Zobrazeno 1 - 10
of 284
pro vyhledávání: '"Paolo, Grieco"'
Autor:
Rosa Bellavita, Annarita Falanga, Francesco Merlino, Gabriella D’Auria, Nicola Molfetta, Anella Saviano, Francesco Maione, Umberto Galdiero, Maria Rosaria Catania, Stefania Galdiero, Paolo Grieco, Emanuela Roscetto, Lucia Falcigno, Elisabetta Buommino
Publikováno v:
Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 38, Iss 1, Pp 36-50 (2023)
The increasing resistance of fungi to conventional antifungal drugs has prompted worldwide the search for new compounds. In this work, we investigated the antifungal properties of acylated Temporin L derivatives, Pent-1B and Dec-1B, against Candida a
Externí odkaz:
https://doaj.org/article/39c43ad04aa145468deb70d283b01f6c
Autor:
Maria Consiglia Trotta, Carlo Gesualdo, Caterina Claudia Lepre, Marina Russo, Franca Ferraraccio, Iacopo Panarese, Ernesto Marano, Paolo Grieco, Francesco Petrillo, Anca Hermenean, Francesca Simonelli, Michele D’Amico, Claudio Bucolo, Francesca Lazzara, Filomena De Nigris, Settimio Rossi, Chiara Bianca Maria Platania
Publikováno v:
Frontiers in Pharmacology, Vol 15 (2024)
Introduction:The purine analog 6-thioguanine (6TG), an old drug approved in the 60s to treat acute myeloid leukemia (AML), was tested in the diabetic retinopathy (DR) experimental in vivo setting along with a molecular modeling approach.Methods:A com
Externí odkaz:
https://doaj.org/article/ce3089b4c44f4ef1bee2c74f13fa2c5b
Autor:
Alessandra Ottani, Maria Galantucci, Ettore Ardimento, Laura Neri, Fabrizio Canalini, Anita Calevro, Davide Zaffe, Ettore Novellino, Paolo Grieco, Daniela Giuliani, Salvatore Guarini
Publikováno v:
Pharmacological Research, Vol 194, Iss , Pp 106852- (2023)
Externí odkaz:
https://doaj.org/article/5bf61ff30f0e4903a71d09fabbaf3e90
Autor:
Roberta Pacifico, Nunzio Del Gaudio, Guglielmo Bove, Lucia Altucci, Lydia Siragusa, Gabriele Cruciani, Menotti Ruvo, Rosa Bellavita, Paolo Grieco, Mauro F. A. Adamo
Publikováno v:
Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 37, Iss 1, Pp 1987-1994 (2022)
We have recently developed a new synthetic methodology that provided both N-aryl-5-hydroxytriazoles and N-pyridine-4-alkyl triazoles. A selection of these products was carried through virtual screening towards targets that are contemporary and valida
Externí odkaz:
https://doaj.org/article/f9c5fcf1b41543b299f0dd8f3efb65c3
Autor:
Alessandro Ottaiano, Roberta Penta de Vera d’Aragona, Anna Maria Trotta, Mariachiara Santorsola, Maria Napolitano, Giosuè Scognamiglio, Fabiana Tatangelo, Paolo Grieco, Silvia Zappavigna, Vincenza Granata, Francesco Perri, Amalia Luce, Giovanni Savarese, Monica Ianniello, Marika Casillo, Nadia Petrillo, Andrea Belli, Francesco Izzo, Guglielmo Nasti, Michele Caraglia, Stefania Scala
Publikováno v:
Frontiers in Immunology, Vol 13 (2022)
BackgroundWe previously reported rare regressive genetic trajectories of KRAS pathogenic mutations as a specific hallmark of the genuine oligometastatic status in colorectal cancer (CRC).MethodsSurvival and prognostic impact of disease extent in 140
Externí odkaz:
https://doaj.org/article/5bcd4ae119204d419da8f4d9556a1316
Autor:
Rosa Bellavita, Annarita Falanga, Elisabetta Buommino, Francesco Merlino, Bruno Casciaro, Floriana Cappiello, Maria Luisa Mangoni, Ettore Novellino, Maria Rosaria Catania, Rossella Paolillo, Paolo Grieco, Stefania Galdiero
Publikováno v:
Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 35, Iss 1, Pp 1751-1764 (2020)
The rapid development of antimicrobial resistance is pushing the search in the discovering of novel antimicrobial molecules to prevent and treat bacterial infections. Self-assembling antimicrobial peptides, as the lipidated peptides, are a novel and
Externí odkaz:
https://doaj.org/article/fbb519ebab4547f6a5bf64777c38cefb
Autor:
Carlo Gesualdo, Cornel Balta, Chiara Bianca Maria Platania, Maria Consiglia Trotta, Hildegard Herman, Sami Gharbia, Marcel Rosu, Francesco Petrillo, Salvatore Giunta, Alberto Della Corte, Paolo Grieco, Rosa Bellavita, Francesca Simonelli, Michele D’Amico, Anca Hermenean, Settimio Rossi, Claudio Bucolo
Publikováno v:
Frontiers in Pharmacology, Vol 12 (2021)
This study aimed to investigate the interactions between fingolimod, a sphingosine 1-phosphate receptor (S1PR) agonist, and melanocortin receptors 1 and 5 (MCR1, MCR5). In particular, we investigated the effects of fingolimod, a drug approved to trea
Externí odkaz:
https://doaj.org/article/8e236853c3f9447d8a2332342fb239dd
Autor:
Rosa Bellavita, Elisabetta Buommino, Bruno Casciaro, Francesco Merlino, Floriana Cappiello, Noemi Marigliano, Anella Saviano, Francesco Maione, Rosaria Santangelo, Maria Luisa Mangoni, Stefania Galdiero, Paolo Grieco, Annarita Falanga
Publikováno v:
Antibiotics, Vol 11, Iss 10, p 1285 (2022)
Temporin family is one of the largest among antimicrobial peptides (AMPs), which act mainly by penetrating and disrupting the bacterial membranes. To further understand the relationship between the physical-chemical properties and their antimicrobial
Externí odkaz:
https://doaj.org/article/cf5b7be86c234404a635bcda627218ea
Autor:
Grazia Bencivenni, Nathalie Saraiva Rosa, Paolo Grieco, Malachi W. Gillick-Healy, Brian G. Kelly, Brendan Twamley, Mauro F. A. Adamo
Publikováno v:
Catalysts, Vol 12, Iss 7, p 803 (2022)
We report herein sharp physical evidence, i.e., single-crystal X-ray diffraction and 1H-NMR spectral data, confirming that quaternary ammonium species interact with anions via a set of directional ion–dipole cooperative +N-C-H unusual H-bonding int
Externí odkaz:
https://doaj.org/article/5b420020620c4a358ad4f28358fdf0a8
Autor:
Carla Zannella, Annalisa Chianese, Luciana Palomba, Maria Elena Marcocci, Rosa Bellavita, Francesco Merlino, Paolo Grieco, Veronica Folliero, Anna De Filippis, Marialuisa Mangoni, Lucia Nencioni, Gianluigi Franci, Massimiliano Galdiero
Publikováno v:
International Journal of Molecular Sciences, Vol 23, Iss 4, p 2060 (2022)
The COVID-19 pandemic has evidenced the urgent need for the discovery of broad-spectrum antiviral therapies that could be deployed in the case of future emergence of novel viral threats, as well as to back up current therapeutic options in the case o
Externí odkaz:
https://doaj.org/article/45b4ad711f0241e494deb9f40a506a0d