Zobrazeno 1 - 2
of 2
pro vyhledávání: '"Qing-Yuan Lan"'
Autor:
Wang Shuxian, Yanle Zhi, Guo Xiaoxing, Cai Jiongheng, Zhang Liang, Shuai Lu, Yatian Huang, Hao Heng, Qin Tianren, Hongmei Li, Xiang Li, Wang Zhijie, Qing-Yuan Lan, Tao Lu, Yadong Chen
Publikováno v:
European Journal of Medicinal Chemistry. 176:248-267
FLT3 mutation is among the most common genetic mutations in acute myeloid leukemia (AML), which is also related with poor overall survival and refractory in AML patients. Recently, FLT3 inhibitors have been approved for AML therapy. Herein, a series
Autor:
Yanle Zhi, Qing-Yuan Lan, Tao Lu, Tian Jieyi, Yadong Chen, Lu Shuai, Guo Xiaoxing, Haichun Liu, Hao Heng
Publikováno v:
Recent Patents on Anti-Cancer Drug Discovery. 12
Background FLT3 is a member of receptor tyrosine kinase III family, mainly expressed in hematopoietic cells. The aberrant expression and function of FLT3 are strongly related to leukemia, especially acute myeloid leukemia. Its varieties of amino-acid