Zobrazeno 1 - 10 of 19 pro vyhledávání: '"N. S. Kula"'
1
Synthesis, Receptor Potency, and Selectivity of Halogenated Diphenylpiperidines as Serotonin 5-HT2A Ligands for PET or SPECT Brain Imaging
Autor: Ronald M. Baldwin, N. S. Kula, Gilles Tamagnan, Robert B. Innis, Ping-Zhong Tan, Ross J. Baldessarini, Xing Fu
Publikováno v: Journal of Medicinal Chemistry. 45:2319-2324
A series of 4'-substituted phenyl-4-piperidinylmethanol and benzoyl-4-piperidine derivatives was synthesized as potential novel serotonin 5-HT2A receptor ligands that can be radiolabeled for in vivo brain imaging. Compounds were prepared by alkylatio
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d4e514a1d25725df931155a5a036d2cb
https://doi.org/10.1021/jm0200411
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6
(R)- and (S)-enantiomers of 11-hydroxy- and 10,11-dihydroxy-N-allylnoraporphine: synthesis and affinity for dopamine receptors in rat brain tissue
Autor: Yigong Gao, John L. Neumeyer, Ross J. Baldessarini, N. S. Kula
Publikováno v: Journal of Medicinal Chemistry. 34:24-28
The R-(-)- and S-(+)-enantiomers of 11-hydroxy-N-allyl (4), and 10,11-dihydroxy-N-allyl (3) congeners of 11-hydroxy-N-n-propylnorapomorphine (11-OH-NPa, 2) or N-n-propylnorapomorphine (NPA, 1) were synthesized. Binding affinity of these compounds at
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::5e8c867efe378e1df0655ec42e6516b0
https://doi.org/10.1021/jm00105a005
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7
Synthesis and Monoamine Transporter Affinity of New 2β-Carbomethoxy-3β-[4-(substituted thiophenyl)]phenyltropanes: Discovery of a Selective SERT Antagonist with Picomolar Potency
Autor: Gilles Tamagnan, David Alagille, Xing Fu, Robert B. Innis, N. S. Kula, Ross J. Baldessarini, Ronald M. Baldwin
Publikováno v: ChemInform. 36
Preparation of cocaine analogues has been aimed largely at development of stable compounds with high affinity and selectivity for the dopamine transporter (DAT). We now report the synthesis and monoamine transporter affinity of 10 new 2β-carbomethox
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::123faad983e5f5587f81f1090dad6b3f
https://doi.org/10.1002/chin.200527194
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9
Synthesis of cyclopentadienyltricarbonyl rhenium phenyltropanes by double ligand transfer: organometallic ligands for the dopamine transporter
Autor: N. S. Kula, Ronald M. Baldwin, Gilles Tamagnan, Ross J. Baldessarini, Sami S. Zoghbi, Richard R. Cesati, John A. Katzenellenbogen, Robert B. Innis
Publikováno v: Bioconjugate chemistry. 13(1)
Cyclopentadienyltricarbonyl rhenium (CpRe(CO)(3)) systems can be prepared from ferrocenes and perrhenate by a double ligand transfer (DLT) reaction that gives reasonable yields and shows excellent functional group tolerance. We used this reaction for
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1350893525d09bba319a81e5408e6a34
https://pubmed.ncbi.nlm.nih.gov/11792176
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