Zobrazeno 1 - 10
of 40
pro vyhledávání: '"Nicolino Pala"'
Autor:
Fabio Esposito, Nicolino Pala, Mauro Carcelli, Samuel T. Boateng, Paolo S. D’Aquila, Alberto Mariani, Sandro Satta, Jean Christopher Chamcheu, Mario Sechi, Vanna Sanna
Publikováno v:
Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 38, Iss 1 (2023)
Natural α-glucosidase inhibitors from plant-based foods such as catechins offer an attractive strategy for their potential anti-diabetic effects. In this study, infusions of three different tea types (green, white, and oolong) were investigated for
Externí odkaz:
https://doaj.org/article/a8426010c28e45e2be3e2b777b431689
Autor:
Mohamed F. Y. Gomaa, Nicolino Pala, Marco Derudas, Jehan Abd-Elrazik Hasanen, El-Sayed H. El-Tamany, Paola Casule, Alberto Mariani, Mario Sechi
Publikováno v:
ARKIVOC, Vol 2011, Iss 9, Pp 1-14 (2011)
Externí odkaz:
https://doaj.org/article/780e241310294e8da4f7aaa35a446632
Autor:
Nouri Neamati, Nicolino Pala, Alessia Cosseddu, Alessandro Dessì, Roberto Dallocchio, Maria Paola Delussu, Ugo Azzena, Mario Sechi
Publikováno v:
Molecules, Vol 13, Iss 10, Pp 2442-2461 (2008)
HIV-1 integrase (IN) is an attractive and validated target for the development of novel therapeutics against AIDS. In the search for new IN inhibitors, we designed and synthesized three series of bis-amide and hydrazide-containing derivatives of malo
Externí odkaz:
https://doaj.org/article/2d98ce6a06194834814132d957c3fd14
Autor:
Nicolino Pala, Francesca Esposito, Dominga Rogolino, Mauro Carcelli, Vanna Sanna, Michele Palomba, Lieve Naesens, Angela Corona, Nicole Grandi, Enzo Tramontano, Mario Sechi
Publikováno v:
International Journal of Molecular Sciences, Vol 17, Iss 8, p 1371 (2016)
The HIV-1 ribonuclease H (RNase H) function of the reverse transcriptase (RT) enzyme catalyzes the selective hydrolysis of the RNA strand of the RNA:DNA heteroduplex replication intermediate, and represents a suitable target for drug development. A p
Externí odkaz:
https://doaj.org/article/e889b18c555b48ffa711891dd25f10a7
Autor:
Daniela Pagnozzi, Nicolino Pala, Grazia Biosa, Roberto Dallocchio, Alessandro Dessì, Pankaj Kumar SinghPankaj Kumar Singh, Pankaj Kumar Singh, Dominga Rogolino, Anna Di Fiore, Giuseppina De Simone, Claudiu T. Supuran, Mario Sechi
Publikováno v:
ACS medicinal chemistry letters 13 (2022): 271–277. doi:10.1021/acsmedchemlett.1c00644
info:cnr-pdr/source/autori:Daniela Pagnozzi, Nicolino Pala, Grazia Biosa, Roberto Dallocchio, Alessandro Dessì, Pankaj Kumar SinghPankaj Kumar Singh, Pankaj Kumar Singh, Dominga Rogolino, Anna Di Fiore, Giuseppina De Simone, Claudiu T. Supuran, and Mario Sechi/titolo:Interaction Studies between Carbonic Anhydrase and a Sulfonamide Inhibitor by Experimental and Theoretical Approaches/doi:10.1021%2Facsmedchemlett.1c00644/rivista:ACS medicinal chemistry letters/anno:2022/pagina_da:271/pagina_a:277/intervallo_pagine:271–277/volume:13
info:cnr-pdr/source/autori:Daniela Pagnozzi, Nicolino Pala, Grazia Biosa, Roberto Dallocchio, Alessandro Dessì, Pankaj Kumar SinghPankaj Kumar Singh, Pankaj Kumar Singh, Dominga Rogolino, Anna Di Fiore, Giuseppina De Simone, Claudiu T. Supuran, and Mario Sechi/titolo:Interaction Studies between Carbonic Anhydrase and a Sulfonamide Inhibitor by Experimental and Theoretical Approaches/doi:10.1021%2Facsmedchemlett.1c00644/rivista:ACS medicinal chemistry letters/anno:2022/pagina_da:271/pagina_a:277/intervallo_pagine:271–277/volume:13
The most used approaches in structure-based drug design possess peculiar characteristics with advantages and limitations, and thus the management of complementary data from various techniques is of particular interest to synergistically achieve the d
Autor:
Nicolino Pala, Sandro Satta, Mario Sechi, Lisa D Haigh, Francesca Esposito, Mauro Carcelli, Vanna Sanna, Enzo Tramontano, Pankaj Kumar Singh
Publikováno v:
ACS Med Chem Lett
[Image: see text] Photoaffinity labeling (PAL) is one of the upcoming and powerful tools in the field of molecular recognition. It includes the determination of dynamic parameters, such as the identification and localization of the target protein and
