Potent bradykinin B 1 receptor antagonists: 4-Substituted phenyl cyclohexanes

Autor: Su, Dai-Shi, Lim, John L., Markowitz, M. Kristine, Wan, Bang-Lin, Murphy, Kathy L., Reiss, Duane R., Harrell, C. Meacham, O’Malley, Stacy S., Ransom, Rick W., Chang, Raymond S.L., Pettibone, Douglas J., Tang, Cuyue, Prueksaritanont, Thomayant, Freidinger, Roger M., Bock, Mark G.

Publikováno v: In Bioorganic & Medicinal Chemistry Letters 2007 17(11):3006-3009

Development of an efficient and selective radioligand for bradykinin B 1 receptor occupancy studies

Autor: Su, Dai-Shi ^*, Markowitz, M. Kristine, Murphy, Kathy L., Wan, Bang-Lin, Zrada, Matthew M., Harrell, C. Meacham, O’Malley, Stacy S., Hess, J. Fred, Ransom, Rick W., Chang, Ray S., Wallace, Michael A., Raab, Conrad E., Dean, Dennis C., Pettibone, Douglas J., Freidinger, Roger M., Bock, Mark G.

Publikováno v: In Bioorganic & Medicinal Chemistry Letters 2004 14(24):6045-6048

Development of an efficient and selective radioligand for bradykinin B1 receptor occupancy studies

Autor: Su,, Dai-Shi¹ daishi_su@merck.com, Markowitz, M. Kristine¹, Murphy, Kathy L.², Wan, Bang-Lin¹, Zrada, Matthew M.¹, Harrell, C. Meacham², O’Malley, Stacy S.², Hess, J. Fred², Ransom, Rick W.², Chang, Ray S.², Wallace, Michael A.³, Raab, Conrad E.³, Dean, Dennis C.³, Pettibone, Douglas J.², Freidinger, Roger M.¹, Bock, Mark G.¹

Publikováno v: Bioorganic & Medicinal Chemistry Letters. Dec2004, Vol. 14 Issue 24, p6045-6048. 4p.

Discovery of a potent, non-peptide bradykinin B1 receptor antagonist.

Autor: Su DS; Departments of Medicinal Chemistry and Neuroscience, Merck Research Laboratories, West Point, PA 19486, USA. daishi_su@merck.com, Markowitz MK, DiPardo RM, Murphy KL, Harrell CM, O'Malley SS, Ransom RW, Chang RS, Ha S, Hess FJ, Pettibone DJ, Mason GS, Boyce S, Freidinger RM, Bock MG

Publikováno v: Journal of the American Chemical Society [J Am Chem Soc] 2003 Jun 25; Vol. 125 (25), pp. 7516-7.