Zobrazeno 1 - 10
of 21
pro vyhledávání: '"Priya Dayananth"'
Autor:
Mihirbaran Mandal, Li Xiao, Weidong Pan, Giovanna Scapin, Guoqing Li, Haiqun Tang, Shu-Wei Yang, Jianping Pan, Yuriko Root, Reynalda Keh de Jesus, Christine Yang, Winnie Prosise, Priya Dayananth, Asra Mirza, Alex G. Therien, Katherine Young, Amy Flattery, Charles Garlisi, Rumin Zhang, Donald Chu, Payal Sheth, Inhou Chu, Jin Wu, Carrie Markgraf, Hai-Young Kim, Ronald Painter, Todd W. Mayhood, Edward DiNunzio, Daniel F. Wyss, Alexei V. Buevich, Thierry Fischmann, Alexander Pasternak, Shuzhi Dong, Jacqueline D. Hicks, Artjohn Villafania, Lianzhu Liang, Nicholas Murgolo, Todd Black, William K. Hagmann, Jim Tata, Emma R. Parmee, Ann E. Weber, Jing Su, Haifeng Tang
Publikováno v:
Journal of Medicinal Chemistry. 65:16234-16251
With the emergence and rapid spreading of NDM-1 and existence of clinically relevant VIM-1 and IMP-1, discovery of pan inhibitors targeting metallo-beta-lactamases (MBLs) became critical in our battle against bacterial infection. Concurrent with our
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::f72a226d0f459e4620537979c8da4d4d
https://doi.org/10.1021/acs.jmedchem.2c00766
https://doi.org/10.1021/acs.jmedchem.2c00766
Autor:
Ahmed A. Samatar, Lata Jayaraman, Leigh Zawel, Stephen Fawell, Alan Cooper, Anthony Mannarino, Nathaniel L. Elsen, Stuart Black, Priya Dayananth, Clifford R. Restaino, Daniel McMasters, Jaren Arbanas, Gottfried K. Schroeder, My Sam Mansueto, Alan Hruza, Erick J. Morris, Sharda Jha
HTRF and Biacore binding data for active and inactive ERK1 in the presence of SCH772984
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::5a41d041f5824e4e438c00c030ecb53b
https://doi.org/10.1158/1535-7163.22509012.v1
https://doi.org/10.1158/1535-7163.22509012.v1
Autor:
Ahmed A. Samatar, Lata Jayaraman, Leigh Zawel, Stephen Fawell, Alan Cooper, Anthony Mannarino, Nathaniel L. Elsen, Stuart Black, Priya Dayananth, Clifford R. Restaino, Daniel McMasters, Jaren Arbanas, Gottfried K. Schroeder, My Sam Mansueto, Alan Hruza, Erick J. Morris, Sharda Jha
Sequencing of HCT116 resistant (HCT116R) cell lines
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1442f7a1e528745fe8ccf1630c426567
https://doi.org/10.1158/1535-7163.22509018
https://doi.org/10.1158/1535-7163.22509018
Autor:
Ahmed A. Samatar, Lata Jayaraman, Leigh Zawel, Stephen Fawell, Alan Cooper, Anthony Mannarino, Nathaniel L. Elsen, Stuart Black, Priya Dayananth, Clifford R. Restaino, Daniel McMasters, Jaren Arbanas, Gottfried K. Schroeder, My Sam Mansueto, Alan Hruza, Erick J. Morris, Sharda Jha
Maximal Velocity and Km values
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::84a8f0265469073b8f28fff17b5baa3a
https://doi.org/10.1158/1535-7163.22509015.v1
https://doi.org/10.1158/1535-7163.22509015.v1
Autor:
Ahmed A. Samatar, Lata Jayaraman, Leigh Zawel, Stephen Fawell, Alan Cooper, Anthony Mannarino, Nathaniel L. Elsen, Stuart Black, Priya Dayananth, Clifford R. Restaino, Daniel McMasters, Jaren Arbanas, Gottfried K. Schroeder, My Sam Mansueto, Alan Hruza, Erick J. Morris, Sharda Jha
Analysis of active ERK2 G169D mutant binding to SCH772984
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::61c1b30d69b770056434325087d8ea20
https://doi.org/10.1158/1535-7163.22509003
https://doi.org/10.1158/1535-7163.22509003
Autor:
Ahmed A. Samatar, Lata Jayaraman, Leigh Zawel, Stephen Fawell, Alan Cooper, Anthony Mannarino, Nathaniel L. Elsen, Stuart Black, Priya Dayananth, Clifford R. Restaino, Daniel McMasters, Jaren Arbanas, Gottfried K. Schroeder, My Sam Mansueto, Alan Hruza, Erick J. Morris, Sharda Jha
