Zobrazeno 1 - 10
of 24
pro vyhledávání: '"Pierre Thesmar"'
Publikováno v:
CHIMIA, Vol 74, Iss 3 (2020)
Externí odkaz:
https://doaj.org/article/c694c4332aa74908bf17e2f0b273b23f
Publikováno v:
CHIMIA, Vol 73, Iss 12 (2019)
Externí odkaz:
https://doaj.org/article/3fb7e7dc892443b7b8608398bf7cc092
Autor:
Anne-Marie Michon, Rab K. Prinjha, Alex Preston, Laurie J. Gordon, Inmaculada Rioja, Pierre Thesmar, Emmanuel Hubert Demont, James Michael Woolven, Stephen John Atkinson, Jon T. Seal, Cassie Messenger, Lee Andrew Harrison, Paola Grandi, Darren Jason Mitchell, Robert J. Watson, Simon Taylor, Chun-wa Chung, James Gray, Antonia J. Lewis, Ian D. Wall, Dave Lugo, Paul Bamborough
Publikováno v:
ACS Med Chem Lett
[Image: see text] Pan-BET inhibitors have shown profound efficacy in a number of in vivo preclinical models and have entered the clinic in oncology trials where adverse events have been reported. These inhibitors interact equipotently with the eight
Autor:
Antonin, Clemenceau, Pierre, Thesmar, Maxime, Gicquel, Alexandre, Le Flohic, Olivier, Baudoin
Publikováno v:
Journal of the American Chemical Society. 142(36)
Cyclopropanes are important structural motifs found in numerous bioactive molecules, and a number of methods are available for their synthesis. However, one of the simplest cyclopropanation reactions involving the intramolecular coupling of two C-H b
Autor:
Pierre, Thesmar, Seemon, Coomar, Alessandro, Prescimone, Daniel, Häussinger, Dennis, Gillingham, Olivier, Baudoin
Publikováno v:
Chemistry (Weinheim an der Bergstrasse, Germany). 26(66)
This article provides a detailed report of our efforts to synthesize the dithiodiketopiperazine (DTP) natural products (-)-epicoccin G and (-)-rostratin A using a double C(sp
Cyclopropanes are important structural motifs found in numerous bioactive molecules, and a number of methods are available for their synthesis. However, one of the simplest cyclopropanation reactions involving the intramolecular coupling of two C–H
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::15e7bf020680e9499c0859595e2586a3
https://doi.org/10.26434/chemrxiv.12408839
https://doi.org/10.26434/chemrxiv.12408839
Cyclopropanes are important structural motifs found in numerous bioactive molecules, and a number of methods are available for their synthesis. However, one of the simplest cyclopropanation reactions involving the intramolecular coupling of two C-H b
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7b648714ac696e329b66b62e6a3742d3
Autor:
Pierre Thesmar, Alessandro Prescimone, Olivier Baudoin, Seemon Coomar, Daniel Häussinger, Dennis Gillingham
This article provides a detailed report of our efforts to synthesize the dithiodiketopiperazine (DTP) natural products (-)-epicoccin G and (-)-rostratin A using a double C(sp3 )-H activation strategy. The strategy's viability was first established on
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::4a3d9cae92bdfe22ad9010b2067abb65
Autor:
Pierre, Thesmar, Olivier, Baudoin
Publikováno v:
Journal of the American Chemical Society. 141(40)
Dithiodiketopiperazines are complex polycyclic natural products possessing a variety of interesting biological activities. Despite their interest, relatively few total syntheses have been completed. We herein report the enantioselective, scalable, an
Publikováno v:
Chimia. 73(6)