Zobrazeno 1 - 10
of 11
pro vyhledávání: '"Naginbhai M. Patel"'
Autor:
Nancy Butkiewicz, Andrea Hart, Frank Bennett, Viyyoor M. Girijavallabhan, Bimal Dasmahapatra, Naginbhai M. Patel
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 8:931-934
Studies involving modifications to the P3 position of previously described HIV-protease inhibitors 1 containing β-hydroxyether and thioether dipeptide isostere replacements led to the discovery of pseudopeptides 8o and 8p with improved antiviral act
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::44c22a791cf4967cb2726082b799ee7a
https://doi.org/10.1016/s0960-894x(98)00144-9
https://doi.org/10.1016/s0960-894x(98)00144-9
Publikováno v:
ChemInform. 24
The title oxiranes were constructed in > 95% enantiomeric excess (e.e.) utilizing a Sharpless asymmetric epoxidation followed by regioselective azide displacement with [Ti(OPri)2(N3)2] as the key steps.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::32f07937b297668fc81fc437b6156e7f
https://doi.org/10.1002/chin.199334151
https://doi.org/10.1002/chin.199334151
Publikováno v:
ChemInform. 25
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::a9d66b5b38636e38fdb65ed7863226e0
https://doi.org/10.1002/chin.199406113
https://doi.org/10.1002/chin.199406113
Autor:
P. J. O'Hanlon, D. F. Rane, Liu Yi-Tsung, Naginbhai M. Patel, A. K. Ganguly, Patrick Pinto, Alan B. Cooper, Raymond G. Lovey, V. Girijavallabhan, P. H. Bentley, Frank Bennett, Jagdish A. Desai, Edwin Jao, Anil K. Saksena, Russell E. Pike, Haiyan Wang
Publikováno v:
ChemInform. 28
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::cb79029f38213dca7476f7bd5db21864
https://doi.org/10.1002/chin.199729284
https://doi.org/10.1002/chin.199729284
Autor:
Andrea Hart, Bimal Dasmahapatra, Frank Bennett, Viyyoor M. Girijavallabhan, Nancy Butkiewicz, Naginbhai M. Patel
Publikováno v:
ChemInform. 29
Studies involving modifications to the P3 position of previously described HIV-protease inhibitors 1 containing β-hydroxyether and thioether dipeptide isostere replacements led to the discovery of pseudopeptides 8o and 8p with improved antiviral act
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::b21e3b406d432237972b70e405907d1d
https://doi.org/10.1002/chin.199832257
https://doi.org/10.1002/chin.199832257
Autor:
Naginbhai M. Patel, Eugene L. Moss, Roberta S. Hare, Frank Bennett, Patrick Pinto, Pike Russell E, Viyyoor M. Girijavallabhan, Anil K. Saksena, Yi-Tsung Liu, Raymond G. Lovey, Edwin Jao, David Loebenberg, Anthony Cacciapuoti, Amin A. Nomeir, Fred Menzel, Ashit K. Ganguly, Haiyan Wang
Publikováno v:
Bioorganicmedicinal chemistry letters. 16(1)
As part of a detailed study, the syntheses, biological activities, and pharmacokinetic properties of hydroxylated analogues of the previously described broad spectrum antifungal agents, Sch 51048 (1), Sch 50001 (3), and Sch 50002 (4), are described.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::f7c2c26e041c8d1f55cc640e41f9603e
https://pubmed.ncbi.nlm.nih.gov/16260134
https://pubmed.ncbi.nlm.nih.gov/16260134
Autor:
Frank Bennett, Ashit K. Ganguly, Nancy Butkiewicz, Naginbhai M. Patel, Viyyoor M. Girijavallabhan, Andrea Hart, Bimalendu Dasmahapatra
Publikováno v:
Bioorganicmedicinal chemistry. 2(10)
The syntheses, enzyme inhibition and antiviral activity of potent HIV-protease inhibitors containing novel β-hydroxy ether and thioethers based on the transition state mimetic concept are discussed.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::bcbde7121c63d738c7f2698a9191c09c
https://pubmed.ncbi.nlm.nih.gov/7773624
https://pubmed.ncbi.nlm.nih.gov/7773624
Publikováno v:
J. Chem. Soc., Chem. Commun.. :737-738
The title oxiranes were constructed in > 95% enantiomeric excess (e.e.) utilizing a Sharpless asymmetric epoxidation followed by regioselective azide displacement with [Ti(OPri)2(N3)2] as the key steps.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::bef2df7be105c2b9ec7ffd38efa0334e
https://doi.org/10.1039/c39930000737
https://doi.org/10.1039/c39930000737
Publikováno v:
Synlett. 1993:703-704
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::891b1270a9946a4c131712ff55a41409
https://doi.org/10.1055/s-1993-22579
https://doi.org/10.1055/s-1993-22579
Autor:
Viyyoor M. Girijavallabhan, Pinto Patrick A, George H. Miller, Roberta H. Hare, Naginbhai M. Patel, Yi-Tsung Liu, Ashit K. Ganguly
Publikováno v:
The Journal of antibiotics. 39(8)
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::40a3b81be90d1a81c8e1579255f4cda2
https://pubmed.ncbi.nlm.nih.gov/3759670
https://pubmed.ncbi.nlm.nih.gov/3759670