Zobrazeno 1 - 10
of 30
pro vyhledávání: '"Pharit, Kamsri"'
Autor:
Somjintana Taveepanich, Kampanart Chayajarus, Jutharat Jittimanee, Naruedon Phusri, Paptawan Thongdee, Khemmisara Sawatdee, Pharit Kamsri, Auradee Punkvang, Khomson Suttisintong, Pornpan Pungpo, Wanwisa Suwannaloet, Ruttiya Thongrung, Kanjana Pangjit
Publikováno v:
Heliyon, Vol 10, Iss 19, Pp e38213- (2024)
Background: Iron overload and inflammation are severe conditions that can lead to various chronic diseases. However, the current iron chelator drugs have their limitations. The phytochemical compounds from herbals, such as brazilin, the major active
Externí odkaz:
https://doaj.org/article/4403abe0166949e7b03f5667679b8e4a
Autor:
Bundit Kamsri, Bongkochawan Pakamwong, Paptawan Thongdee, Naruedon Phusi, Pharit Kamsri, Auradee Punkvang, Sombat Ketrat, Patchreenart Saparpakorn, Supa Hannongbua, Jidapa Sangswan, Khomson Suttisintong, Sanya Sureram, Prasat Kittakoop, Poonpilas Hongmanee, Pitak Santanirand, Jiraporn Leanpolchareanchai, Kirsty E. Goudar, James Spencer, Adrian J. Mulholland, Pornpan Pungpo
Publikováno v:
Journal of Chemical Information and Modeling. 63:2707-2718
Autor:
Pharit Kamsri, Auradee Punkvang, Somjintana Taveepanich, Sombat Ketrat, Patchreenart Saparpakorn, Supa Hannongbua, Khomson Suttisintong, Kanjana Pangjit, Pornpan Pungpo
Publikováno v:
Future Medicinal Chemistry. 14:1297-1308
Background: JAK2 inhibitors have been proposed as a new therapeutic option for thalassemia therapy. The objective of this study was to discover the key structural features for improving 2-aminopyrimidine derivatives as potential JAK2 inhibitors. Mate
Autor:
Paptawan Thongdee, Chayanin Hanwarinroj, Bongkochawan Pakamwong, Pharit Kamsri, Auradee Punkvang, Jiraporn Leanpolchareanchai, Sombat Ketrat, Patchreenart Saparpakorn, Supa Hannongbua, Kanchiyaphat Ariyachaokun, Khomson Suttisintong, Sanya Sureram, Prasat Kittakoop, Poonpilas Hongmanee, Pitak Santanirand, Galina V. Mukamolova, Rosemary A. Blood, Yuiko Takebayashi, James Spencer, Adrian J. Mulholland, Pornpan Pungpo
Publikováno v:
Journal of Chemical Information and Modeling. 62:6508-6518
Autor:
Chayanin Hanwarinroj, Nareudon Phusi, Bundit Kamsri, Pharit Kamsri, Auradee Punkvang, Sombat Ketrat, Patchreenart Saparpakorn, Supa Hannongbua, Khomson Suttisintong, Prasat Kittakoop, James Spencer, Adrian J Mulholland, Pornpan Pungpo
Publikováno v:
Hanwarinroj, C, Phusi, N, Kamsri, B, Kamsri, P, Punkvang, A, Ketrat, S, Saparpakorn, P, Hannongbua, S, Suttisintong, K, Kittakoop, P, Spencer, J, Mulholland, A J & Pungpo, P 2022, ' Discovery of novel and potent InhA inhibitors by an in silico screening and pharmacokinetic prediction ', Future Medicinal Chemistry, vol. 14, no. 10, pp. 717-729 . https://doi.org/10.4155/fmc-2021-0348
Aim: In silico screening approaches were performed to discover novel InhA inhibitors. Methods: Candidate InhA inhibitors were obtained from the combination of virtual screening and pharmacokinetic prediction. In addition, molecular mechanics Poisson
Autor:
Bongkochawan Pakamwong, Paptawan Thongdee, Bundit Kamsri, Naruedon Phusi, Pharit Kamsri, Auradee Punkvang, Sombat Ketrat, Patchreenart Saparpakorn, Supa Hannongbua, Kanchiyaphat Ariyachaokun, Khomson Suttisintong, Sanya Sureram, Prasat Kittakoop, Poonpilas Hongmanee, Pitak Santanirand, James Spencer, Adrian J. Mulholland, Pornpan Pungpo
Publikováno v:
