Zobrazeno 1 - 2
of 2
pro vyhledávání: '"Norihito Ohi"'
Autor:
Fumihiro Ozaki, Osamu Takenaka, Atsushi Kamada, Kenzo Muramoto, Tetsuya Kawahara, Masayoshi Ohkuro, Richard Clark, Kazuo Okano, Norihito Ohi, Toshihiko Kaneko, Seiichi Kobayashi, Hiromitsu Yokohama
Publikováno v:
Chemicalpharmaceutical bulletin. 52(6)
Novel piperidine carboxylic acid derivatives of 10H-pyrazino[2,3-b][1,4]benzothiazine were prepared and evaluated for their inhibitory activity on the upregulation of adhesion molecules such as intercellular adhesion molecule-1 (ICAM-1). Replacement
Autor:
Fumihiro Ozaki, Osamu Takenaka, Kenzo Muramoto, Seiichi Kobayashi, Atsushi Kamada, Masayoshi Ohkuro, Toshihiko Kaneko, Hiroshi Akamatsu, Norihito Ohi, Richard Clark, Kazuo Okano, Tetsuya Kawahara, Hiromitsu Yokohama
Publikováno v:
Chemicalpharmaceutical bulletin. 50(7)
During a search for novel, orally-active inhibitors of upregulation of adhesion molecules such as intercellular adhesion molecule-1 (ICAM-1), we found a new series of 10H-pyrazino[2,3-b][1,4]benzothiazine derivatives to be potent ICAM-1 inhibitors. O