Zobrazeno 1 - 10
of 23
pro vyhledávání: '"Monica Palme"'
Autor:
Monica Palmerini
Publikováno v:
Círculo de Lingüística Aplicada a la Comunicación, Vol 32 (2023)
Externí odkaz:
https://doaj.org/article/9934497d51584a3a8bfd118fea59c79a
Autor:
Charles-André Lemelin, Boris M. Seletsky, Kimberley K. Aalfs, Paul J. Lydon, Davis Heather, Yoshito Kishi, Kathleen A. Salvato, Bruce A. Littlefield, Lynda Tremblay, Murray J. Towle, Charles E. Chase, Yongchun Shen, Lori A. Singer, Melvin J. Yu, Wanjun Zheng, Bruce F. Wels, Monica Palme
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 14:5551-5554
Structurally simplified macrocyclic ketone analogues of halichondrin B were prepared by total synthesis and found to retain the potent cell growth inhibitory activity in vitro, stability in mouse serum, and in vivo efficacy of the natural product.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::4462039df1979f9c23e2ed5bf322971f
https://doi.org/10.1016/j.bmcl.2004.08.069
https://doi.org/10.1016/j.bmcl.2004.08.069
Autor:
Yoshida Kenichi, William J. Watkins, Monica Palme, Aesop Cho, Katsuya Akimoto, Kazuki Hoshino, Ving J. Lee, Atsunobu Sakamoto, Jason Z. Zhang, Haruko Kawato, Kiyoshi Nakayama, Hiroko Ishida, Masami Ohtsuka, Yoshihiro Yokomizo, Noriko Kuru, Toshiharu Ohta, Junko Itoh
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 14:2493-2497
Exchange of the ethylene tether in a series of pyridopyrimidine-based MexAB-OprM specific efflux pump inhibitors to an amide bond stabilized the olefin of the acrylic acid moiety, preventing facile photoisomerization to the Z-isomer. Furthermore, the
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7d9735d100912fc40fc6ce377c87008a
https://doi.org/10.1016/j.bmcl.2004.03.007
https://doi.org/10.1016/j.bmcl.2004.03.007
Autor:
Aesop Cho, Yoshida Kenichi, Monica Palme, William J. Watkins, Atsunobu Sakamoto, Toshiharu Ohta, Noriko Kuru, Ving J. Lee, Masami Ohtsuka, Jun Watanabe, Haruko Kawato, Jason Z. Zhang, Hiroko Ishida, Kiyoshi Nakayama, Kazuki Hoshino, Yoshihiro Yokomizo, Kumi Yoshida
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 14:475-479
The addition of substituents to the pyridopyrimidine scaffold of MexAB-OprM specific efflux pump inhibitors was explored. As predicted by a pharmacophore model, the incorporation substituents at the 2-position improved potency. Piperidines were found
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::bc608919c67dc6a90ece8c90d78138ea
https://doi.org/10.1016/j.bmcl.2003.10.060
https://doi.org/10.1016/j.bmcl.2003.10.060
Autor:
Andrea Vasella, Monica Palme
Publikováno v:
Helvetica Chimica Acta. 78:959-969
A number of new glycosyl donors, O-(1-phenyl-1H-tetrazol-5-yl) glycosides, are prepared from the corresponding hemiacetals, commercially available 5-chloro-1-phenyl-1H-tetrazole (2), and tetrabutylammonium fluoride (Bu4NF) in either THF or DMF. The m
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::54dae5daf3c767e45f560422e60fb515
https://doi.org/10.1002/hlca.19950780418
https://doi.org/10.1002/hlca.19950780418
Autor:
Monica Palme, Andrea Vasella
Publikováno v:
Bioorganic & Medicinal Chemistry. 2:1169-1177
A new glycosyl donor possessing an anomeric O -(1-phenyltetrazol-5-yl) group is prepared from 2,3,4,6-tetra- O -benzyl- d -glucose ( 2 ) and commercially available 5-chloro-1-phenyl-1 H -tetrazole ( 1 ). The synthesis of glycosides derived from the d
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::f7e1ed6c7f8df24a28e9a7f4e7c3520d
https://doi.org/10.1016/s0968-0896(00)82068-4
https://doi.org/10.1016/s0968-0896(00)82068-4
Autor:
Satish Rao, Monica Palme, Adrian Davies, Padmapriya Kumaraswamy, Pascal Druzgala, S. Scott Bowersox, Luke K. Lightning, Renee Coleman, Dave J. Ellis
Publikováno v:
Drug metabolism and disposition: the biological fate of chemicals. 39(7)
The absorption and disposition of the serotonin 5-HT(4) receptor agonist, naronapride (6-[(3S,4R)-4-(4-amino-5-chloro-2-methoxy-benzoylamino)-3-methoxy-piperidin-1-yl]-hexanoic acid 1-aza-bicyclo[2,2,2]oct-(R)-3-yl ester dihydrochloride; ATI-7505), w
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::5be71c72e5eb97d58622f8892f637f56
https://pubmed.ncbi.nlm.nih.gov/21447732
https://pubmed.ncbi.nlm.nih.gov/21447732
Autor:
Andrea Vasella, Monica Palme
Publikováno v:
ChemInform. 26
A number of new glycosyl donors, O-(1-phenyl-1H-tetrazol-5-yl) glycosides, are prepared from the corresponding hemiacetals, commercially available 5-chloro-1-phenyl-1H-tetrazole (2), and tetrabutylammonium fluoride (Bu4NF) in either THF or DMF. The m
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::0bbb10754b01ab6372cd6632a40afeff
https://doi.org/10.1002/chin.199538256
https://doi.org/10.1002/chin.199538256
Publikováno v:
The FASEB Journal. 24
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::4a091721b79a03d80209066815389b2a
https://doi.org/10.1096/fasebj.24.1_supplement.967.10
https://doi.org/10.1096/fasebj.24.1_supplement.967.10
Autor:
Monica Palme, Renee Coleman, Padmapriya Kumaraswamy, Pascal Druzgala, Ian Irwin, Luke K. Lightning
Publikováno v:
The FASEB Journal. 24
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::8dc53c2021fc15a4cdcc12e099f9055c
https://doi.org/10.1096/fasebj.24.1_supplement.967.1
https://doi.org/10.1096/fasebj.24.1_supplement.967.1