Efficient Synthesis of 2-Amino-6-Arylbenzothiazoles via Pd(0) Suzuki Cross Coupling Reactions: Potent Urease Enzyme Inhibition and Nitric Oxide Scavenging Activities of the Products

Autor: Md. Saiful Islam, Muhammad Zubair, Iftikhar Hussain Bukhari, Asma Yaqoob, Umer Rashid, Shazia Kousar, Faiz-ul-Hassan Nasim, Mnaza Noreen, Nasir Rasool, Yasmeen Gull

Publikováno v: Molecules, Vol 18, Iss 8, Pp 8845-8857 (2013)

In general, benzothiazole derivatives have attracted great interest due to thier pharmaceutical and biological importance. New 2-amino-6-arylbenzothiazoles were synthesized in moderate to excellent yields via Suzuki cross coupling reactions using var

Externí odkaz: https://doaj.org/article/6b03ed0a8e9040c28d7c7a88397995c0

A convenient method for the synthesis of (prop-2-ynyloxy)benzene derivatives via reaction with propargyl bromide, their optimization, scope and biological evaluation.

Autor: Tannaza Batool, Nasir Rasool, Yasmeen Gull, Mnaza Noreen, Faiz-ul-Hassan Nasim, Asma Yaqoob, Muhammad Zubair, Usman Ali Rana, Salah Ud-Din Khan, M Zia-Ul-Haq, Hawa Z E Jaafar

Publikováno v: PLoS ONE, Vol 9, Iss 12, p e115457 (2014)

A highly convenient method has been developed for the synthesis of (prop-2-ynyloxy) benzene and its derivatives. Differently substituted phenol and aniline derivatives were allowed to react with propargyl bromide in the presence of K2CO3 base and ace

Externí odkaz: https://doaj.org/article/ed7fc025ed684f98ab34fc510161a4b8

Palladium (0) catalyzed Suzuki cross-coupling reactions of 2,4-dibromothiophene: selectivity, characterization and biological applications

Autor: Muhammad Zubair, Yasmeen Gull, Usman Ali Rana, Nasir Rasool, Mnaza Noreen, Aman Ullah, Tehmina Rasheed

Publikováno v: Journal of Sulfur Chemistry. 36:240-250

A series of novel 2-aryl1-4-bromothiophenes (2a–f), biarylthiophenes with non-identical aryl groups (3a–e) and biarylthiophenes with identical aryl groups (4a–f) were synthesized in moderate to excellent yields by using different arylboronic ac

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::630257ab606196f061ec90138dc69ac9
https://doi.org/10.1080/17415993.2015.1020493

Synthesis, Density Functional Theory (DFT), Urease Inhibition and Antimicrobial Activities of 5-Aryl Thiophenes Bearing Sulphonylacetamide Moieties

Autor: Tariq Mahmood, Faiz-ul-Hassan Nasim, Muhammad Zubair, Khurshid Ayub, Yasmeen Gull, Asma Yaqoob, Muhammad Zia-Ul-Haq, Vincenzo De Feo, Mnaza Noreen, Nasir Rasool

Publikováno v: Molecules
Volume 20
Issue 11
Pages 19914-19928
Molecules; Volume 20; Issue 11; Pages: 19914-19928
Molecules, Vol 20, Iss 11, Pp 19914-19928 (2015)

A variety of novel 5-aryl thiophenes 4a–g containing sulphonylacetamide (sulfacetamide) groups were synthesized in appreciable yields via Pd[0] Suzuki cross coupling reactions. The structures of these newly synthesized compounds were determined usi

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::050d3fdc32957524e4eb0da177946835
https://pubmed.ncbi.nlm.nih.gov/26556326

A Convenient Method for the Synthesis of (Prop-2-Ynyloxy)Benzene Derivatives via Reaction with Propargyl Bromide, Their Optimization, Scope and Biological Evaluation

Autor: Mnaza Noreen, Asma Yaqoob, Hawa Z. E. Jaafar, Muhammad Zia-Ul-Haq, Muhammad Zubair, Tannaza Batool, Faiz-ul-Hassan Nasim, Yasmeen Gull, Salah Ud-Din Khan, Usman Ali Rana, Nasir Rasool

Publikováno v: PLoS ONE
PLoS ONE, Vol 9, Iss 12, p e115457 (2014)

A highly convenient method has been developed for the synthesis of (prop-2-ynyloxy) benzene and its derivatives. Differently substituted phenol and aniline derivatives were allowed to react with propargyl bromide in the presence of K2CO3 base and ace

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::82c8f8836247126fe93527ad02472ef8
http://europepmc.org/articles/PMC4278708