Zobrazeno 1 - 4
of 4
pro vyhledávání: '"Niklas, Rosier"'
Autor:
Lukas Grätz, Jan Möller, Laura J Humphrys, Steffen Pockes, Ali Işbilir, Niklas Rosier, Martin J. Lohse, Hannes Schihada, Martin Nagl, Ulla Seibel
Publikováno v:
Journal of Medicinal Chemistry. 64:11695-11708
The histamine H3 receptor (H3R) is considered an attractive drug target for various neurological diseases. We here report the synthesis of UR-NR266, a novel fluorescent H3R ligand. Broad pharmacological characterization revealed UR-NR266 as a sub-nan
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::92f12c3455be4acdb437e98401731849
https://doi.org/10.1021/acs.jmedchem.1c01089
https://doi.org/10.1021/acs.jmedchem.1c01089
Autor:
Katarzyna Szczepańska, Sabina Podlewska, Maria Dichiara, Davide Gentile, Vincenzo Patamia, Niklas Rosier, Denise Mönnich, Ma Carmen Ruiz Cantero, Tadeusz Karcz, Dorota Łażewska, Agata Siwek, Steffen Pockes, Enrique J. Cobos, Agostino Marrazzo, Holger Stark, Antonio Rescifina, Andrzej J. Bojarski, Emanuele Amata, Katarzyna Kieć-Kononowicz
Publikováno v:
Digibug. Repositorio Institucional de la Universidad de Granada
instname
instname
We are pleased to acknowledge the generous support of the National Science Center, Poland, granted based on decision No. 2020/36/C/NZ7/00284. Support by ERNEST COST Action 18133 is also acknowledged. K. Szczepan ' ska is supported by the Foundation o
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::899d6f96dabb782c74c11794c8b27ca6
https://ruj.uj.edu.pl/xmlui/handle/item/286264
https://ruj.uj.edu.pl/xmlui/handle/item/286264
Autor:
Katarzyna, Szczepańska, Sabina, Podlewska, Maria, Dichiara, Davide, Gentile, Vincenzo, Patamia, Niklas, Rosier, Denise, Mönnich, Ma Carmen, Ruiz Cantero, Tadeusz, Karcz, Dorota, Łażewska, Agata, Siwek, Steffen, Pockes, Enrique J, Cobos, Agostino, Marrazzo, Holger, Stark, Antonio, Rescifina, Andrzej J, Bojarski, Emanuele, Amata, Katarzyna, Kieć-Kononowicz
Publikováno v:
ACS Chemical Neuroscience
In an attempt to extend recent studies showing that some clinically evaluated histamine H3 receptor (H3R) antagonists possess nanomolar affinity at sigma-1 receptors (σ1R), we selected 20 representative structures among our previously reported H3R l
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=pmid________::a7e5927b4895ade85a653b732c303e37
https://pubmed.ncbi.nlm.nih.gov/34908391
https://pubmed.ncbi.nlm.nih.gov/34908391
Autor:
Niklas, Rosier, Lukas, Grätz, Hannes, Schihada, Jan, Möller, Ali, Işbilir, Laura J, Humphrys, Martin, Nagl, Ulla, Seibel, Martin J, Lohse, Steffen, Pockes
Publikováno v:
Journal of medicinal chemistry. 64(15)
The histamine H
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=pmid________::70d784c26ad8231fa531b420cc9e178e
https://pubmed.ncbi.nlm.nih.gov/34309390
https://pubmed.ncbi.nlm.nih.gov/34309390