Zobrazeno 1 - 3
of 3
pro vyhledávání: '"Paolo G. Cassarà"'
Autor:
Aldo Feriani, Karen L Roberts, Beatrice Oliosi, Giovanna Tedesco, Robert J. Barnaby, Carla Marchioro, Maria Elvira Tranquillini, Paolo G. Cassarà, A. Ursini, Franciscus T.M. van Amsterdam, Angelo Reggiani, Mauro Corsi, S. Polinelli, Emiliangelo Ratti, Daniele Donati, Giovanni Curotto, David G. Trist, Daniela Niccolai, Gabriella Finizia
Publikováno v:
Bioorganic & Medicinal Chemistry. 19:4257-4273
This article deals with the synthesis and the activities of some 1,5-dialkyl-3-arylureido-1,5-benzodiazepin-2,4-diones which were prepared as potential CCK2 antagonists, with the intention to find a possible follow up of our lead compound GV150013, s
Autor:
Gabriella Finizia, Daniele Donati, Paolo G. Cassarà, A. Ursini, Giovanni Curotto, S. Polinelli, Giorgio Tarzia, F. T. M. Van Amsterdam, Giorgio Pentassuglia, Mauro Corsi, Maria Elvira Tranquillini
Publikováno v:
Archiv der Pharmazie. 330:353-357
The synthesis and biological evaluation as potential CCK-B receptor ligands of a number of 1-isopentyl-3-aryloxycarbamoyl-5-aryl-1,5-benzodiazepines substituted with halogen atoms on the benzo-fused ring is here briefly discussed.
Autor:
Bruce D. Dorsey, Mohamed Iqbal, Sankar Chatterjee, Bruce Ruggeri, Mark A. Ator, Michael Williams, John P. Mallamo, Ernesto Menta, Raffaella Bernardini, Alberto Bernareggi, Paolo G. Cassarà, Germano D’Arasmo, Edmondo Ferretti, Sergio De Munari, Ambrogio Oliva, Gabriella Pezzoni, Cecilia Allievi, Ivan Strepponi
Publikováno v:
Journal of Medicinal Chemistry; Jan2008, Vol. 51 Issue 4, p1068-1072, 5p