Zobrazeno 1 - 10
of 21
pro vyhledávání: '"Pål, Rongved"'
Publikováno v:
Beilstein Journal of Organic Chemistry, Vol 15, Iss 1, Pp 2156-2160 (2019)
We present a short and efficient way of synthesizing two synthetically versatile 4-quinolone-3-carboxylate building blocks by cyclopropanation-ring expansion of 3-chloroindoles with α-halodiazoacetates as the key step. This novel transformation was
Externí odkaz:
https://doaj.org/article/2e452eae7e684699a5f7a7757958d459
Autor:
Samar Issa, Anthony Prandina, Nicolas Bedel, Pål Rongved, Saïd Yous, Marc Le Borgne, Zouhair Bouaziz
Publikováno v:
Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 34, Iss 1, Pp 1321-1346 (2019)
For over half a century, the carbazole skeleton has been the key structural motif of many biologically active compounds including natural and synthetic products. Carbazoles have taken an important part in all the existing anti-cancer drugs because of
Externí odkaz:
https://doaj.org/article/b6722b80ea7e4f35b7f6658a192d0578
Autor:
Anthony Prandina, Lars Herfindal, Sylvie Radix, Pål Rongved, Stein O. Døskeland, Marc Le Borgne, Florent Perret
Publikováno v:
Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 33, Iss 1, Pp 370-375 (2018)
Phenazine is known to regroup planar nitrogen-containing heterocyclic compounds. It was used here to enhance the bioavailability of the biologically important compound iodinin, which is near insoluble in aqueous solutions. Its water solubility has le
Externí odkaz:
https://doaj.org/article/f8efd2d694984d28a404868dc1bc4ce7
Autor:
Fatema Rahman, Imin Wushur, Nabin Malla, Ove Alexander Høgmoen Åstrand, Pål Rongved, Jan-Olof Winberg, Ingebrigt Sylte
Publikováno v:
Molecules, Vol 27, Iss 1, p 56 (2021)
Inhibition of bacterial virulence is believed to be a new treatment option for bacterial infections. In the present study, we tested dipicolylamine (DPA), tripicolylamine (TPA), tris pyridine ethylene diamine (TPED), pyridine and thiophene derivative
Externí odkaz:
https://doaj.org/article/82d8428881e047cba6314decdca3320b
Autor:
Christine Olsen, Frøydis Sved Skottvoll, Ole Kristian Brandtzaeg, Christian Schnaars, Pål Rongved, Elsa Lundanes, Steven Ray Wilson
Publikováno v:
Frontiers in Chemistry, Vol 7 (2019)
Prior to mass spectrometry, on-line sample preparation can be beneficial to reduce manual steps, increase speed, and enable analysis of limited sample amounts. For example, bottom-up proteomics sample preparation and analysis can be accelerated by di
Externí odkaz:
https://doaj.org/article/f2206022749244db81d6728fd767713f
Autor:
Elvar Ørn Viktorsson, Ove Alexander Høgmoen Åstrand, Rasha Sabah Haseeb, Carl Henrik Görbitz, Pål Rongved
Publikováno v:
Acta Crystallographica Section E: Crystallographic Communications, Vol 71, Iss 3, Pp 275-277 (2015)
The literature compound 3β-hydroxy-bisnor-5-cholenic aldehyde is an important intermediate for the synthesis of new modulators of the nuclear oxysterol receptor Liver X. As part of our ongoing search for new LXR antagonists, the title compound, C24H
Externí odkaz:
https://doaj.org/article/2fda1afcf24b48d0acb33685cf62a3ab
Publikováno v:
Molecules, Vol 15, Iss 9, Pp 6638-6677 (2010)
Applications of ring-closing alkene metathesis (RCM) in acyclic α- and β-peptides and closely related systems are reviewed, with a special emphasis on the structural and pharmacological effects of cyclization by RCM.
Externí odkaz:
https://doaj.org/article/242fa582408245af94d352776358700d
Publikováno v:
Acta Crystallographica Section E, Vol 69, Iss 2, Pp m112-m113 (2013)
In the title salt, [Zn(C22H24N4O)(CH3CN)][Zn(ClO4)(C22H24N4O)(CH3CN)](ClO4)3, two differently coordinated zinc cations occur. In the first complex, the metal ion is coordinated by the N,N′,N′′,O-tetradentate acetamide ligand and an acetonitrile
Externí odkaz:
https://doaj.org/article/50941bbc18824ed98d20dd3cd0cf5842
Autor:
Elvar Ørn Viktorsson, Ove Alexander Høgmoen Åstrand, Rasha Sabah Haseeb, Carl Henrik Görbitz, Pål Rongved
Publikováno v:
Acta Crystallographica Section E: Crystallographic Communications, Vol 71, Iss 3, Pp 275-277 (2015)
The literature compound 3[beta]-hydroxy-bisnor-5-cholenic aldehyde is an important intermediate for the synthesis of new modulators of the nuclear oxysterol receptor Liver X. As part of our ongoing search for new LXR antagonists, the title comp
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=dedup_wf_001::246a582cc9da93800af2e8fd1b17801f
http://hdl.handle.net/10852/58867
http://hdl.handle.net/10852/58867
Autor:
Elvar Ørn, Viktorsson, Ove Alexander Høgmoen, Åstrand, Rasha Sabah, Haseeb, Carl Henrik, Görbitz, Pål, Rongved
Publikováno v:
Acta Crystallographica Section E: Crystallographic Communications
In research towards new antagonists against the Liver X receptor, the important intermediate Fernholz acid Weinreb amide has been synthesized and characterized.
The literature compound 3β-hydroxy-bisnor-5-cholenic aldehyde is an important
The literature compound 3β-hydroxy-bisnor-5-cholenic aldehyde is an important