Synthesis and SAR of benzyl and phenoxymethylene oxadiazole benzenesulfonamides as selective b3 adrenergic receptor agonist antiobesity agents

Autor: Biftu, T., Feng, D. D., Liang, G. B., Kuo, H., Qian, X., Naylor, E. M., Colandrea, V. J., Candelore, M. R., Cascieri, M. A., Jr., L. F. Colwell

Publikováno v: Bioorganic & Medicinal Chemistry Letters; 2000, Vol. 10 Issue: 13 p1431-1434, 4p

Human ~3 adrenergic receptor agonists containing cyclic ureidobenzene-sulfonamides

Autor: Parmee, E. R., Naylor, E. M., Perkins, L., Colandrea, V. J., Ok, H. O., Candelore, M. R., Cascleri, M. A., Deng, L., Feeney, W. P., Forrest, M. J.

Publikováno v: Bioorganic & Medicinal Chemistry Letters; 1999, Vol. 9 Issue: 5 p749-754, 6p

Pharmacology of L-744,453, a Novel Nonpeptidyl Endothelin Antagonist

Autor: Williams, D. L., Murphy, K. L., Nolan, N. A., O'Brien, J. A., Lis, E. V., Pettibone, D. J., Clineschmidt, B. V., Krause, S. M., Veber, D. F., Naylor, E. M.

Publikováno v: Life Sciences; 1996, Vol. 58 Issue: 14 p1149-1157, 9p

Development of [^1^1C]L-159,884: a radiolabelled, nonpeptide angiotensin II antagonist that is useful for angiotensin II, AT~1 receptor imaging

Autor: Hamill, T. G., Burns, H. D., Dannals, R. F., Mathews, W. B., Musachio, J. L., Ravert, H. T., Naylor, E. M.

Publikováno v: Applied Radiation and Isotopes: Including Data, Instrumentation, and Methods for Use in Agriculture, Industry, and Medicine; 1996, Vol. 47 Issue: 2 p211-218, 8p

Triazolinones as nonpeptide angiotensin II antagonists-II. Discovery of a potent and orally active triazolinone acylsulfonamide

Autor: Chang, L. L., Ashton, W. T., Flanagan, K. L., Naylor, E. M.

Publikováno v: Bioorganic & Medicinal Chemistry Letters; 1994, Vol. 4 Issue: 1 p115-115, 1p