Zobrazeno 1 - 10 of 89 pro vyhledávání: '"Nour-Eddine Aouf"'
1
Akademický článek
Synthesis, ADME/T, and Carbonic Anhydrase Binding of Hydroxycarboxamide Compounds
Autor: Abdeslem Bouzina, Yousra Ouafa Bouone, Rachida Mansouri, Nour-Eddine Aouf
Publikováno v: Medical Sciences Forum, Vol 14, Iss 1, p 6 (2022)
The interconversion of carbon dioxide and the bicarbonate ion is carried out by carbonic anhydrases (CA), which are ubiquitous metalloenzymes with Zn in their active site. Disorder of CA enzymes can cause several diseases such as glaucoma, epilepsy,
Externí odkaz: https://doaj.org/article/54d2a1154da9438da07c0cdbcd277b80
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2
Akademický článek
Synthesis, Molecular Docking Analysis, ADMET and Drug Likeness Prediction of a Benzenesulfonamide Derivative Analogue of SLC-0111
Autor: Yousra Ouafa Bouone, Abdeslem Bouzina, Nour-Eddine Aouf
Publikováno v: Medical Sciences Forum, Vol 14, Iss 1, p 24 (2022)
Carbonic anhydrases are metalloenzymes that regulate the interconversion of CO2 and H2CO3, a reaction involved in many physiological processes. A disfunction of these enzymes is known to induce many diseases such as glaucoma, epilepsy and cancer. As
Externí odkaz: https://doaj.org/article/469c4ef5efae416f86f1d023ac651aa2
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3
Akademický článek
Synthesis and antibacterial activity of novel N-acylsulfonamides
Autor: Malika Berredjem, Fouzia Bouchareb, Samira Ait Kaki, Maazouz Dekhil, Nour-Eddine Aouf
Publikováno v: Arabian Journal of Chemistry, Vol 10, Iss S1, Pp S1095-S1099 (2017)
A series of novel N-acylsulfonamide derivatives were synthesized and characterized by 1H NMR, 13C NMR and HRMS. The N-acylsulfonamides were prepared in four steps (carbamoylation, sulfamoylation, deprotection and acylation) starting from chlorosulfon
Externí odkaz: https://doaj.org/article/b2928a82757345ce932b387b9e9b36f4
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4
Akademický článek
A New Class of Heterocycles: 1,4,3,5-Oxathiadiazepane 4,4-dioxides
Autor: Amel Bendjeddou, Tahar Abbaz, Zine Regainia, Nour-Eddine Aouf
Publikováno v: Molecules, Vol 17, Iss 2, Pp 1890-1899 (2012)
This work reports the synthesis of novel 1,4,3,5-oxathiadiazepanes 4,4-dioxides from the reaction of N’-benzyl-N-(2-hydroxyethyl)-sarcosine or proline sulfamide with aromatic aldehydes under acid catalysis. To prepare the starting materials N-Boc-s
Externí odkaz: https://doaj.org/article/2e4bef1523ac429bad00e362a47e1f1c
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5
Akademický článek
1,2,3,4-Tetrahydroisoquinoline-2-sulfonamide
Autor: Carole Barbey, Nour-Eddine Aouf, Malika Berredjem, Radia Bouasla
Publikováno v: Acta Crystallographica Section E, Vol 64, Iss 2, Pp o432-o432 (2008)
The title compound, C9H12N2O2S, is a useful precursor of a variety of modified sulfonamide molecules. Due to the importance of these molecules in biological systems (antibacterials, antidepressants and many other applications), there is a growing int
Externí odkaz: https://doaj.org/article/7208cf89afc94347bbc68b2278ae5d4d
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6
Synthesis, in silico study, and biological evaluation of cyclosulfamide derivatives as new anticholinesterase inhibitors
Autor: Abdeslem Bouzina, Abdelhak Djemel, Omar Sekiou, Imededdine Kadi, Yousra Ouafa Bouone, Rachida Mansouri, Zineb Aouf, Malika Ibrahim-ouali, Nour Eddine Aouf
Publikováno v: Journal of Molecular Structure
Journal of Molecular Structure, 2023, pp.135527. ⟨10.1016/j.molstruc.2023.135527⟩
International audience; After the great spread of Alzheimer's disease (AD) in the past few years, many researchers directed their work toward developing an effective treatment for this disease and to discovering very advanced drugs. Cyclosulfamides a
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::98ea418ca94a9c309e590414fd2ea995
https://hal-amu.archives-ouvertes.fr/hal-04063526
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8
Novel pseudonucleosides and sulfamoyl-oxazolidinone β - D -glucosamine derivative as anti-COVID-19: design, synthesis, and in silico study
Autor: Rachida Mansouri, Abdeslem Bouzina, Omar Sekiou, Zineb Aouf, Rachida Zerrouki, Malika Ibrahim-ouali, Nour eddine Aouf
Publikováno v: Journal of Biomolecular Structure and Dynamics
Journal of Biomolecular Structure and Dynamics, 2023, pp.1-18. ⟨10.1080/07391102.2023.2203246⟩
New pseudonucleosides containing cyclic sulfamide moiety and sulfamoyl β-D-glucosamine derivative are described. These pseudonucleosides are synthesized in good yields starting from chlorosulfonyl isocyanate and β-D-glucosamine hydrochloride in fiv
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ebb62d74f8f7692040c4f4f97a79780c
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9
A new family of sulfamidophosphonates derivatives: Microwave-accelerated multicomponent synthesis, characterization and X-Ray Crystallographic Study
Autor: Racha GHODBANE, Hacène K'TIR, sofiane BOUACIDA, malika ibrahim-ouali, zineb aouf, nour-eddine aouf
In this present study we describe a simple, effective and greener one-pot microwave-assisted synthesis of novel α-sulfamidophosphonates 4(a-n) that were rationally designed and synthesized following the principle of the superposition of bioactive su
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::ebf6eeca67b89f34da35402f85941af3
https://doi.org/10.21203/rs.3.rs-2232064/v1
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