Zobrazeno 1 - 10
of 16
pro vyhledávání: '"Pakamas Tongcharoensirikul"'
Autor:
Timothy A. Coulther, David Labaree, Jessa L. Silver, Robert Dilis, Edward Hua, Richard B. Hochberg, Emmett McCaskill, Robert N. Hanson, Mary Jo Ondrechen, Pakamas Tongcharoensirikul
Publikováno v:
Steroids. 144:15-20
A series consisting of substituted benzoylbenzamide derivatives of 17α-E-vinyl estradiol 6a-i and 7a-d was prepared in good overall yields from the corresponding novel iodinated benzoylbenzamide precursors using Pd(0)-catalyzed Stille coupling. Biol
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::bd16f6deaa0e9a5ccb0c5f49b75c6cfc
https://doi.org/10.1016/j.steroids.2019.02.003
https://doi.org/10.1016/j.steroids.2019.02.003
Autor:
Kelton Barnsley, Robert N. Hanson, Mary Jo Ondrechen, Eugene R. DeSombre, Alun Hughes, Pakamas Tongcharoensirikul
Publikováno v:
Steroids. 96:50-62
A series of three 1,1-bis(4-hydroxyphenyl)-2-(3-hydroxyphenyl)-ethylene derivatives was prepared and evaluated as potential estrogen receptor imaging agents. The compounds display high binding affinity compared to estradiol, with the 2-iodo and 2-bro
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::aa49a86722fa343f0b8eb067462724c8
https://doi.org/10.1016/j.steroids.2015.01.013
https://doi.org/10.1016/j.steroids.2015.01.013
Autor:
Robert Dilis, Emmett McCaskill, David Labaree, Robert N. Hanson, Pakamas Tongcharoensirikul, Richard B. Hochberg
Publikováno v:
Steroids. 77:471-476
As part of our program to explore the influence of small structural modifications on the biological response of the estrogen receptor-α (ERα), we prepared and evaluated a series of mono-and di-substituted phenyl vinyl estradiols. The target compoun
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a9e2a36dbf45d8de5937d49724e7a65c
https://doi.org/10.1016/j.steroids.2012.01.003
https://doi.org/10.1016/j.steroids.2012.01.003
Publikováno v:
The Journal of Organic Chemistry. 69:2322-2326
Dimethyl thiophosphite (DMTP) was synthesized from dimethyl phosphite, and the diastereoselective addition of DMTP to benzaldimines bearing chiral auxiliary groups was examined. Yields of the product alpha-aminophosphonothionates ranged from 17% to 7
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8a4f5b7b77c30e217839e19734199bd1
https://doi.org/10.1021/jo035707t
https://doi.org/10.1021/jo035707t
Autor:
R D Bartlett, Charles M. Thompson, Christina N. Carrigan, C. Sean Esslinger, Kimberly A. Cybulski, Richard J. Bridges, Pakamas Tongcharoensirikul
Publikováno v:
Journal of Medicinal Chemistry. 45:2260-2276
The vesicular glutamate transport (VGLUT) system selectively mediates the uptake of L-glutamate into synaptic vesicles. Uptake is linked to an H+-ATPase that provides coupling among ATP hydrolysis, an electrochemical proton gradient, and glutamate tr
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7ccbce1756fca085e3110fe9962c1bbf
https://doi.org/10.1021/jm010261z
https://doi.org/10.1021/jm010261z
Autor:
Charles M. Thompson, Pakamas Tongcharoensirikul, Jeffrey Trautmann, Alírica I. Suárez, Gregory W. Muth
Publikováno v:
Phosphorus, Sulfur, and Silicon and the Related Elements. 177:471-477
Dimethyl thiophosphite reacts with aliphatic aldehydes and ketones, Michael acceptors, and N-benzyl imines to afford excellent yields of f -hydroxy phosphonothionates, g -substituted phosphonothionates and f -amino phosphonothionates, respectively. D
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::9dba4bc168920ef53aac8e4cd1579ed4
https://doi.org/10.1080/10426500210253
https://doi.org/10.1080/10426500210253
Publikováno v:
The Journal of Organic Chemistry. 65:3626-3632
5-Phenylisothiazole undergoes phototransposition via the electrocyclic ring closure-heteroatom migration pathway and by the N(2)-C(3) interchange reaction pathway. The latter route is enhanced by the addition of triethylamine (TEA) to the reaction me
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ffba7b86e5247094ff05a3384b7b4b9e
https://doi.org/10.1021/jo991785y
https://doi.org/10.1021/jo991785y
Publikováno v:
The Journal of Organic Chemistry. 63:5592-5603
Upon irradiation in the presence of a small quantity of base, 4-substituted isothiazoles undergo photocleavage to yield substituted cyanosulfides, which can be trapped as their benzyl thioether derivatives, and substituted isocyanosulfides. Both prod
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::9d4dc20cc3472afb451889dcec99dc4f
https://doi.org/10.1021/jo980936e
https://doi.org/10.1021/jo980936e
Autor:
Richard B. Hochberg, David Labaree, Sandra L. Olmsted, Karla Gandiaga, Pakamas Tongcharoensirikul, Emmett McCaskill, Robert N. Hanson
Publikováno v:
ChemInform. 43
A series of 17α-(heteroaryl)vinyl estradiols (III) is synthesized to evaluate the influence of heteroatom on the affinity and efficacy of estrogenic ligands for the estrogen receptor-alpha ligand binding domain.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::b1a53276ffc805a9c3cc7424c8f703d8
https://doi.org/10.1002/chin.201242199
https://doi.org/10.1002/chin.201242199
Publikováno v:
Journal of the American Chemical Society. 116:2292-2300
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::c686c63cee93362d23a40ae33bfda48c
https://doi.org/10.1021/ja00085a008
https://doi.org/10.1021/ja00085a008