Zobrazeno 1 - 10
of 37
pro vyhledávání: '"Patrizia Minetti"'
Autor:
Gianluca Giorgi, Massimo Valoti, Beatrice Gorelli, Mascia Benedusi, Nicola Relitti, Roberto Colangeli, Sandra Gemma, Mauro Maccarrone, Roberto Di Maio, Stefano Federico, Filomena Fezza, Giuseppe Valacchi, Simone Brogi, Giuseppe Di Giovanni, Alessandro Papa, Stefania Lamponi, Giulia Chemi, Alessandra Pecorelli, Alessandro Grillo, Giuseppe Campiani, Simona Saponara, Patrizia Minetti, Stefania Butini, Domenico Fazio
Temporal lobe epilepsy is the most common form of epilepsy, and current antiepileptic drugs are ineffective in many patients. The endocannabinoid system has been associated with an on-demand protective response to seizures. Blocking endocannabinoid c
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::22b2bc937d2e3fdb998f3f44e0cfe562
http://hdl.handle.net/11697/172837
http://hdl.handle.net/11697/172837
Autor:
Vincenzo Di Marzo, Stefania Butini, Marco Paolino, Patrizia Minetti, Mascia Benedusi, Margherita Brindisi, Marco Allarà, Simone Brogi, Samuele Maramai, Sandra Gemma, Giuseppe Borrelli, Giuseppe Valacchi, Carla Ghelardini, Alessia Ligresti, Alessandra Pecorelli, Alessandro Grillo, Lorenzo Di Cesare Mannelli, Giuseppe Campiani
Publikováno v:
ChemMedChem
13 (2018): 2090–2103. doi:10.1002/cmdc.201800397
info:cnr-pdr/source/autori:Brindisi, Margherita; Borrelli, Giuseppe; Brogi, Simone; Grillo, Alessandro; Maramai, Samuele; Paolino, Marco; Benedusi, Mascia; Pecorelli, Alessandra; Valacchi, Giuseppe; Mannelli, Lorenzo Di Cesare; Ghelardini, Carla; Allara, Marco; Ligresti, Alessia; Minetti, Patrizia; Campiani, Giuseppe; di Marzo, Vincenzo; Butini, Stefania; Gemma, Sandra/titolo:Development of Potent Inhibitors of Fatty Acid Amide Hydrolase Useful for the Treatment of Neuropathic Pain/doi:10.1002%2Fcmdc.201800397/rivista:ChemMedChem (Print)/anno:2018/pagina_da:2090/pagina_a:2103/intervallo_pagine:2090–2103/volume:13
13 (2018): 2090–2103. doi:10.1002/cmdc.201800397
info:cnr-pdr/source/autori:Brindisi, Margherita; Borrelli, Giuseppe; Brogi, Simone; Grillo, Alessandro; Maramai, Samuele; Paolino, Marco; Benedusi, Mascia; Pecorelli, Alessandra; Valacchi, Giuseppe; Mannelli, Lorenzo Di Cesare; Ghelardini, Carla; Allara, Marco; Ligresti, Alessia; Minetti, Patrizia; Campiani, Giuseppe; di Marzo, Vincenzo; Butini, Stefania; Gemma, Sandra/titolo:Development of Potent Inhibitors of Fatty Acid Amide Hydrolase Useful for the Treatment of Neuropathic Pain/doi:10.1002%2Fcmdc.201800397/rivista:ChemMedChem (Print)/anno:2018/pagina_da:2090/pagina_a:2103/intervallo_pagine:2090–2103/volume:13
The unique role of fatty acid amide hydrolase (FAAH) in terminating endocannabinoid (EC) signaling supports its relevance as a therapeutic target. Inhibition of EC metabolizing enzymes elicits indirect agonism of cannabinoid receptors (CBRs) and ther
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ca3f35358017e829cc25aa116a66d3c0
http://hdl.handle.net/11588/760585
http://hdl.handle.net/11588/760585
Autor:
Mario Vertechy, Silvia Pace, Katia Lombardo, Franco Borsini, Antonio Caprioli, Patrizia Minetti, Stefano Di Serio, Teresa Riccioni, Maria Antonietta Stasi
Publikováno v:
European Journal of Pharmacology. 761:353-361
Antagonism of the adenosine A2A receptor represents a promising strategy for non-dopaminergic treatment of Parkinson׳s disease (PD). Previously, the adenosine A2A receptor antagonist ST1535 was shown to possess potential beneficial effects in animal
Autor:
Diana Celona, Franco Borsini, Mauro Marzi, Gilberto Spadoni, Silvia Rivara, Patrizia Minetti, Annalida Bedini, Teresa Riccioni, Marco Mor, Giorgio Tarzia, Walter Cabri, Silvia Bartolucci, Daniele Pala
Publikováno v:
European Journal of Medicinal Chemistry. 80:8-35
