Zobrazeno 1 - 10 of 32 pro vyhledávání: '"Pierre, Brouant"'
1
The Mechanisms of Alpha-Amylase Inhibition by Flavan-3-Ols and the Possible Impacts of Drinking Green Tea on Starch Digestion
Autor: Pierre Brouant, El Hassan Ajandouz, Véronique Desseaux, Pierre Stocker
Publikováno v: Journal of Food Science. 83:2858-2865
Many studies have shown that flavan-3-ols inhibit mammalian alpha-amylases but the published IC50 and Ki values vary up to a thousand times. We therefore tested the effects of 6 pure flavan-3-ols-abundant in green tea-on the activity of pure porcine
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::d8051e96a686c8dfdb40ba0c84a2ff5f
https://doi.org/10.1111/1750-3841.14353
Zobrazit plný text záznamu
3
Inhibition of Cryptosporidium parvum in vitro by 9-(Alkylthio)acridine Derivatives
Autor: Maria‐Jose Rosales, Nadia Bsiri, Latifa Khalifa, Jacques Barbe, Carmen Mascaro, Pierre Brouant, Janina Karolak-Wojciechowska
Publikováno v: Arzneimittelforschung. 50:163-166
The synthesis of several acridinic thioethers is described. Compounds prepared were tested in vitro as potential drugs against the opportunistic infection known as cryptosporidiosis. With a view to predict activity, the quantitative structure-activit
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1bd1fa4f419570c42b18e4199dbf3ec0
https://doi.org/10.1055/s-0031-1300183
Zobrazit plný text záznamu
4
Alkylaminoquinolines inhibit the bacterial antibiotic efflux pump in multidrug-resistant clinical isolates
Autor: Jacques Barbe, Pierre Brouant, Abdallah Mahamoud, Jacqueline Chevalier, Monique Malléa, Sandrine Alibert-Franco, Jean-Marie Pagès
Publikováno v: Biochemical Journal. 376:801-805
Over the last decade, MDR (multidrug resistance) has increased worldwide in microbial pathogens by efflux mechanisms, leading to treatment failures in human infections. Several Gram-negative bacteria efflux pumps have been described. These proteinace
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c4d1e7ad8969ca5855135222154fc09d
https://doi.org/10.1042/bj20030963
Zobrazit plný text záznamu
5
Modified electrodes with new phenothiazine derivatives for electrocatyltic oxidation of NADH
Autor: Delia Dicu, Castelia Cristea, Ioan A. Silberg, Pierre Brouant, Liana Maria Muresan, Ionel Catalin Popescu
Publikováno v: Electrochimica Acta. 45:3951-3957
Phenothiazine derivatives containing two linearly condensed phenothiazine moieties, 16H,18H-dibenzo[c,l]-7,9-dithia-16,18-diazapentacene (I), dibenzo[c,l]-16,18-diacetyl-7,9-dithia-16,18-diazapentacene (II) dibenzo[c,l]-16,18-dibenzoyl-7,9-dithia-16,
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::09ba27d3190b29fd5dcc65632391a721
https://doi.org/10.1016/s0013-4686(00)00485-0
Zobrazit plný text záznamu
6
Structure and conformational analysis of 5,11-dibenzyldibenzo[b,f][1,5]diazocine-6,12-dione. A novel approach for new chemosensitizers
Autor: E Nonnenmacher, Pierre Brouant, J. Barbe, A. Mrozek, Janina Karolak-Wojciechowska
Publikováno v: Journal of Molecular Structure. 522:263-269
On the basis of structural similarities between various calcium channel antagonists (Verapamil or Diltiazem) a novel series of derivatives belonging to the dibenzodiazocinedione family were designed and synthesised to obtain drugs able to revert mult
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::f234ee58d8184418335ab690056e277e
https://doi.org/10.1016/s0022-2860(99)00369-5
Zobrazit plný text záznamu
7
Un sel de Maprotiline (Ludiomil), Médicament Psychotrope, C20H24N+.C21H22NO2−.0,5H2O
Autor: Jean-Claude Soyfer, G. Pèpe, Pierre Brouant, J. Barbe, J. P. Reboul, Didier Siri
Publikováno v: Acta Crystallographica Section C Crystal Structure Communications. 51:970-974
Maprotiline (ludiomil) is a tetracyclic antidepressant drug which crystallized in DMF as the salt [3-(9,10-dihydro-9,10-ethano-9-anthracenyl)propyl]methylammonium N-[3-(9,10-dihydro-9,10-ethano-9-anthracenyl)propyl]-N-methylcarbamate hemihydrate. The
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::851d4af32481cf905c25ecb96e250d57
https://doi.org/10.1107/s0108270194006049
Zobrazit plný text záznamu
8
Antimicrobial activity of 9-oxo and 9-thio acridines: Correlation with intercalation into DNA and effects on macromolecular biosynthesis
Autor: A Crémieux, A.-M. Galy, Derek Sharples, J Chevalier, J. Barbe, J. P. Galy, H Berny, Pierre Brouant
Publikováno v: Research in Microbiology. 146:73-83
The antimicrobial activity of several new 9-acridinones and 9-thioalkylacridines towards Escherichia coli, Staphylococcus aureus, Mycobacterium smegmatis and Candida albicans was investigated. Minimal inhibitory, bactericidal and fungicidal concentra
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::13e602f4ac418709a17550d975fbcb35
https://doi.org/10.1016/0923-2508(96)80272-5
Zobrazit plný text záznamu
10
ChemInform Abstract: A Potential Antiprotozoal Drug Containing Acridine and Thiadiazole Moieties
Autor: P. Amiel, Pierre Brouant, A. Mrozek, Janina Karolak-Wojciechowska, Jacques Barbe
Publikováno v: ChemInform. 28
The title compound, 3-(6-chloro-2-methoxy-9-acridinyl)-5-[2-(diethylamino)ethylthio]-1,3,4-thiadiazol-2(3H)-one, C 22 H 23 ClN 4 OS 3 , belongs to a series of new potential antiprotozoal drugs containing the acridine and thiadiazole systems. These tw
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::d0403d0c07c59c9d345e94e2abec5966
https://doi.org/10.1002/chin.199714039
Zobrazit plný text záznamu

Vyhledávací nástroje:

Upřesnit hledání

Omezení vyhledávání
Plný text Recenzováno Digitální knihovna AV ČR
Zdroje