Scalable synthesis and antibacterial evaluation of 2‐(3‐( N ‐(substituted phenyl)sulfamoyl)ureido)benzothiazoles

Autor: Abbas Boukhari, Zinelaabidine Cheraiet, Zine Regainia, Mounir Nessaib, Sihem Hessainia, Abdelghani Djahoudi, Saida Meliani

Publikováno v: Archiv der Pharmazie. 352:1800341

A new series of 2-(3-(N-(substituted phenyl)sulfamoyl)ureido)benzothiazoles was synthesized via a one-pot efficient and scalable method, involving the condensation of 2-aminobenzothiazoles derivatives, substituted anilines, and chlorosulfonyl isocyan

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::375b9ee9eacd6c95e6d3bc3388c1dd3f
https://doi.org/10.1002/ardp.201800341

Synthesis of substituted N-aryl-N'-sulfamoyl-oxazolidin-2-ones with potential antibacterial activity

Autor: Jean-Yves Winum, Mekki Kadri, Mounir Nessaib, Abed el Ghani Djahoudi, Mohamed Abdaoui

Publikováno v: Recent Patents Anti-Infectives Drug Discovery
Recent Patents Anti-Infectives Drug Discovery, 2007, 2, pp.131-139. ⟨10.2174/157489107780832604⟩

Three series of derived compounds of N, Aryl-N',Sulfamoyloxazolidin-2-ones were synthesized starting from chloro-sulfonylisocyanate (CSI) by carbomoylation, sulfamoylation and intramolecular cyclization reactions followed by methylation and heterocyc

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::9f77086227f4cc0b339b6c230df33d5b
https://hal.archives-ouvertes.fr/hal-00355557