HTRF and Biacore binding data for active and inactive ERK1 in the presence of SCH772984
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::3185945c7ae768bd2e93b8d986a09ade
https://doi.org/10.1158/1535-7163.22508997
https://doi.org/10.1158/1535-7163.22508997
Autor:
Ahmed A. Samatar, Stephen Fawell, Leigh Zawel, Lata Jayaraman, D. Gary Gilliland, Daniel Hicklin, W. Robert Bishop, Paul Kirschmeier, David Witter, Phieng Siliphaivanh, Ulrike Philippar, Marc R. Pelletier, Bart A. Lutterbach, Ling Zhang, Pierre Daublain, Liang Zhu, Boga Sobhana Babu, Xiaolei Gao, Sunil Paliwal, Joe Kelly, James Wang, Alan Hruza, Gerald Shipps, Li Xiao, Jagdish Desai, Elaine M. Pinheiro, Minilik H. Angagaw, Shuxia Zhao, Rumin Zhang, William Windsor, Edward DiNunzio, Jenny Liu, Brian Long, Stuart Black, Weihong Jin, Yongi Deng, Donna Carr, Alan Cooper, Hugh Zhu, Priya Dayananth, Clifford R. Restaino, Sharda Jha, Erick J. Morris
Supplementary Figures - PDF file 1385K, File contains Supplementary figures of resistant cell lines, proliferation assay of a panel of cell lines, TdF binding assay transcriptional out and kinome selectivity
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::043d9dc9ddac3082860a77d7c7fbd235
https://doi.org/10.1158/2159-8290.22530809
https://doi.org/10.1158/2159-8290.22530809
Autor:
Ahmed A. Samatar, Lata Jayaraman, Leigh Zawel, Stephen Fawell, Alan Cooper, Anthony Mannarino, Nathaniel L. Elsen, Stuart Black, Priya Dayananth, Clifford R. Restaino, Daniel McMasters, Jaren Arbanas, Gottfried K. Schroeder, My Sam Mansueto, Alan Hruza, Erick J. Morris, Sharda Jha
Theoretical maximum binding capacity of immobilized ligand
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::cae21590fd6fe473ad9f65db7f2896fb
https://doi.org/10.1158/1535-7163.22509000.v1
https://doi.org/10.1158/1535-7163.22509000.v1
Autor:
Ahmed A. Samatar, Lata Jayaraman, Leigh Zawel, Stephen Fawell, Alan Cooper, Anthony Mannarino, Nathaniel L. Elsen, Stuart Black, Priya Dayananth, Clifford R. Restaino, Daniel McMasters, Jaren Arbanas, Gottfried K. Schroeder, My Sam Mansueto, Alan Hruza, Erick J. Morris, Sharda Jha
Analysis of active ERK1 G186D mutant binding to SCH772984
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1bffb3b4b7e43c78f92829fdde765183
https://doi.org/10.1158/1535-7163.22509006.v1
https://doi.org/10.1158/1535-7163.22509006.v1
Autor:
Liang Zhu, Weihong Jin, Xin Yao, Hong Mei, Abdul Basit Alhassan, William T. Windsor, Donna Carr, Li Xiao, Sunil Paliwal, Neng-Yang Shih, Sun Robert, Gerald W. Shipps, Sobhana Babu Boga, Yang Nan, Joseph Kelly, Alexei V. Buevich, Brian Long, Paul Kirschmeier, Bradley Sherborne, Kiran Muppalla, Stuart Black, Hon-Chung Tsui, Doll Ronald J, Hugh Y. Zhu, Stacey A. Taylor, Subrahmanyam Gudipati, Gongjie Liu, Alan B. Cooper, Li-Kang Zhang, Kathleen Cox, Robert Bishop, David Hesk, Yongqi Deng, Alan Hruza, Mehul D. Patel, Xiaolei Gao, Priya Dayananth, Tong Wang, Desai Jagdish A, Wang James J-S, Ahmed A. Samatar
[Image: see text] The emergence and evolution of new immunological cancer therapies has sparked a rapidly growing interest in discovering novel pathways to treat cancer. Toward this aim, a novel series of pyrrolidine derivatives (compound 5) were ide
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ab2250ac0d2e55d7a37e61d512ca2156
https://europepmc.org/articles/PMC6047169/
https://europepmc.org/articles/PMC6047169/