Zobrazeno 1 - 4
of 4
pro vyhledávání: '"Philipp Cueni"'
Publikováno v:
Bioorganic & Medicinal Chemistry. 26:970-976
A scalable 5-step synthesis of the diazacarbazole derivative 1 used as tau PET tracer precursor is reported. Key features of this synthesis include a Buchwald-Hartwig amination, a Pd catalyzed CH activation and a Suzuki-Miyaura cross-coupling.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::38113eab8b54092d1cfce0e5acb11b83
https://doi.org/10.1016/j.bmc.2017.10.007
https://doi.org/10.1016/j.bmc.2017.10.007
Autor:
Hayden T. Ravert, Daniel P. Holt, Guy Zielinski, Philipp Schmid, Emmanuel Pinard, Roger David Norcross, Robert F. Dannals, Philipp Cueni, Serge Burner, Thomas Hartung, Pius Waldmeier
Publikováno v:
Journal of Labelled Compounds and Radiopharmaceuticals. 54:702-707
The glycine transporter type 1 (GlyT1) has emerged as a key novel target for the treatment of schizophrenia. We have recently discovered and developed [11C]RO5013853 as a novel positron emission tomography tracer for GlyT1 for which a reliable five-s
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::2c081394253d0cab9fe66478d5ed671f
https://doi.org/10.1002/jlcr.1911
https://doi.org/10.1002/jlcr.1911
ChemInform Abstract: Cu-Catalyzed Aerobic Oxidative Cyclization of Guanidylpyridines and Derivatives
Autor:
Serena Fantasia, Bjoern Bartels, Nicolas Gaeng, Philipp Cueni, Conor Gordon Bolas, Andrada Stefania Trita
Publikováno v:
ChemInform. 46
A simple and highly efficient system produces a series of 2-amino-[1,2,4]triazolo[1,5-a]pyridine structures and analogues such as (X) and (XII).
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::549145031b5217cb312c1032ada08d20
https://doi.org/10.1002/chin.201524178
https://doi.org/10.1002/chin.201524178
Autor:
Andrada Stefania Trita, Nicolas Gaeng, Serena Fantasia, Bjoern Bartels, Conor Gordon Bolas, Philipp Cueni
Publikováno v:
The Journal of organic chemistry. 80(2)
A new method for the straightforward synthesis of 2-amino-[1,2,4]triazolo[1,5-a]pyridines and derivatives is presented. The target products are synthesized in high yields from guanidylpyridines and analogues via copper-catalyzed N–N coupling. The p
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::f481e403f2e2ccda153d03310bab24aa
https://pubmed.ncbi.nlm.nih.gov/25495477
https://pubmed.ncbi.nlm.nih.gov/25495477