Zobrazeno 1 - 10
of 33
pro vyhledávání: '"Osama I, Alwassil"'
Publikováno v:
Humanities & Social Sciences Communications, Vol 11, Iss 1, Pp 1-8 (2024)
Abstract Medicinal chemistry educators face challenges in providing students with essential tools to ensure an ideal learning environment. The suspension of on-site classes during the COVID-19 pandemic introduced further obstacles. This study investi
Externí odkaz:
https://doaj.org/article/20616bcec18548e1a39c3e15933b6856
Autor:
Katharigatta N. Venugopala, Sandeep Chandrashekharappa, Christophe Tratrat, Pran Kishore Deb, Rahul D. Nagdeve, Susanta K. Nayak, Mohamed A. Morsy, Pobitra Borah, Fawzi M. Mahomoodally, Raghu Prasad Mailavaram, Mahesh Attimarad, Bandar E. Aldhubiab, Nagaraja Sreeharsha, Anroop B. Nair, Osama I. Alwassil, Michelyne Haroun, Viresh Mohanlall, Pottathil Shinu, Rashmi Venugopala, Mahmoud Kandeel, Belakatte P. Nandeshwarappa, Yasmine F. Ibrahim
Publikováno v:
Molecules, Vol 26, Iss 12, p 3550 (2021)
The cyclooxygenase-2 (COX-2) enzyme is an important target for drug discovery and development of novel anti-inflammatory agents. Selective COX-2 inhibitors have the advantage of reduced side-effects, which result from COX-1 inhibition that is usually
Externí odkaz:
https://doaj.org/article/a93033df97874456b6deecfd06366840
Publikováno v:
PLoS ONE, Vol 14, Iss 10, p e0223413 (2019)
Neisseria meningitidis is the primary cause of bacterial meningitis in many parts of the world, with considerable mortality rates among neonates and adults. In Saudi Arabia, serious outbreaks of N. meningitidis affecting several hundreds of pilgrims
Externí odkaz:
https://doaj.org/article/c0b392a7d8ed441fb04b645f6be68ba2
Autor:
Katharigatta N. Venugopala, Mohammed A. Khedr, Yarabahally R. Girish, Subhrajyoti Bhandary, Deepak Chopra, Mohamed A. Morsy, Bandar E. Aldhubiab, Pran Kishore Deb, Mahesh Attimarad, Anroop B. Nair, Nagaraja Sreeharsha, Rashmi V, Mahmoud Kandeel, Sabah H. Akrawi, Madhusudana Reddy M B, Sheena Shashikanth, Osama I. Alwassil, Viresh Mohanlall
Publikováno v:
Antibiotics, Vol 9, Iss 6, p 350 (2020)
A series of 2,4,5 trisubstituted-1,2,3-triazole analogues have been screened for their antifungal activity against five fungal strains, Candida parapsilosis, Candida albicans, Candida tropicalis, Aspergillus niger, and Trichophyton rubrum, via a 3-[4
Externí odkaz:
https://doaj.org/article/ad540e01a94d4a088b8f1a757c24e83c
Autor:
Katharigatta N. Venugopala, Pushpalatha Ramachandra, Christophe Tratrat, Raquel M. Gleiser, Subhrajyoti Bhandary, Deepak Chopra, Mohamed A. Morsy, Bandar E. Aldhubiab, Mahesh Attimarad, Anroop B. Nair, Nagaraja Sreeharsha, Rashmi Venugopala, Pran Kishore Deb, Sandeep Chandrashekharappa, Hany Ezzat Khalil, Osama I. Alwassil, Sara Nidal Abed, Yazan A. Bataineh, Ramachandra Palenge, Michelyne Haroun, Shinu Pottathil, Meravanige B. Girish, Sabah H. Akrawi, Viresh Mohanlall
Publikováno v:
Molecules, Vol 25, Iss 6, p 1316 (2020)
Malaria, affecting all continents, remains one of the life-threatening diseases introduced by parasites that are transmitted to humans through the bites of infected Anopheles mosquitoes. Although insecticides are currently used to reduce malaria tran
Externí odkaz:
https://doaj.org/article/37b7430a0c384986a7049bc93f211b1e
Autor:
Deepak Chopra, Rohit Bhowal, Keshab M. Bairagi, Avantika Hasija, Osama I. Alwassil, Smital A. Mohurle, Katharigatta N. Venugopala, Susanta K. Nayak, Kapil S. Ingle
Publikováno v:
ChemPlusChem. 86:1167-1176
A solvent-assisted grinding method has been used to prepare co-crystals in substituted dihydropyrimidines (DHPM) that constitutes pharmacologically active compounds. These were characterized using FT-IR, PXRD, and single-crystal X-ray diffraction. In
Autor:
Osama I. Alwassil, Marvin K. Schulte, Sanjay S Aripaka, Malgorzata Dukat, Jens D. Mikkelsen, Shailesh Khatri
Publikováno v:
ACS Chemical Neuroscience. 12:2194-2201
We previously reported that N-(3-chlorophenyl)guanidine (1) represents a novel α7 nicotinic ACh (nACh) receptor antagonist chemotype. In the present study, a small series of compounds was synthesized with the intent to investigate the structure-acti
Autor:
Katharigatta N. Venugopala, Omar H.A. Al-Attraqchi, Christophe Tratrat, Susanta K. Nayak, Mohamed A. Morsy, Bandar E. Aldhubiab, Mahesh Attimarad, Anroop B. Nair, Nagaraja Sreeharsha, Rashmi Venugopala, Michelyne Haroun, Meravanige B. Girish, Sandeep Chandrashekharappa, Osama I. Alwassil, Bharti Odhav
Publikováno v:
Biomolecules, Vol 9, Iss 11, p 661 (2019)
The cyclooxygenase-2 (COX-2) enzyme is considered to be an important target for developing novel anti-inflammatory agents. Selective COX-2 inhibitors offer the advantage of lower adverse effects that are commonly associated with non-selective COX inh
Externí odkaz:
https://doaj.org/article/9599fd4cb793455fb3fcee7f328c1195
Autor:
Nancy S. Younis, Katharigatta N. Venugopala, Ekta Sangtani, Susanta K. Nayak, Hany Ezzat Khalil, Keshab M. Bairagi, Rajesh G. Gonnade, Promise Madu Emeka, Osama I. Alwassil
Publikováno v:
Medicinal Chemistry. 16:996-1003
Background: This research project is designed to identify the anti-diabetic effects of the newly synthesized compounds to conclude the perspective of consuming one or more of these new synthetic compounds for diabetes management. Introduction: A seri
Autor:
Osama I. Alwassil, Rashmi Venugopala, Vijayakumar Uppar, Supratik Kar, Sandeep Chandrashekharappa, Basavaraj Padmashali, Raquel M. Gleiser, Daniel A. García, Mahendra K. Mohan, Bharti Odhav, Pran Kishore Deb, Katharigatta N. Venugopala
Publikováno v:
Structural Chemistry. 31:1533-1543
Certain tetrahydropyrido[1,2-a]quinolines and pyrroloquinoline homologs have shown various biological activities such as antimicrobials, crop-protectings, diuretics, antioxidants, anticoagulants, and antimalarial activities. Keeping this observation