Zobrazeno 1 - 4
of 4
pro vyhledávání: '"Natalia S. Dashkova"'
Autor:
Nikolai Y. Zyk, Anastasiia S. Garanina, Ekaterina A. Plotnikova, Anton P. Ber, Ekaterina A. Nimenko, Natalia S. Dashkova, Anastasiia A. Uspenskaia, Radik R. Shafikov, Dmitry A. Skvortsov, Stanislav A. Petrov, Andrey A. Pankratov, Nikolai V. Zyk, Alexander G. Majouga, Elena K. Beloglazkina, Aleksei E. Machulkin
Publikováno v:
International Journal of Molecular Sciences, Vol 24, Iss 14, p 11327 (2023)
Prostate cancer is the second most common cancer among men. We designed and synthesized new ligands targeting prostate-specific membrane antigen and suitable for bimodal conjugates with diagnostic and therapeutic agents. In vitro studies of the affin
Externí odkaz:
https://doaj.org/article/a8378698c0ce4a6eae024f4e4f123eb9
Autor:
Anastasiia A. Uspenskaya, Ekaterina A. Nimenko, Radik R. Shafikov, Nikolay Y. Zyk, Sergei A. Evteev, Natalia S. Dashkova, Yan A. Ivanenkov, Alexander G. Majouga, Dmitry A. Skvortsov, Anastasiia S. Garanina, Elena K. Beloglazkina, Aleksei E. Machulkin
Publikováno v:
Medicinal Chemistry Research. 32:32-37
Autor:
Nikolai Y. Zyk, Anton P. Ber, Ekaterina A. Nimenko, Radik R. Shafikov, Sergei A. Evteev, Stanislav A. Petrov, Anastasia A. Uspenskaya, Natalia S. Dashkova, Yan A. Ivanenkov, Dmitry A. Skvortsov, Elena K. Beloglazkina, Alexander G. Majouga, Aleksei E. Machulkin
Publikováno v:
Bioorganicmedicinal chemistry letters. 71
We report an improved series of ligands targeting prostate specific membrane antigen (PSMA). The new compounds were designed by the introduction of changes in the structure of the aromatic fragment at ε-nitrogen atom of lysine that resulted in impro
Autor:
Pavel A. Ignatov, Pavel A. Panchenko, Svetlana V Lavrushkina, Igor I. Kireev, Vladislav M Malinnikov, Elena K. Beloglazkina, Irina V. Grishina, Sergey S Kovalev, Nikolay V. Zyk, Olga O. Krasnovskaya, Dmitry A. Skvortsov, Vasily M. Gerasimov, Marina A. Zakharko, Olga A. Fedorova, Alexander G. Majouga, Natalia S Dashkova, Gediminas Jonusauskas
Publikováno v:
Bioconjugate Chemistry
Bioconjugate Chemistry, American Chemical Society, 2019, 30 (3), pp.741-750. ⟨10.1021/acs.bioconjchem.8b00885⟩
Bioconjugate Chemistry, American Chemical Society, 2019, 30 (3), pp.741-750. ⟨10.1021/acs.bioconjchem.8b00885⟩
International audience; A novel approach to the synthesis of pH-sensitive prodrugs has been proposed: thiourea drug modification. Resulting prodrugs can release the cytotoxic agent and the biologically active 2-thiohydantoin in the acidic environment
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::397611eaa0536cac056ce61dd5ab2de2
https://hal.archives-ouvertes.fr/hal-02404558/file/GJ_acs_bioconjchem_2019.pdf
https://hal.archives-ouvertes.fr/hal-02404558/file/GJ_acs_bioconjchem_2019.pdf