Zobrazeno 1 - 10
of 36
pro vyhledávání: '"Mohammed Khaled bin Break"'
Autor:
Mazdida Sulaiman, Layane Ebehairy, Veeranoot Nissapatorn, Mohammed Rahmatullah, Jhonnel Villegas, Helina Jean Dupa, Ricksterlie C. Verzosa, Karma G. Dolma, Muhamad Shabaz, Scholastica Lanting, Nor Azizun Rusdi, Nor Hayati Abdullah, Mohammed Khaled Bin Break, Teng Jin Khoo, Wei Wang, Christophe Wiart
Publikováno v:
Pharmaceutical Biology, Vol 62, Iss 1, Pp 713-766 (2024)
Context The emergence of pan-resistant bacteria requires the development of new antibiotics and antibiotic potentiators.Objective This review identifies antibacterial phenolic compounds that have been identified in Asian and Pacific Angiosperms from
Externí odkaz:
https://doaj.org/article/638843fdcd1d4d7093fba4195265ce41
Autor:
Muhammad Taha, Fazal Rahim, Bushra Adalath, Syahrul Imran, Khalid Mohammed Khan, Syed Adnan Ali shah, Nizam Uddin, Muhammad Nawaz, Mohammed Khaled Bin Break, Sami M. Magam, Saad Alqarni
Publikováno v:
Arabian Journal of Chemistry, Vol 17, Iss 4, Pp 105700- (2024)
Diabetes and ulcer are the major health problems all over the world. The present study reports synthesis and bio-evaluation of 19 benzimidazole analogs in search of antiglycation, antioxidant and antiulcer agents. The synthetic analogs were character
Externí odkaz:
https://doaj.org/article/ca721f4862044af5828f678474121fcc
Autor:
Amal M. Alosaimy, Amr S. Abouzied, Amani M. R. Alsaedi, Ahmed Alafnan, Abdulwahab Alamri, Mubarak A. Alamri, Mohammed Khaled Bin Break, Rehab Sabour, Thoraya A. Farghaly
Publikováno v:
Arabian Journal of Chemistry, Vol 16, Iss 4, Pp 104569- (2023)
Inhibition of Heat-shock protein 90 (Hsp90) is considered an attractive route in fighting against cancer proliferation. Herein, new indene derivatives targeting Hsp90 were synthesized, and biologically evaluated. The new series of indeno-pyrimidine a
Externí odkaz:
https://doaj.org/article/c9b5c632c22e4a7981ef702db198bbcb
Autor:
Faiza Qureshi, Muhammad Nawaz, Soleiman Hisaindee, Sarah Ameen Almofty, Mohammad Azam Ansari, Qazi Mohammad Sajid Jamal, Nisar Ullah, Muhammad Taha, Ohood Alshehri, Bader Huwaimel, Mohammed Khaled Bin Break
Publikováno v:
Arabian Journal of Chemistry, Vol 15, Iss 12, Pp 104366- (2022)
We report microwave synthesis of seven unique pyrimidine anchored derivatives (1–7) incorporating multifunctional amino derivatives along with their in vitro anticancer activity and their activity against COVID-19 in silico. 1–7 were characterize
Externí odkaz:
https://doaj.org/article/f7ae75344161420d98bc0244e441a388
Autor:
Rahamat Unissa Syed, Sivakumar Sivagurunathan Moni, Mohammed Khaled Bin Break, Weam M. A. Khojali, Mohammed Jafar, Maali D. Alshammari, Karim Abdelsalam, Soha Taymour, Khetam Saad Mutni Alreshidi, Manal Mohamed Elhassan Taha, Syam Mohan
Publikováno v:
Antibiotics, Vol 12, Iss 7, p 1157 (2023)
Broccoli, Brassica oleracea var. italica, has recently gained considerable attention due to its remarkable nutritional composition and numerous health benefits. In this review, the nutritional aspects of broccoli are examined, highlighting its rich n
Externí odkaz:
https://doaj.org/article/373673d45c074bffac296efb4a333368
Autor:
Mohammed Khaled Bin Break, Tan Yew Fung, May Zie Koh, Wan Yong Ho, Mohamed Ibrahim Mohamed Tahir, Omar Ashraf Elfar, Rahamat Unissa Syed, Weam M. A. Khojali, Turki Mubarak Alluhaibi, Bader Huwaimel, Christophe Wiart, Teng-Jin Khoo
Publikováno v:
Molecules, Vol 28, Iss 13, p 5009 (2023)
A series of novel macroacyclic Schiff base ligands and their Cu (II) complexes were synthesised via reacting dicarbonyls of varying chain lengths with S-methyl dithiocarbazate (SMDTC) and S-benzyl dithiocarbazate (SBDTC) followed by coordination with
Externí odkaz:
https://doaj.org/article/e75e33d31c7d4645a5dd533c859cec6a
Autor:
Rahamat Unissa Syed, Sivakumar S. Moni, Muhammad Nawaz, Mohammed Khaled Bin Break, Nasrin E. Khalifa, Siddig Ibrahim Abdelwahab, Reham Meshal Alharbi, Raghad Huraid Alfaisal, Bayan Naif Al Basher, Entsar Mohammed Alhaidan
Publikováno v:
Pharmaceutics, Vol 15, Iss 4, p 1082 (2023)
Amikacin sulfate-loaded dextran sulfate sodium nanoparticles were formulated, lyophilized (LADNP), and then analyzed. The LADNP had a −20.9 ± 8.35 mV zeta potential, PDI of 0.256, and % PDI of 67.7. The zeta average nano size of LADNP was 317.9 z.
Externí odkaz:
https://doaj.org/article/5bf137cb5230467c85f6de6317070df5
Autor:
Weam M. A. Khojali, Weiam Hussein, Mohammed Khaled Bin Break, Ahmed Alafnan, Bader Huwaimel, Nasrin E. Khalifa, Wafa F. S. Badulla, Raghad Abdulkarem Alshammari, Lama Khalid Alshammari, Rehab Aladham Raji Alshammari, Sara Mohsen Albarak, Enas Hmdan Alrkad, Tooba Mahboob, Hisham Alshammari
Publikováno v:
Medicina, Vol 59, Iss 3, p 546 (2023)
Background and Objectives: Ochradenus baccatus belongs to the family Resedaceae. It is widely spread in Saudi Arabia and other countries in Southwest Asia. O. baccatus is extensively used in traditional medicine as an anti-inflammatory and antibacter
Externí odkaz:
https://doaj.org/article/e055ee2d74f644cfaaa76e20a83ac61b
Autor:
Mazdida Sulaiman, Khoshnur Jannat, Veeranoot Nissapatorn, Mohammed Rahmatullah, Alok K. Paul, Maria de Lourdes Pereira, Mogana Rajagopal, Monica Suleiman, Mark S. Butler, Mohammed Khaled Bin Break, Jean-Frédéric Weber, Polrat Wilairatana, Christophe Wiart
Publikováno v:
Antibiotics, Vol 11, Iss 9, p 1146 (2022)
The emergence of multidrug-resistant bacteria and fungi requires the development of antibiotics and antifungal agents. This review identified natural products isolated from Asian angiosperms with antibacterial and/or antifungal activities and analyze
Externí odkaz:
https://doaj.org/article/e6e3b2b2dedf489e806d129a3fd4a310
Autor:
Afrasim Moin, Bader Huwaimel, Ahmed Alobaida, Mohammed Khaled Bin Break, Danish Iqbal, Rahamat Unissa, Qazi Mohammad Sajid Jamal, Talib Hussain, Dinesh C. Sharma, Syed Mohd Danish Rizvi
Publikováno v:
Life, Vol 12, Iss 7, p 1076 (2022)
The COVID-19 era has prompted several researchers to search for a linkage between COVID-19 and its associated neurological manifestation. Toll-like receptor 4 (TLR-4) acts as one such connecting link. spike protein of SARS-CoV-2 can bind either to AC
Externí odkaz:
https://doaj.org/article/845e28718074415aacc2163bd163033e