Autor:
Mario Sechi, Deeba N. Syed, Nicolino Pala, Alberto Mariani, Antonio Brunetti, Hasan Mukhtar, Salvatore Marceddu, Vanna Sanna
Publikováno v:
Materials Science and Engineering: C. 68:594-602
The bioactive flavonoid fisetin (FS) is a diet-derived antioxidant that is being increasingly investigated for its health-promoting effects. Unfortunately, the poor physicochemical and pharmacokinetic properties affect and limit the clinical applicat
Autor:
Mamuka Kvaratskhelia, Pratibha C. Koneru, Ettore Novellino, Nicolino Pala, Vincenzo Maria D'Amore, Francesca Esposito, Adele Sanna, Sandro Cosconati, Nicole Grandi, Enzo Tramontano, Francesco Saverio Di Leva, Lieve Naesens, Angela Corona, Roberto Di Santo, Mario Sechi
Publikováno v:
Antiviral research. 174
The management of Human Immunodeficiency Virus type 1 (HIV-1) infection requires life-long treatment that is associated with chronic toxicity and possible selection of drug-resistant strains. A new opportunity for drug intervention is offered by anti
Autor:
Daniela Pagnozzi, Nicolino Pala, Grazia Biosa, Roberto Dallocchio, Alessandro Dessì, Pankaj Kumar Singh, Dominga Rogolino, Giuseppina De Simone, Claudiu Supuran, Mario Sechi
Publikováno v:
4st Satellite Meeting on Carbonic Anhydrase, Parma, 14-17/11/2019
info:cnr-pdr/source/autori:Daniela Pagnozzi, Nicolino Pala, Grazia Biosa, Roberto Dallocchio, Alessandro Dessì, Pankaj Kumar Singh, Dominga Rogolino, Giuseppina De Simone, Claudiu Supuran, Mario Sechi/congresso_nome:4st Satellite Meeting on Carbonic Anhydrase/congresso_luogo:Parma/congresso_data:14-17%2F11%2F2019/anno:2019/pagina_da:/pagina_a:/intervallo_pagine
info:cnr-pdr/source/autori:Daniela Pagnozzi, Nicolino Pala, Grazia Biosa, Roberto Dallocchio, Alessandro Dessì, Pankaj Kumar Singh, Dominga Rogolino, Giuseppina De Simone, Claudiu Supuran, Mario Sechi/congresso_nome:4st Satellite Meeting on Carbonic Anhydrase/congresso_luogo:Parma/congresso_data:14-17%2F11%2F2019/anno:2019/pagina_da:/pagina_a:/intervallo_pagine
A prerequisite for the structure-based drug design is an understanding of the principles of molecular recognition in protein-ligand complexes. Photoaffinity labelling (PAL), ie the 'capture' of proteins by small molecules via photoactivation-mediated
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=cnr_________::7a8c120da10c74a2d8a9135f903444e8
http://www.cnr.it/prodotto/i/409895
http://www.cnr.it/prodotto/i/409895
Autor:
Nicolino Pala, Roberta Cadoni, Carrie Lomelino, Brian P. Mahon, Robert McKenna, Roberto Dallocchio, Alessandro Dessì, Mauro Carcelli, Viengsavanh Pimxayvong, Claudia Crosio, Rino Weber, Daniela Vullo, Claudiu Supuran, Mario Sechi
Publikováno v:
4st Satellite Meeting on Carbonic Anhydrase, Parma, 14-17/11/2019
info:cnr-pdr/source/autori:Nicolino Pala, Roberta Cadoni, Carrie Lomelino, Brian P. Mahon, Robert McKenna, Roberto Dallocchio, Alessandro Dessì, Mauro Carcelli, Viengsavanh Pimxayvong, Claudia Crosio, Rino Weber, Daniela Vullo, Claudiu Supuran, Mario Sechi/congresso_nome:4st Satellite Meeting on Carbonic Anhydrase/congresso_luogo:Parma/congresso_data:14-17%2F11%2F2019/anno:2019/pagina_da:/pagina_a:/intervallo_pagine
info:cnr-pdr/source/autori:Nicolino Pala, Roberta Cadoni, Carrie Lomelino, Brian P. Mahon, Robert McKenna, Roberto Dallocchio, Alessandro Dessì, Mauro Carcelli, Viengsavanh Pimxayvong, Claudia Crosio, Rino Weber, Daniela Vullo, Claudiu Supuran, Mario Sechi/congresso_nome:4st Satellite Meeting on Carbonic Anhydrase/congresso_luogo:Parma/congresso_data:14-17%2F11%2F2019/anno:2019/pagina_da:/pagina_a:/intervallo_pagine
Carbonic anhydrases (CAs) are emerging as potential biological targets for cancer therapy. In particular, hCA IX isoform has been found to be expressed in a wide variety of malignancies and appear to be tightly regulated by micro-environmental hypoxi
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=cnr_________::43c3340500f9bd67a50f6ba6662982ed
http://www.cnr.it/prodotto/i/409899
http://www.cnr.it/prodotto/i/409899