Zobrazeno 1 - 10
of 17
pro vyhledávání: '"Olga Wronikowska-Denysiuk"'
Autor:
Piotr Stępnicki, Olga Wronikowska-Denysiuk, Agata Zięba, Katarzyna M. Targowska-Duda, Agata Bartyzel, Martyna Z. Wróbel, Tomasz M. Wróbel, Klaudia Szałaj, Andrzej Chodkowski, Karolina Mirecka, Barbara Budzyńska, Emilia Fornal, Jadwiga Turło, Marián Castro, Agnieszka A. Kaczor
Publikováno v:
Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 38, Iss 1 (2023)
Schizophrenia is a chronic mental disorder that is not satisfactorily treated with available antipsychotics. The presented study focuses on the search for new antipsychotics by optimising the compound D2AAK3, a multi-target ligand of G-protein-couple
Externí odkaz:
https://doaj.org/article/7d0e4b8d609e40c3b4670a0604436c47
Autor:
Damian Bartuzi, Ewa Kędzierska, Katarzyna M. Targowska-Duda, Oliwia Koszła, Tomasz M. Wróbel, Simon Jademyr, Tadeusz Karcz, Katarzyna Szczepańska, Piotr Stępnicki, Olga Wronikowska-Denysiuk, Grażyna Biała, Jadwiga Handzlik, Jesper L. Kristensen, Antti Poso, Agnieszka A. Kaczor
Publikováno v:
Scientific Reports, Vol 12, Iss 1, Pp 1-14 (2022)
Abstract Anxiety is a troublesome symptom for many patients, especially those suffering from schizophrenia. Its regulation involves serotonin receptors, targeted e.g. by antipsychotics or psychedelics such as LSD. 5-HT2A receptors are known for an ex
Externí odkaz:
https://doaj.org/article/e8d54c16692c4f768e6532bff908e43f
Autor:
Justyna Socha, Pawel Grochecki, Irena Smaga, Joanna Jastrzębska, Olga Wronikowska-Denysiuk, Marta Marszalek-Grabska, Tymoteusz Slowik, Robert Kotlinski, Małgorzata Filip, Gert Lubec, Jolanta H. Kotlinska
Publikováno v:
International Journal of Molecular Sciences, Vol 25, Iss 2, p 1041 (2024)
Children with fetal alcohol spectrum disorders (FASDs) demonstrate deficits in social functioning that contribute to early withdrawal from school and delinquency, as well as the development of anxiety and depression. Dopamine is involved in reward, m
Externí odkaz:
https://doaj.org/article/605a9989d3534565bb7691298daa9613
Autor:
Olga Wronikowska-Denysiuk, Agnieszka Michalak, Anna Pankowska, Łukasz Kurach, Paulina Kozioł, Artur Łazorczyk, Katarzyna Kochalska, Katarzyna Targowska-Duda, Anna Boguszewska-Czubara, Barbara Budzyńska
Publikováno v:
International Journal of Molecular Sciences, Vol 24, Iss 12, p 9958 (2023)
Mephedrone is a psychoactive drug that increases dopamine, serotonin and noradrenaline levels in the central nervous system via interaction with transporters or monoamines. The aim of the presented study was to assess the role of the GABA-ergic syste
Externí odkaz:
https://doaj.org/article/b79e7d9e5b454c17ba8f4e98494560c4
Publikováno v:
Biomolecules, Vol 13, Iss 3, p 405 (2023)
Drug abuse is a worldwide problem that leads to negative physical, mental, and economic consequences. Although pharmacological strategies for drug addiction management have been widely studied, therapeutic options with high efficacy and a low side-ef
Externí odkaz:
https://doaj.org/article/92008e56e13f4ac6a794f82c4a4d20a7
Autor:
Łukasz Pecio, Solomiia Kozachok, Ion Brinza, Razvan Stefan Boiangiu, Lucian Hritcu, Cornelia Mircea, Ana Flavia Burlec, Oana Cioanca, Monica Hancianu, Olga Wronikowska-Denysiuk, Krystyna Skalicka-Woźniak, Wiesław Oleszek
Publikováno v:
Molecules, Vol 27, Iss 12, p 3692 (2022)
Y. schidigera contains a number of unusual polyphenols, derivatives of resveratrol and naringenin, called spiro-flavostilbenoids, which have potent in vitro anti-inflammatory, antioxidant, and moderate cholinesterase inhibitory activities. To date, t
Externí odkaz:
https://doaj.org/article/6d88ce63776340fd82ddc6b2f1583651
Autor:
Szymon Sip, Daria Szymanowska, Justyna Chanaj-Kaczmarek, Krystyna Skalicka-Woźniak, Barbara Budzyńska, Olga Wronikowska-Denysiuk, Tymoteusz Słowik, Piotr Szulc, Judyta Cielecka-Piontek
Publikováno v:
Antioxidants, Vol 11, Iss 2, p 380 (2022)
As a systemic disease, diabetes mellitus (DM) is characterized by the disruption of many glucose metabolic pathways. Therefore, it seems critical to study new therapies to support treatment to develop therapeutic systems that can operate across a bro
Externí odkaz:
https://doaj.org/article/9a3463651f2146238750b4f6aae1c595
Autor:
Budzyńska, Olga Wronikowska-Denysiuk, Agnieszka Michalak, Anna Pankowska, Łukasz Kurach, Paulina Kozioł, Artur Łazorczyk, Katarzyna Kochalska, Katarzyna Targowska-Duda, Anna Boguszewska-Czubara, Barbara
Publikováno v:
International Journal of Molecular Sciences; Volume 24; Issue 12; Pages: 9958
Mephedrone is a psychoactive drug that increases dopamine, serotonin and noradrenaline levels in the central nervous system via interaction with transporters or monoamines. The aim of the presented study was to assess the role of the GABA-ergic syste
Autor:
Magda Kondej, Tomasz M. Wróbel, Katarzyna M. Targowska‐Duda, Antón Leandro Martínez, Oliwia Koszła, Piotr Stępnicki, Agata Zięba, Alba Paz, Olga Wronikowska‐Denysiuk, Maria I. Loza, Marián Castro, Agnieszka A. Kaczor
Publikováno v:
ChemMedChem. 17(15)
Schizophrenia is a complex disease which is best treated with multitarget drugs, such as atypical antipsychotics. Previously, using structure-based virtual screening, we found a virtual hit, D2AAK1, with nanomolar affinity for dopamine and serotonin
Autor:
Piotr Stępnicki, Katarzyna M. Targowska-Duda, Antón L. Martínez, Agata Zięba, Olga Wronikowska-Denysiuk, Martyna Z. Wróbel, Agata Bartyzel, Alicja Trzpil, Tomasz M. Wróbel, Andrzej Chodkowski, Karolina Mirecka, Tadeusz Karcz, Katarzyna Szczepańska, Maria I. Loza, Barbara Budzyńska, Jadwiga Turło, Jadwiga Handzlik, Emilia Fornal, Ewa Poleszak, Marián Castro, Agnieszka A. Kaczor
Publikováno v:
European Journal of Medicinal Chemistry. 252:115285