Pakamwong, B, Thongdee, P, Spencer, J, Kamsri, B, Mulholland, A J & Pungpo, P 2022, ' Identification of potent DNA Gyrase inhibitors active against mycobacterium tuberculosis ', Journal of Chemical Information and Modeling, vol. 62, no. 7, pp. 1680-1690 . https://doi.org/10.1021/acs.jcim.1c01390
Mycobacterium tuberculosis DNA gyrase manipulates the DNA topology using controlled breakage and religation of DNA driven by ATP hydrolysis. DNA gyrase has been validated as the enzyme target of fluoroquinolones (FQs), second-line antibiotics used fo
Autor:
Thi-Kim-Dung Le, Ade Danova, Thammarat Aree, Thuc-Huy Duong, Mamoru Koketsu, Masayuki Ninomiya, Yoshiharu Sawada, Pharit Kamsri, Pornpun Pungpo, Warinthorn Chavasiri
Publikováno v:
Journal of Natural Products. 85:776-786
Autor:
Potjanee Srimanote, Pornpan Pungpo, Bongkochawan Pakamwong, Auradee Punkvang, Prasat Kittakoop, James Spencer, Khomson Suttisintong, Chayanin Hanwarinroj, Pharit Kamsri, Nitima Suttipanta, Sanya Sureram, Chomphunuch Songsiriritthigul
Publikováno v:
Songsiriritthigul, C, Hanwarinroj, C, Pakamwong, B, Srimanote, P, Suttipanta, N, Sureram, S, Suttisintong, K, Kamsri, P, Punkvang, A, Spencer, J, Kittakoop, P & Pungpo, P 2021, ' Inhibition of Mycobacterium tuberculosis InhA by 3-nitropropanoic acid ', Proteins: Structure, Function, and Bioinformatics, vol. 90, no. 3, pp. 898-904 . https://doi.org/10.1002/prot.26268
3-Nitropropanoic acid (3NP), a bioactive fungal natural product, was previously demonstrated to inhibit growth of Mycobacterium tuberculosis. Here we demonstrate that 3NP inhibits the 2-trans-enoyl-acyl carrier protein reductase (InhA) from Mycobacte
Autor:
Prasat Kittakoop, Anuchit Phanumartwiwath, Pharit Kamsri, Chatchakorn Eurtivong, Chatchai Kesornpun, Sanya Sureram, Auradee Punkvang, Somsak Ruchirawat, Pornpan Pungpo, Poonpilas Hongmanee
Publikováno v:
Journal of Chemical Research. 45:1003-1015
Isoxazoline derivatives of the natural products eugenol, 1’- S-acetoxychavicol acetate and sclareol are prepared through 1,3-dipolar cycloaddition reactions in an aqueous buffered system. The compounds are evaluated for their antitubercular and ant
Autor:
Chayanin Hanwarinroj, Paptawan Thongdee, Darunee Sukchit, Somjintana Taveepanich, Pharit Kamsri, Auradee Punkvang, Sombat Ketrat, Patchreenart Saparpakorn, Supa Hannongbua, Khomson Suttisintong, Prasat Kittakoop, James Spencer, Adrian J. Mulholland, Pornpan Pungpo
Publikováno v:
Hanwarinroj, C, Thongdee, P, Sukchit, D, Taveepanich, S, Punkvang, A, Kamsri, P, Saparpakorn, P, Ketrat, S K, Hannongbua, S, Suttisintong, K, Kittakoop, P, Spencer, J, Mulholland, A J & Pungpo, P 2022, ' In silico design of novel quinazoline-based compounds as potential Mycobacterium tuberculosis PknB inhibitors through 2D and 3D-QSAR, molecular dynamics simulations combined with pharmacokinetic predictions ', Journal of Molecular Graphics and Modelling, vol. 115, 108231 . https://doi.org/10.1016/j.jmgm.2022.108231
Serine/threonine protein kinase B (PknB) is essential to Mycobacterium tuberculosis (M. tuberculosis) cell division and metabolism and a potential anti-tuberculosis drug target. Here we apply Hologram Quantitative Structure Activity Relationship (HQS
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::285b19034deaaebc63ba52c3420cdfe5
https://research-information.bris.ac.uk/ws/files/326367115/R1_Maintext_PknB_Final_submitted.pdf
https://research-information.bris.ac.uk/ws/files/326367115/R1_Maintext_PknB_Final_submitted.pdf