Zobrazeno 1 - 3
of 3
pro vyhledávání: '"Morten Lysen"'
Publikováno v:
Tetrahedron. 73:1576-1582
Morpholine amides are cheap and safe alternative to Weinreb amides as acylating agents of organometallic species. Herein, the in-situ lithiation/borylation of 18 ortho- meta- and para-substituted morpholine benzamides has been investigated. 10 of the
Autor:
Morten Lysen, Klaus Koehler
Publikováno v:
Synlett. :1671-1674
Aqueous reaction conditions that activate various aryl chlorides in Suzuki-Miyaura cross-coupling have been developed. These environment friendly conditions utilize ligandless Pd/C (Pd concentrations 0.2-2 mol%) that allow easy separation of the cata
Publikováno v:
The Journal of organic chemistry. 71(6)
The synthesis of substituted 2-cyanoarylboronic esters is described via lithiation/in situ trapping of the corresponding methoxy-, trifluoromethyl-, fluoro-, chloro-, and bromobenzonitriles. The crude arylboronic esters were obtained in high yields a