Zobrazeno 1 - 10
of 10
pro vyhledávání: '"Pierre-Marc Léo"'
Publikováno v:
Beilstein Journal of Organic Chemistry, Vol 6, Iss 1, Pp 1022-1024 (2010)
Conversion of a myo-inositol derivative into a scyllo-inositol-derived scaffold with C3v symmetry bearing three axial pyridyl appendages is presented. This pre-organized hexadentate ligand allows complexation of silver(I). The crystal structure of th
Externí odkaz:
https://doaj.org/article/95ba14127c4f43ad9ce209d4cfb1402a
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 17:4934-4937
All- O -undec-en-10-yl derivatives of d -glucose have been prepared and their affinities for the Plasmodium falciparum hexose transporter (PfHT) determined; the O -2 derivative displays a good apparent affinity for PfHT ( K I = 2 μM) with no signifi
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::52b151baa43788e678bc6782a959574e
https://doi.org/10.1016/j.bmcl.2007.06.021
https://doi.org/10.1016/j.bmcl.2007.06.021
Publikováno v:
Beilstein Journal of Organic Chemistry
Beilstein Journal of Organic Chemistry, Vol 6, Iss 1, Pp 1022-1024 (2010)
Beilstein Journal of Organic Chemistry, Vol 6, Iss 1, Pp 1022-1024 (2010)
Conversion of a myo-inositol derivative into a scyllo-inositol-derived scaffold with C3v symmetry bearing three axial pyridyl appendages is presented. This pre-organized hexadentate ligand allows complexation of silver(I). The crystal structure of th
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::5d8224dcd6fabf6a16d8cbbaa2bd380e
https://doi.org/10.3762/bjoc.6.115
https://doi.org/10.3762/bjoc.6.115
Publikováno v:
Tetrahedron: Asymmetry. 11:2885-2898
A method has been developed for determining the enantiomeric purity and the absolute configuration of β-aminoalcohols of type ArOCH2CH(OH)CH2NHR (R=iPr, tBu). To determine enantiomeric purity, the amine function was first protected by a benzyl group
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::185260719675e88be916b39127755b52
https://doi.org/10.1016/s0957-4166(00)00254-8
https://doi.org/10.1016/s0957-4166(00)00254-8
Publikováno v:
European Journal of Organic Chemistry. 2000:1007-1012
The iodinatied carbamates 3 (E + Z), with potential β-blocking properties, were synthesized. The first route chosen, from 4-aminophenol and the chloroformate β7, had to be abandoned because of the formation of the oxazolidinone 10 during the epoxid
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::0caa23d9e555da690f4e89aaf2f445bb
https://doi.org/10.1002/(sici)1099-0690(200003)2000:6<1007::aid-ejoc1007>3.0.co
https://doi.org/10.1002/(sici)1099-0690(200003)2000:6<1007::aid-ejoc1007>3.0.co
Publikováno v:
Journal of Labelled Compounds and Radiopharmaceuticals. 42:1195-1202
AMI-9S was synthesized in the S configuration with an enantiomeric purity of over 97% and labelled with iodine-123 with a specific activity of 300 Ci/mmol. Enantiomeric purity was determined by 19 F NMR spectroscopy following derivatisation using (R)
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::c22d55d7571d5ad6cb9082f8bf50ec9f
https://doi.org/10.1002/(sici)1099-1344(199912)42:12<1195::aid-jlcr275>3.0.co
https://doi.org/10.1002/(sici)1099-1344(199912)42:12<1195::aid-jlcr275>3.0.co
Autor:
Rafika Jarray, Stéphanie Kolb, Emmanuelle Braud, Christiane Garbay, Pierre-Marc Léo, Christophe Morin, Tatiana Besset
Publikováno v:
Central European Journal of Chemistry
Central European Journal of Chemistry, 2011, 2 (4), pp.433-440. ⟨10.5155/eurjchem.2.4.433-440.400⟩
Central European Journal of Chemistry, Springer Verlag, 2011, 2 (4), pp.433-440. ⟨10.5155/eurjchem.2.4.433-440.400⟩
Central European Journal of Chemistry, 2011, 2 (4), pp.433-440. ⟨10.5155/eurjchem.2.4.433-440.400⟩
Central European Journal of Chemistry, Springer Verlag, 2011, 2 (4), pp.433-440. ⟨10.5155/eurjchem.2.4.433-440.400⟩
A set of new heteroquinone derivatives bearing two methoxycarbonylmethylthio groups on the benzoquinone ring were synthesized and evaluated for CDC25B phosphatase inhibitory activity. All compounds inhibited the enzyme with IC 50 values in the microm
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c28a41a58007760f3f8b010922a78565
https://normandie-univ.hal.science/hal-02541860
https://normandie-univ.hal.science/hal-02541860
Publikováno v:
ChemInform. 31
The iodinatied carbamates 3 (E + Z), with potential β-blocking properties, were synthesized. The first route chosen, from 4-aminophenol and the chloroformate β7, had to be abandoned because of the formation of the oxazolidinone 10 during the epoxid
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::0e7ded2502716e547b4dda98c69995d3
https://doi.org/10.1002/chin.200020084
https://doi.org/10.1002/chin.200020084
Publikováno v:
ChemInform. 33
On the basis of chemical and spectral data, the structure of the medermycin/lactoquinomycin A has been revised, which has also led to the revision of related C-glycosylated naphthoquinone antibiotics such as lactoquinomycin B, menoxymycins A and B, G
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::fa6084e5e8d9f4e8631b7a56a5c7cd3e
https://doi.org/10.1002/chin.200250198
https://doi.org/10.1002/chin.200250198
Publikováno v:
Organic letters. 4(16)
[reaction: see text] On the basis of chemical and spectral data, the structure of the medermycin/lactoquinomycin A has been revised, which has also led to the revision of related C-glycosylated naphthoquinone antibiotics such as lactoquinomycin B, me
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::46945bfbb43665c5facd063ada97c0a0
https://pubmed.ncbi.nlm.nih.gov/12153216
https://pubmed.ncbi.nlm.nih.gov/12153216