Zobrazeno 1 - 10
of 40
pro vyhledávání: '"Nobuaki Yasuo"'
Publikováno v:
ACS Omega, Vol 8, Iss 40, Pp 37431-37441 (2023)
Externí odkaz:
https://doaj.org/article/c4c3c5e823f44708b36c1ead9cc94806
Autor:
Han Xu, Ryo Nakayama, Takefumi Kimura, Ryota Shimizu, Yasunobu Ando, Shigeru Kobayashi, Nobuaki Yasuo, Masakazu Sekijima, Taro Hitosugi
Publikováno v:
Science and Technology of Advanced Materials: Methods, Vol 3, Iss 1 (2023)
Compared to the optimization of a 1D synthesis parameter in materials synthesis, the optimization of multi-dimensional synthesis parameters is challenging for researchers. Bayesian optimization (BO) has shown high performance in optimizing high-dimen
Externí odkaz:
https://doaj.org/article/5e00057767434578901ac1f3a4b327b4
Autor:
Ryo Nakayama, Ryota Shimizu, Taishi Haga, Takefumi Kimura, Yasunobu Ando, Shigeru Kobayashi, Nobuaki Yasuo, Masakazu Sekijima, Taro Hitosugi
Publikováno v:
Science and Technology of Advanced Materials: Methods, Vol 2, Iss 1, Pp 119-128 (2022)
Materials exploration requires the optimization of a multidimensional space including the chemical composition and synthesis parameters such as temperature and pressure. Bayesian optimization has attracted attention as a method for efficient multidim
Externí odkaz:
https://doaj.org/article/f6d489e50a724da3a4bfcd279db222a9
Publikováno v:
Journal of Cheminformatics, Vol 13, Iss 1, Pp 1-10 (2021)
Abstract The hit-to-lead process makes the physicochemical properties of the hit molecules that show the desired type of activity obtained in the screening assay more drug-like. Deep learning-based molecular generative models are expected to contribu
Externí odkaz:
https://doaj.org/article/25b685331a2b4355b8bd8e12c68c8c7d
Autor:
Kazuki Takeda, Kosuke Manago, Ayuko Morita, Yusuke K. Kawai, Nobuaki Yasuo, Masakazu Sekijima, Yoshinori Ikenaka, Takuma Hashimoto, Ryuichi Minato, Yusuke Oyamada, Kazuo Horikoshi, Hajime Suzuki, Mayumi Ishizuka, Shouta M.M. Nakayama
Publikováno v:
Ecotoxicology and Environmental Safety, Vol 243, Iss , Pp 113971- (2022)
Anticoagulant rodenticides have been widely used to eliminate wild rodents, which as invasive species on remote islands can disturb ecosystems. Since rodenticides can cause wildlife poisoning, it is necessary to evaluate the sensitivity of local mamm
Externí odkaz:
https://doaj.org/article/4d9296e3730d43039848894925e469d8
Autor:
Yu Miyazaki, Ryo Nakayama, Nobuaki Yasuo, Yuki Watanabe, Ryota Shimizu, Daniel M. Packwood, Kazunori Nishio, Yasunobu Ando, Masakazu Sekijima, Taro Hitosugi
Publikováno v:
AIP Advances, Vol 10, Iss 4, Pp 045231-045231-6 (2020)
AC impedance spectroscopy is an important method for evaluating ionic, electronic, and dielectric properties of materials. In conventional analysis of AC impedance spectra, the selection of an equivalent circuit model and its initial parameters are v
Externí odkaz:
https://doaj.org/article/80811188222b40dd97de2fcba27b2b72
Autor:
Ryunosuke Yoshino, Nobuaki Yasuo, Yohsuke Hagiwara, Takashi Ishida, Daniel Ken Inaoka, Yasushi Amano, Yukihiro Tateishi, Kazuki Ohno, Ichiji Namatame, Tatsuya Niimi, Masaya Orita, Kiyoshi Kita, Yutaka Akiyama, Masakazu Sekijima
Publikováno v:
Scientific Reports, Vol 7, Iss 1, Pp 1-9 (2017)
Abstract Chagas disease results from infection by Trypanosoma cruzi and is a neglected tropical disease (NTD). Although some treatment drugs are available, their use is associated with severe problems, including adverse effects and limited effectiven
Externí odkaz:
https://doaj.org/article/9864fe2ce67f43499bde2b3251ec52d6
Autor:
Ryunosuke Yoshino, Nobuaki Yasuo, Daniel Ken Inaoka, Yohsuke Hagiwara, Kazuki Ohno, Masaya Orita, Masayuki Inoue, Tomoo Shiba, Shigeharu Harada, Teruki Honma, Emmanuel Oluwadare Balogun, Josmar Rodrigues da Rocha, Carlos Alberto Montanari, Kiyoshi Kita, Masakazu Sekijima
Publikováno v:
PLoS ONE, Vol 10, Iss 5, p e0125829 (2015)
Chagas disease, caused by the parasite Trypanosoma cruzi, is a neglected tropical disease that causes severe human health problems. To develop a new chemotherapeutic agent for the treatment of Chagas disease, we predicted a pharmacophore model for T.
Externí odkaz:
https://doaj.org/article/4b0bac0f018a4bb7a714642595f2c480
Publikováno v:
Journal of Chemical Information and Modeling
In addition to vaccines, antiviral drugs are essential for suppressing COVID-19. Although several inhibitor candidates were reported for SARS-CoV-2 main protease, most are highly polar peptidomimetics with poor oral bioavailability and cell membrane
Publikováno v:
2022 IEEE 22nd International Conference on Bioinformatics and Bioengineering (BIBE).