on the key reaction of a 4-methyl-3,4-dihydro
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=pmid________::6833738acdd8f9b0bd8d3a40bb8a1e93
https://pubmed.ncbi.nlm.nih.gov/11707114
https://pubmed.ncbi.nlm.nih.gov/11707114
Publikováno v:
Journal of pharmaceutical sciences. 89(10)
The crystal structures of two enantiotropic polymorphs of the aza-steroid finasteride (N-(1-1-di-methylethyl)-3-oxo-4-aza-5 alpha-and rost-1-ene-17 beta-carboxam ide ) have been determined. The solid-state nuclear magnetic resonance spectra, infrared
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=pmid________::732e649930035c610330fbc867fb4b6f
https://pubmed.ncbi.nlm.nih.gov/10980502
https://pubmed.ncbi.nlm.nih.gov/10980502
Publikováno v:
European journal of biochemistry. 259(1-2)
The crystal structure of the human B blood group related trisaccharide alpha-L-Fucp-(1--2)-[alpha-D-Galp]-(1--3)-beta-D-Galp-OCH3 (1) has been determined. The solution structure of 1 was studied by two-dimensional NMR techniques at 600 MHz in D2O sol
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=pmid________::a4f247975dc198a70083652debc4e342
https://pubmed.ncbi.nlm.nih.gov/9914506
https://pubmed.ncbi.nlm.nih.gov/9914506
Publikováno v:
Acta Crystallographica Section C Crystal Structure Communications. 46:2491-2493
C 23 H 34 N 2 O 2 cristallise dans P2 1 /c avec a=11,0578, b=23,740, c=8,8991 A, β=111,117 o , Z=4; affinement jusqu'a R=0,059. Les longueurs et les angles de liaison a l'interieur de la molecule sont normaux. La longueur etroite de la liaison hydro
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::23a3575f04f6b3924b7b839e86f493fd
https://doi.org/10.1107/s0108270190003833
https://doi.org/10.1107/s0108270190003833
Publikováno v:
Acta Crystallographica Section C Crystal Structure Communications. 54:1493-1494
In the title triaryloxazolone derivative, C 24 H 18 ClNO 6 S, the three phenyl rings are oriented in a propeller-like fashion around the central oxazolone ring, with dihedral angles of 55.7 (1) (acetoxyphenyl), 56.4 (1) (methylsulfonylphenyl) and 25.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::115f9e726cff896ecb5427c93a323199
https://doi.org/10.1107/s0108270198003928
https://doi.org/10.1107/s0108270198003928
Publikováno v:
Journal of the American Chemical Society. 107:7669-7679
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::dd611168610f0f02e618cb3fcf79308f
https://doi.org/10.1021/ja00311a074
https://doi.org/10.1021/ja00311a074