Zobrazeno 1 - 4
of 4
pro vyhledávání: '"Peter K. Dornan"'
Development of a Commercial Manufacturing Process for Sotorasib, a First-in-Class KRASG12C Inhibitor
Autor:
Liang Zhang, Daniel J. Griffin, Matthew G. Beaver, Laura E. Blue, Christopher J. Borths, Derek B. Brown, Seb Caille, Ying Chen, Alan H. Cherney, Brian M. Cochran, John T. Colyer, Michael T. Corbett, Tiffany L. Correll, Richard D. Crockett, Xi-Jie Dai, Peter K. Dornan, Robert P. Farrell, Simon J. Hedley, Hsiao-Wu Hsieh, Liang Huang, Seth Huggins, Min Liu, Michael A. Lovette, Kyle Quasdorf, William Powazinik, Jonathan Reifman, Jo Anna Robinson, Rahul P. Sangodkar, Sonika Sharma, Srividya Sharvan Kumar, Austin G. Smith, Gabrielle St-Pierre, Jason S. Tedrow, Oliver R. Thiel, Jonathan V. Truong, Shawn D. Walker, Carolyn S. Wei, Ashraf Wilsily, Yong Xie, Ning Yang, Andrew T. Parsons
Publikováno v:
Organic Process Research & Development. 26:3115-3125
Autor:
Xi-Jie Dai, Paul Krolikowski, James I. Murray, Carolyn S. Wei, Peter K. Dornan, Andreas R. Rötheli, Seb Caille, Oliver R. Thiel, Austin G. Smith, Andrew T. Parsons
Publikováno v:
The Journal of Organic Chemistry. 87:8437-8444
An organocatalyzed, formal (3+3) cycloaddition reaction is described for the practical synthesis of substituted pyridines. Starting from readily available enamines and enal/ynal/enone substrates, the protocol affords tri- or tetrasubstituted pyridine
Autor:
Guilong Charles Cheng, Neil F. Langille, Alicia Zeng, Jenil Patel, Chris Scardino, Travis Anthoine, William E. Lake, Scott W. Roberts, Matthew G. Beaver, John L. Tucker, Shawn D. Walker, Dawn E. Cohen, William Powazinik, Peter K. Dornan, Sheng Cui, Simone Spada, Susan P. Lucas
Publikováno v:
Organic Process Research & Development. 24:481-489
Epoxyketone 4 is an isolated intermediate in the manufacturing route to the commercial proteasome inhibitor carfilzomib (Kyprolis). Commercial process development and optimization efforts toward th...
Publikováno v:
ChemInform. 42