Zobrazeno 1 - 10
of 12
pro vyhledávání: '"Paula Pérez-Faginas"'
Autor:
Paula Pérez-Faginas, M Teresa Aranda, M Teresa García-López, Lourdes Infantes, Asia Fernández-Carvajal, José Manuel González-Ros, Antonio Ferrer-Montiel, Rosario González-Muñiz
Publikováno v:
PLoS ONE, Vol 8, Iss 1, p e53231 (2013)
1,2-Diamine derivatives are valuable building blocks to heterocyclic compounds and important precursors of biologically relevant compounds. In this respect, amino acid-derived β-keto esters are a suitable starting point for the synthesis of β,γ-di
Externí odkaz:
https://doaj.org/article/7dfdae62614e42498e3fa7f83dc0793c
Autor:
Roberto de la Torre-Martínez, M. Teresa Aranda, Antonio Ferrer-Montiel, Rosario González-Muñiz, Susana Quirce, Paula Pérez-Faginas, Asia Fernández-Carvajal
Publikováno v:
Digital.CSIC. Repositorio Institucional del CSIC
instname
instname
Electronic supplementary information (ESI) available: Protocol for the evaluation of compound 4b in the CFA-induced paw inflammation model and obtained results. See DOI: 10.1039/c5ra25709c
A high throughput screening campaign identified nine b,g
A high throughput screening campaign identified nine b,g
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8dbc6eb2d6d27e1ace7c1181d2d6e2e4
http://hdl.handle.net/10261/141530
http://hdl.handle.net/10261/141530
Publikováno v:
Current Organic Synthesis. 6:325-341
Autor:
M. Teresa Aranda, Paula Pérez-Faginas, Asia Fernández-Carvajal, Lourdes Infantes, Antonio Ferrer-Montiel, M. Teresa García-López, José M. González-Ros, Rosario González-Muñiz
Publikováno v:
PLoS ONE
PLoS ONE, Vol 8, Iss 1, p e53231 (2013)
Digital.CSIC. Repositorio Institucional del CSIC
instname
PLoS ONE, Vol 8, Iss 1, p e53231 (2013)
Digital.CSIC. Repositorio Institucional del CSIC
instname
1,2-Diamine derivatives are valuable building blocks to heterocyclic compounds and important precursors of biologically relevant compounds. In this respect, amino acid-derived β-keto esters are a suitable starting point for the synthesis of β,γ-di
Autor:
Paula Pérez-Faginas, Carmen Cuevas, Andrés Francesch, M. Teresa García-López, M. Teresa Aranda, Rosario González-Muñiz
Publikováno v:
European journal of medicinal chemistry. 46(10)
The in vitro cytotoxicity assays of several enantiopure (3S,4S)- and (3R,4R)-1,3,4,4-tetrasubstituted β-lactams derived from amino acids have shown that the (3S,4S)-4-benzyl-1-p-methoxybenzyl-3-methyl-4-methoxycarbonyl derivative 2a, obtained from P
Autor:
Jan Balzarini, Paula Pérez-Faginas, M. Teresa Aranda, Graciela Andrei, M. Teresa García-López, Robert Snoeck, Rosario González-Muñiz
Publikováno v:
Bioorganic & Medicinal Chemistry
Graphical abstract
SAR studies on an azetidine-containing dipeptide prototype inhibitor of HCMV are described. Three series of structurally modified analogues, involving substitutions at the N- and C-terminus, and at the C-terminal side-chain we
SAR studies on an azetidine-containing dipeptide prototype inhibitor of HCMV are described. Three series of structurally modified analogues, involving substitutions at the N- and C-terminus, and at the C-terminal side-chain we
Publikováno v:
ChemInform. 41
Review: [asymmetric synthesis of β-lactams through [2 + 2] cycloaddition reactions; 285 refs.].
Publikováno v:
Digital.CSIC. Repositorio Institucional del CSIC
instname
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Theoretical calculations on the transition states of the cyclization of 2S-chloropropionyl amino acid derivatives to the corresponding β-lactams have served to explain the high stereoselectivity of the reaction, and have been the driving force to ex
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d5120cff71eb5ccdc70ab22dcf0f703a
http://hdl.handle.net/10261/81196
http://hdl.handle.net/10261/81196
Autor:
Rosario González-Muñiz, Aisling O'Byrne, Fran O'Reilly, Paula Pérez-Faginas, M. Teresa García-López, M. Jesús Pérez de Vega, Carlos García-Aparicio, Mercedes Martín-Martínez
Publikováno v:
Organic letters. 9(8)
[reaction: see text] The base-promoted cyclization of optically pure N-(p-methoxybenzyl)-N-(2-chloro)propionyl amino acid derivatives resulted in a diastereo- and enantioselective approach to valuable 1,3,4,4-tetrasubstituted beta-lactams. The stereo