Zobrazeno 1 - 10
of 21
pro vyhledávání: '"Natalia Monakhova"'
Autor:
Brindha Gap-Gaupool, Sarah M. Glenn, Emily Milburn, Obolbek Turapov, Marialuisa Crosatti, Jennifer Hincks, Bradley Stewart, Joanna Bacon, Sharon L. Kendall, Martin I. Voskuil, Olga Riabova, Natalia Monakhova, Jeffrey Green, Simon J. Waddell, Vadim A. Makarov, Galina V. Mukamolova
Publikováno v:
Communications Biology, Vol 7, Iss 1, Pp 1-12 (2024)
Abstract During infection Mycobacterium tuberculosis (Mtb) forms physiologically distinct subpopulations that are recalcitrant to treatment and undetectable using standard diagnostics. These difficult to culture or differentially culturable (DC) Mtb
Externí odkaz:
https://doaj.org/article/036ab31366e34a5191d2bed82482e8a4
Autor:
Andrea Bonacorsi, Gabriele Trespidi, Viola C. Scoffone, Samuele Irudal, Giulia Barbieri, Olga Riabova, Natalia Monakhova, Vadim Makarov, Silvia Buroni
Publikováno v:
Frontiers in Microbiology, Vol 15 (2024)
Pseudomonas aeruginosa is a major human pathogen, able to establish difficult-to-treat infections in immunocompromised and people with cystic fibrosis (CF). The high rate of antibiotic treatment failure is due to its notorious drug resistance, often
Externí odkaz:
https://doaj.org/article/eecec8b29cb24247927d9450f0859610
Autor:
Thane Jones, Natalia Monakhova, Florence Guivel-Benhassine, Alexander Lepioshkin, Timothée Bruel, Thomas R. Lane, Olivier Schwartz, Ana C. Puhl, Vadim Makarov, Sean Ekins
Publikováno v:
ACS Omega, Vol 8, Iss 43, Pp 40817-40822 (2023)
Externí odkaz:
https://doaj.org/article/837556e13c3e4a1aa59e31dcd50f48c2
Autor:
Elena G. Salina, Umberto Postiglione, Laurent R. Chiarelli, Deborah Recchia, Monika Záhorszká, Alexander Lepioshkin, Natalia Monakhova, Adrian Pál, Alessio Porta, Giuseppe Zanoni, Jana Korduláková, Elena Kazakova, Davide Sassera, Maria Rosalia Pasca, Vadim Makarov, Giulia Degiacomi
Publikováno v:
mSphere, Vol 7, Iss 6 (2022)
ABSTRACT Tuberculosis (TB) still poses a global menace as one of the deadliest infectious diseases. A quarter of the human population is indeed latently infected with Mycobacterium tuberculosis. People with latent infection have a 5 to 10% lifetime r
Externí odkaz:
https://doaj.org/article/df59359de4744e088c1593f4deded2ce
Autor:
Laurent R. Chiarelli, Viola Camilla Scoffone, Gabriele Trespidi, Giulia Barbieri, Olga Riabova, Natalia Monakhova, Alessio Porta, Giulia Manina, Giovanna Riccardi, Vadim Makarov, Silvia Buroni
Publikováno v:
Frontiers in Microbiology, Vol 11 (2020)
There is an urgent need for new antimicrobials to treat the opportunistic Gram-negative Burkholderia cenocepacia, which represents a problematic challenge for cystic fibrosis patients. Recently, a benzothiadiazole derivative, C109, was shown to be ef
Externí odkaz:
https://doaj.org/article/771a8688f6c042509aba8391a0500a4d
Autor:
Andréanne Lupien, Caroline Shi-Yan Foo, Svetlana Savina, Anthony Vocat, Jérémie Piton, Natalia Monakhova, Andrej Benjak, Dirk A Lamprecht, Adrie J C Steyn, Kevin Pethe, Vadim A Makarov, Stewart T Cole
Publikováno v:
PLoS Pathogens, Vol 16, Iss 1, p e1008270 (2020)
The emergence of multi-drug (MDR-TB) and extensively-drug resistant tuberculosis (XDR-TB) is a major threat to the global management of tuberculosis (TB) worldwide. New chemical entities are of need to treat drug-resistant TB. In this study, the mode
Externí odkaz:
https://doaj.org/article/b7f8b7461a4442bc8a002d6f37ec16b1
Autor:
Thomas Lane, Vadim Makarov, Julie A. E. Nelson, Rick B. Meeker, Giuseppina Sanna, Olga Riabova, Elena Kazakova, Natalia Monakhova, Andrey Tsedilin, Fabio Urbina, Thane Jones, Ashley Suchy, Sean Ekins
Publikováno v:
Journal of Medicinal Chemistry. 66:6193-6217
Autor:
Ana C. Puhl, Giovanni F. Gomes, Samara Damasceno, Andre S. Godoy, Gabriela D. Noske, Aline M. Nakamura, Victor O. Gawriljuk, Rafaela S. Fernandes, Natalia Monakhova, Olga Riabova, Thomas R. Lane, Vadim Makarov, Flavio P. Veras, Sabrina S. Batah, Alexandre T. Fabro, Glaucius Oliva, Fernando Q. Cunha, José C. Alves-Filho, Thiago M. Cunha, Sean Ekins
Publikováno v:
Repositório Institucional da USP (Biblioteca Digital da Produção Intelectual)
Universidade de São Paulo (USP)
instacron:USP
Universidade de São Paulo (USP)
instacron:USP
There are currently relatively few small-molecule antiviral drugs that are either approved or emergency-approved for use against severe acute respiratory coronavirus 2 (SARS-CoV-2). One of these is remdesivir, which was originally repurposed from its
Autor:
Eva Repková, Jaroslav Roh, Júlia Zemanová, Jana Korduláková, Natalia Monakhova, Jozef Nosek, Maria Rosalia Pasca, Anna Egorova, Josè Camilla Sammartino, Giulia Degiacomi, Vadim Makarov, Elena G. Salina, Renáta Górová, Anthony Vocat, Alexander Lepioshkin, Katarína Mikušová, Helena Jurdáková, Stewart T. Cole
Publikováno v:
ACS Infectious Diseases. 7:88-100
Latent Mycobacterium tuberculosis infection presents one of the largest challenges for tuberculosis control and novel antimycobacterial drug development. A series of pyrano[3,2-b]indolone-based compounds was designed and synthesized via an original e
Autor:
Laura Rank, Ana C. Puhl, Tammy M. Havener, Edward Anderson, Daniel H. Foil, Kimberley M. Zorn, Natalia Monakhova, Olga Riabova, Anthony J. Hickey, Vadim Makarov, Sean Ekins
Publikováno v:
Bioorganic & Medicinal Chemistry. 73:117043
Neuroblastoma (NB) is the second leading extracranial solid tumor of early childhood with about two-thirds of cases presenting before the age of 5, and accounts for roughly 15 percent of all pediatric cancer fatalities in the United States. Treatment