Many known 5-HT7 ligands contain either a serotonin-like or an arylpiperazine structure that, in published SAR studies, are generally supposed to bind the same receptor pocket. Conversely, we explored the hypothesis that two such moieties can co-exis
Autor:
Luca Pescatori, Orlando Ghirardi, Roberto Di Santo, Diana Celona, Giovanna Guiso, Federica Rosi, Fabrizio Giorgi, Roberta Costi, Mario Vertechy, Patrizia Minetti, Paola Piovesan, Luigi Scipione, Mauro Marzi, Giuliana Cuzzucoli Crucitti, Silvio Caccia
Publikováno v:
Journal of Medicinal Chemistry
Journal of Medicinal Chemistry, American Chemical Society, 2012, 55 (19), pp.8538-48. ⟨10.1021/jm301105m⟩
Journal of Medicinal Chemistry, American Chemical Society, 2012, 55 (19), pp.8538-48. ⟨10.1021/jm301105m⟩
International audience; Dyes like CR are able to inhibit the aggregation of Aβ fibrils. Thus, a screening of a series of dyes including ABBB (1) was performed. Its main component 2 tested in an in vitro assay (i.e., ThT assay) showed good potency at
Autor:
Hyewhon Rhim, Bo Hye Im, Franco Borsini, Fabio Bordi, Hyung Mun Yun, Patrizia Minetti, Gilberto Spadoni, Teresa Riccioni, Giorgio Tarzia
Publikováno v:
European Journal of Pharmacology. 661:8-14
5-HT(6) receptor is one of the most recently cloned serotonin receptors, and it might play important roles in Alzheimer's disease, depression, and learning and memory disorders. Availability of only very few 5-HT(6) receptor agonists, however, does n
Autor:
Patrizia Minetti, Francesca Bartoccini, Diana Celona, Giorgio Tarzia, Walter Cabri, Giovanni Piersanti
Publikováno v:
The Journal of Organic Chemistry. 75:5398-5401
The scope and limitations of using palladium-catalyzed cross-coupling reactions of diverse butyl metal species with two different 2-halopurines were evaluated. While tributylboranes reacted readily and regioselectively with both 2-chloro-6-dibenzylam
Autor:
Carlo Tallarico, Patrizia Minetti, Simone Lucarini, Francesca Bartoccini, Michele Bassi, Federica Vacondio, Francesca Capocasa, Pietro Grossi, Francesco Manera, Giandomenico Brogin, Teresa Riccioni, Silvia Pace, Franco Borsini, Giorgio Tarzia, Maria Antonietta Stasi, Giovanni Piersanti, Walter Cabri
Inhibition of adenosine A2A receptors has been shown to elicit a therapeutic response in preclinical animal models of Parkinson's disease (PD). We previously identified the triazolo-9H-purine, ST1535, as a potent A(2A)R antagonist. Studies revealed t
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2b673ef244e177a5845a09fa10895219
http://hdl.handle.net/11585/756673
http://hdl.handle.net/11585/756673
Autor:
Alexander Schmid, Diana Celona, Markus Müller, Andreas Krcal, Kurt Kletter, Aiman Abrahim, Oliver Langer, Dirk Roeda, Patrizia Minetti, Frédéric Dollé
Publikováno v:
Journal of Labelled Compounds and Radiopharmaceuticals. 48:577-587
1,1′-Methylene-di-(2-naphthol) (ST1859), a candidate drug for the treatment of Alzheimer's disease, was radiolabelled with carbon-11 with the aim to perform PET microdosing studies in humans. The radiosynthesis was automated in a commercial synthes
Autor:
Filomena Fezza, Stefania Butini, Giuseppe Borrelli, Stefano Di Serio, Silvia Vincenti, Antonio Caprioli, Samuele Maramai, Giuseppe Campiani, Mauro Maccarrone, Grazia Gallo, Margherita Brindisi, Sandra Gemma, Walter Cabri, Emanuela Talamonti, Sindu Ros, Franco Borsini, Patrizia Minetti, Maria Antonietta Stasi
Fatty acid amide hydrolase (FAAH, EC 3.5.1.99) is the main enzyme catabolizing endocannabinoid fatty acid amides. FAAH inactivation promotes beneficial effects upon pain and anxiety without the side effects accompanying agonists of type-1 cannabinoid
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2ff2174021bc05c27c215f18d35616fc
http://hdl.handle.net/11697/155949
http://hdl.handle.net/11697/155949