Zobrazeno 1 - 5
of 5
pro vyhledávání: '"Nicola Paesano"'
Autor:
Nicola Paesano, Jean-Charles Lancelot, Mariafrancesca Buonerba, Giovanni De Martino, Carmela Saturnino
Publikováno v:
Il Farmaco. 58:819-822
The anti-amoebic power of a series of bis-thioureidic derivatives against amoeba, responsible for a serious form of keratitis of the cornea, has been analysed. The synthesis of these products is also described.
Autor:
Nicola Paesano, Marino Artico, Dante Rotili, Corrado Spadafora, Antonello Mai, Sara Bartolini, Gianluca Sbardella
Publikováno v:
Journal of Medicinal Chemistry. 48:6776-6778
Two 2,6-difluoro-DABO derivatives (MC 1047, 1, and MC 1220, 2, respectively) were tested against endogenous, nontelomeric reverse transcriptase (endo-RT) in human differentiating cell systems to investigate their antiproliferative and cytodifferentia
Autor:
Corrado Spadafora, Antonello Mai, Sabrina Castellano, Sara Bartolini, Nicola Paesano, Marino Artico, Gianluca Sbardella, Dante Rotili
Novel triazine analogues of 5-alkyl-2-alkylthio-6-[1-(2,6-difluorophenyl)alkyl]-3,4-dihydropyrimidin-4(3H)-ones (F(2)-DABOs), previously described by us as nonnucleoside HIV-1 reverse transcriptase inhibitors (NNRTIs), were tested for their antiproli
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::47f2898858b988f4890b01562bd5572e
http://hdl.handle.net/11386/1529752
http://hdl.handle.net/11386/1529752
Autor:
Giovanni De Martino, Carmela Saturnino, Giuseppina Autore, Caterina Vicidomini, Nicola Paesano, Gianluca Sbardella, Stefania Marzocco
Novel benzyl- and phenyl-isothioureidic derivatives have been synthesised and evaluated as inhibitors of nitric oxide synthesis, induced in lipopolysaccharide (LPS)-activated J774.A1 macrophage cell line. The most potent iNOS inhibitor resulting was
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1cde10c532134733fc493d3ee6e6b85d
http://hdl.handle.net/11386/1000470
http://hdl.handle.net/11386/1000470
Autor:
Giovanni De Martino, Marta D'Auria, Carmela Saturnino, Daniele Saponiero, Nicola Paesano, Giuseppina Cioffi, Mariafrancesca Buonerba
Publikováno v:
Farmaco (Societa chimica italiana : 1989). 58(9)
Recent developments in biomedical science have shown that free radicals are involved in many diseases. They attack the unsaturated fatty acids in the biomembrane resulting in membrane lipid peroxidation, which is strongly connected to aging, carcinog