Zobrazeno 1 - 10
of 62
pro vyhledávání: '"N Dereu"'
Publikováno v:
Bulletin des Sociétés Chimiques Belges. 89:773-778
Synthesis of five new fundamental biheterocyclic systems was realized through condensation of the isothiazole or isoselenazole ring on the thiophene or selenophene ring. These new heterocycles were characterized by elemental analysis, U. V., N. M. R.
Autor:
A. Bousseau, Y. Lelievre, Y. Ribeill, N Dereu, J.-C. Gueguen, Y. Henin, J.-B. Le Pecq, M. Evers, F. Soler, E. De Clercq, D. Reisdorf, I. Morize, J F Mayaux, Rudi Pauwels, C Poujade, C. James
Publikováno v:
Journal of Medicinal Chemistry. 39:1056-1068
A series of omega-undecanoic amides of lup-20(29)-en-28-oic acid derivatives were synthesized and evaluated for activity in CEM 4 and MT-4 cell cultures against human immunodeficiency virus type 1 (HIV-1) strain IIIB/LAI. The potent HIV inhibitors wh
Autor:
E. De Clercq, C Poujade, N Dereu, Y. Henin, T Huet, Francoise Soler, Michel Dr Evers, Jean-François Mayaux, Anne Bousseau, Rudi Wilfried Jan Pauwels
Publikováno v:
Proceedings of the National Academy of Sciences. 91:3564-3568
A series of triterpene compounds characterized by a stringent structure-activity relationship were identified as potent and selective inhibitors of human immunodeficiency virus type 1 (HIV-1) replication. Currently studied botulinic derivatives have
Autor:
A. Bousseau, Y. Lelievre, Y. Henin, M. Evers, J.-B. Le Pecq, C Poujade, C. James, E. De Clercq, J F Mayaux, Rudi Pauwels, I. Morize, D. Reisdorf, Y. Ribeill, F. Soler, N Dereu, J.-C. Gueguen
Publikováno v:
ChemInform. 27
A series of omega-undecanoic amides of lup-20(29)-en-28-oic acid derivatives were synthesized and evaluated for activity in CEM 4 and MT-4 cell cultures against human immunodeficiency virus type 1 (HIV-1) strain IIIB/LAI. The potent HIV inhibitors wh
Autor:
C Poujade, J F Mayaux, T Huet, A. Bousseau, Rudi Pauwels, J.‐C. Carry, N Dereu, F. Soler, Y. Henin, J.-B. Le Pecq, M. Evers, E. De Clercq
Publikováno v:
ChemInform. 27
A novel series of omega-aminoalkanoic acid derivatives of betulinic acid were synthesized and evaluated for their activity against human immunodeficiency virus (HIV). The anti-HIV-1 activity of several members of this new series was found to be in th
Publikováno v:
Electrochimica Acta. 36:631-637
Autor:
Rudi Pauwels, A. Bousseau, Y. Henin, J.-B. Le Pecq, M. Evers, C Poujade, E. De Clercq, F. Soler, T Huet, J F Mayaux, J.‐C. Carry, N Dereu
Publikováno v:
Journal of medicinal chemistry. 39(5)
A novel series of omega-aminoalkanoic acid derivatives of betulinic acid were synthesized and evaluated for their activity against human immunodeficiency virus (HIV). The anti-HIV-1 activity of several members of this new series was found to be in th
Publikováno v:
Photochemistry and photobiology. 54(5)
The bimolecular rate constants (k) of quenching of molecular singlet oxygen 1O2 (1 delta g) by organo-selenium compounds exhibiting glutathione peroxidase activity and by sulfur analogs have been determined by time resolved phosphorescence detection
[Benzisoselenazolinones and their derivatives, a new series of anti-inflammatories and antioxidants]
Publikováno v:
Journal de pharmacie de Belgique. 45(5)
Ebselen, a benzisoselenazolinone, displays antiinflammatory properties and antioxidant capacity similar to the enzyme glutathione peroxydase. Structural modifications were realized. The presence of substituents ortho to selenium, and in particular of
Publikováno v:
Journal of Molecular Structure. 67:251-267
Analysis of the dipole moments of chalcogenoanisoles, the directions of which are given by those of their p -bromo derivatives, shows that the mesomeric moment decreases on passing from anisole to thioanisole, selenoanisole and telluroanisole ( m = 1