Zobrazeno 1 - 9
of 9
pro vyhledávání: '"Pierre Beuchet"'
Autor:
Stephane Larrouture, Jean-Michel Léger, Arlette Neveu, Gérard Deffieux, Pierre Beuchet, Martine Varache-Lembège, A. Nuhrich, Joseph Vercauteren
Publikováno v:
European Journal of Medicinal Chemistry. 34:773-779
Polymethoxylated and polyhydroxylated derivatives of 2-amino-4-arylthiazoles bearing a halogenobenzenesulfonamide moiety at position 2 were synthesized as azole antifungal analogues. X-ray crystallography studies revealed the predominance of the 2-im
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::f4d9b3349e4a6957c90154699b959642
https://doi.org/10.1016/s0223-5234(99)00215-9
https://doi.org/10.1016/s0223-5234(99)00215-9
Publikováno v:
Tetrahedron Letters. 36:6055-6058
New reactions of enamines were observed with allyl bromide or methyl bromoacetate in the presence of indium powder in THF, yielding respectively homoallylamines and β-aminoesters.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::71b0102b41ccea2ac60af99f25831a01
https://doi.org/10.1016/0040-4039(95)01241-9
https://doi.org/10.1016/0040-4039(95)01241-9
Publikováno v:
ChemInform. 24
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::7db34d9c11047c2feec02db7c5e706ab
https://doi.org/10.1002/chin.199312097
https://doi.org/10.1002/chin.199312097
Publikováno v:
ChemInform. 26
New reactions of enamines were observed with allyl bromide or methyl bromoacetate in the presence of indium powder in THF, yielding respectively homoallylamines and β-aminoesters.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::f8edadb9c81ecf376a16744a8a16325a
https://doi.org/10.1002/chin.199550014
https://doi.org/10.1002/chin.199550014
Publikováno v:
ChemInform. 30
Δ 7 -5-Desaturase catalyses one of the last steps in ergosterol biosynthesis in fungi. Moreover Δ 5 -unsaturation is necessary for the sparking function. Synthesis of three pairs of C-6 epimeric cholestanol derivatives are described as potential gr
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::a69753d877c91736b76a10898bf30052
https://doi.org/10.1002/chin.199917194
https://doi.org/10.1002/chin.199917194
Autor:
Arlette Neveu, Stephane Larrouture, Martine Varache-Lembège, A. Nuhrich, Jean-Michel Léger, Gérard Deffieux, Pierre Beuchet, Joseph Vercauteren
Publikováno v:
ChemInform. 31
Polymethoxylated and polyhydroxylated derivatives of 2-amino-4-arylthiazoles bearing a halogenobenzenesulfonamide moiety at position 2 were synthesized as azole antifungal analogues. X-ray crystallography studies revealed the predominance of the 2-im
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::fb49a682b2fe52a58922ee0d693e7d19
https://doi.org/10.1002/chin.200006119
https://doi.org/10.1002/chin.200006119
Publikováno v:
Bioorganicmedicinal chemistry letters. 8(24)
Δ 7 -5-Desaturase catalyses one of the last steps in ergosterol biosynthesis in fungi. Moreover Δ 5 -unsaturation is necessary for the sparking function. Synthesis of three pairs of C-6 epimeric cholestanol derivatives are described as potential gr
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1d3ca99c0015fffa12d8447cffc776f8
https://pubmed.ncbi.nlm.nih.gov/9934483
https://pubmed.ncbi.nlm.nih.gov/9934483
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 9:1599-1600
25-aminolanostenol 1 and 25-aminocholesterol 2 were hemisynthesized from natural sterols and tested in vitro against Candida albicans. The biological activity of compound 1 was rather weak, whereas 2 exhibited in vitro antifungal activity with MIC va
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::5f7871ccafc96b85a78edfcc13cfa7e4
https://doi.org/10.1016/s0960-894x(99)00233-4
https://doi.org/10.1016/s0960-894x(99)00233-4
Publikováno v:
Tetrahedron Letters. 33:5959-5960
Aldimines are allylated under simple Barbier type conditions using ally] bromide and indium powder in THF.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::d0ccc871d7f0cc9c6e450aace2ca9b2a
https://doi.org/10.1016/s0040-4039(00)61099-7
https://doi.org/10.1016/s0040-4039(00)61099-7