Octreotide Conjugates for Tumor Targeting and Imaging

Autor: Eduard Figueras, Ana Martins, Adina Borbély, Vadim Le Joncour, Paola Cordella, Raffaella Perego, Daniela Modena, Paolo Pagani, Simone Esposito, Giulio Auciello, Marcel Frese, Paola Gallinari, Pirjo Laakkonen, Christian Steinkühler, Norbert Sewald

Publikováno v: Pharmaceutics, Vol 11, Iss 5, p 220 (2019)

Tumor targeting has emerged as an advantageous approach to improving the efficacy and safety of cytotoxic agents or radiolabeled ligands that do not preferentially accumulate in the tumor tissue. The somatostatin receptors (SSTRs) belong to the G-pro

Externí odkaz: https://doaj.org/article/04c4cbe3d3224ffab4063a1f948b8f66

Conjugates of Cryptophycin and RGD or isoDGR Peptidomimetics for Targeted Drug Delivery

Autor: Adina Borbély, Dr. Eduard Figueras, Ana Martins, Dr. Lizeth Bodero, Dr. André Raposo Moreira Dias, Dr. Paula López Rivas, Dr. Arianna Pina, Dr. Daniela Arosio, Dr. Paola Gallinari, Dr. Marcel Frese, Dr. Christian Steinkühler, Prof. Dr. Cesare Gennari, Prof. Dr. Umberto Piarulli, Prof. Dr. Norbert Sewald

Publikováno v: ChemistryOpen, Vol 8, Iss 6, Pp 737-742 (2019)

Abstract RGD‐cryptophycin and isoDGR‐cryptophycin conjugates were synthetized by combining peptidomimetic integrin ligands and cryptophycin, a highly potent tubulin‐binding antimitotic agent across lysosomally cleavable Val‐Ala or uncleavable

Externí odkaz: https://doaj.org/article/d3a79dc0bab74335b6cc1b9cbbeb2934

Supplementary Table 1 from Loss of Histone Deacetylase 4 Causes Segregation Defects during Mitosis of p53-Deficient Human Tumor Cells

Autor: Gessica Filocamo, Christian Steinkühler, Raffaele De Francesco, Paola Gallinari, Claudio Dello Russo, Emanuele de Rinaldis, Silvia Fedeli, Sabina Coppari, Mirko Brunetti, Bruno Cadot

Supplementary Table 1 from Loss of Histone Deacetylase 4 Causes Segregation Defects during Mitosis of p53-Deficient Human Tumor Cells

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::06c90259f3a23fa4707b75dadedb6c77
https://doi.org/10.1158/0008-5472.22378029

Supplementary Figure 2 from Loss of Histone Deacetylase 4 Causes Segregation Defects during Mitosis of p53-Deficient Human Tumor Cells

Autor: Gessica Filocamo, Christian Steinkühler, Raffaele De Francesco, Paola Gallinari, Claudio Dello Russo, Emanuele de Rinaldis, Silvia Fedeli, Sabina Coppari, Mirko Brunetti, Bruno Cadot

Supplementary Figure 2 from Loss of Histone Deacetylase 4 Causes Segregation Defects during Mitosis of p53-Deficient Human Tumor Cells

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::49e881e1aa242905c41f37bfd67ddde0
https://doi.org/10.1158/0008-5472.22378041.v1

Conjugates of Cryptophycin and RGD or isoDGR Peptidomimetics for Targeted Drug Delivery

Autor: Paula López Rivas, Eduard Figueras, Paola Gallinari, Umberto Piarulli, Cesare Gennari, Daniela Arosio, Marcel Frese, Arianna Pina, Ana Martins, Lizeth Bodero, Adina Borbély, Norbert Sewald, André Raposo Moreira Dias, Christian Steinkühler

Publikováno v: ChemistryOpen 8 (2019): 737–742. doi:10.1002/open.201900110
info:cnr-pdr/source/autori:Borbély, Adina; Figueras, Eduard; Martins, Ana; Bodero, Lizeth; Raposo Moreira Dias, André; López Rivas, Paula; Pina, Arianna; Arosio, Daniela; Gallinari, Paola; Frese, Marcel; Steinkühler, Christian; Gennari, Cesare; Piarulli, Umberto; Sewald, Norbert/titolo:Conjugates of Cryptophycin and RGD or isoDGR Peptidomimetics for Targeted Drug Delivery/doi:10.1002%2Fopen.201900110/rivista:ChemistryOpen/anno:2019/pagina_da:737/pagina_a:742/intervallo_pagine:737–742/volume:8
ChemistryOpen, Vol 8, Iss 6, Pp 737-742 (2019)
ChemistryOpen

RGD-cryptophycin and isoDGR-cryptophycin conjugates were synthetized by combining peptidomimetic integrin ligands and cryptophycin, a highly potent tubulin-binding antimitotic agent across lysosomally cleavable Val-Ala or uncleavable linkers. The con

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::9b5f6b95347262e1abd4af16e58236b7
https://publications.cnr.it/doc/405120