Zobrazeno 1 - 10
of 14
pro vyhledávání: '"Mitsuo Sugiyama"'
Autor:
Katsuyoshi Nakajima, Mitsuo Sugiyama, Hiroyoshi Horikoshi, Takahide Nishi, Yuki Sugioka, Koki Ishibashi, Hamada Takakazu
Publikováno v:
Chemical and Pharmaceutical Bulletin. 47:226-240
A series of 2-phenylbenzofuran derivatives with a carbamoyl, alkylamino, or alkyloxy group at the 5 or 6 position of the benzofuran ring were synthesized and evaluated for rat and human testosterone 5 alpha-reductase inhibitory activities in vitro. A
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::041dcdf86e52f4d5bb1164c8405a617a
https://doi.org/10.1248/cpb.47.226
https://doi.org/10.1248/cpb.47.226
Autor:
Hamada Takakazu, Takahide Nishi, Yuki Sugioka, Katsuyoshi Nakajima, Mitsuo Sugiyama, Koki Ishibashi, Hiroyoshi Horikoshi
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 8:561-566
A series of 2-phenylbenzofuran derivatives with a diphenylmethylcarbamoyl group at the 5 or 6 position of the benzofuran ring were synthesized and evaluated for rat and human testosterone 5α-reductase inhibitory activities in vitro. They had inhibit
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8a1eed4e2fb958d7b98577590857f1bf
https://doi.org/10.1016/s0960-894x(98)00001-8
https://doi.org/10.1016/s0960-894x(98)00001-8
Autor:
Kazuhiro Itoh, Toshiaki Sakamoto, Yumiko Kamigaki, Yumiko Satoh, Takeshi Yamaguchi, Mitsuo Sugiyama, Fukumi Hiroshi
Publikováno v:
ChemInform. 26
A new series of piperidineacrylate derivatives was prepared and evaluated for antiallergic activity. Most of the compounds showed potent activities in the rat passive cutaneous anaphylaxis (PCA) assay. In particular, ethyl 1-[2-bis(4-fluorophenyl)met
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::34094ca6fdd724b259da961ca86fcd04
https://doi.org/10.1002/chin.199506153
https://doi.org/10.1002/chin.199506153
Autor:
Hiroyoshi Horikoshi, Mitsuo Sugiyama, Takahide Nishi, Hamada Takakazu, Koki Ishibashi, Katsuyoshi Nakajima, Yuki Sugioka
Publikováno v:
ChemInform. 29
A series of 2-phenylbenzofuran derivatives with a diphenylmethylcarbamoyl group at the 5 or 6 position of the benzofuran ring were synthesized and evaluated for rat and human testosterone 5α-reductase inhibitory activities in vitro. They had inhibit
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::23877a3e3370e8072920d6531a8e0339
https://doi.org/10.1002/chin.199828136
https://doi.org/10.1002/chin.199828136
Autor:
Takahide Nishi, Hamada Takakazu, Mitsuo Sugiyama, Hiroyoshi Horikoshi, Yuki Sugioka, Koki Ishibashi, Katsuyoshi Nakajima
Publikováno v:
ChemInform. 30
A series of 2-phenylbenzofuran derivatives with a carbamoyl, alkylamino, or alkyloxy group at the 5 or 6 position of the benzofuran ring were synthesized and evaluated for rat and human testosterone 5α-reductase inhibitory activities in vitro. Again
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::45d4764af392ca73b9a81dab09e7869b
https://doi.org/10.1002/chin.199937113
https://doi.org/10.1002/chin.199937113
Autor:
Yumiko Satoh, Fukumi Hiroshi, Toshiaki Sakamoto, Kazuhiro Itoh, Takeshi Yamaguchi, Mitsuo Sugiyama, Yumiko Kamigaki
Publikováno v:
Chemicalpharmaceutical bulletin. 41(5)
A new series of piperidineacrylate derivatives was prepared and evaluated for antiallergic activity. Most of the compounds showed potent activities in the rat passive cutaneous anaphylaxis (PCA) assay. In particular, ethyl 1-[2-bis(4-fluorophenyl)met
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::dcc37749e7c9de25bfb33347e7a4db6f
https://pubmed.ncbi.nlm.nih.gov/8339335
https://pubmed.ncbi.nlm.nih.gov/8339335
Publikováno v:
ChemInform. 21
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::437a30ca5189ff745bc3f7a242067d29
https://doi.org/10.1002/chin.199016190
https://doi.org/10.1002/chin.199016190
Publikováno v:
ChemInform. 21
A practical preparation of 2, 3-dihydro-5H-oxazolo[3, 2-a]thieno[3, 2-d]pyrimidin-5-oen (2) from methyl 3-aminothiophene-2-carboxylate in two steps was developed. The addition reactions of various nucleophiles to 2 were investigated and oxazole-ring-
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::b5ab2957e40be82a5198a919847284db
https://doi.org/10.1002/chin.199001237
https://doi.org/10.1002/chin.199001237
Autor:
Mitsuko Kobayashi, Keiichi Ito, Keiichi Tabata, Fukumi Hiroshi, Kazuo Endo, Mitsuo Sugiyama, Toshiaki Sakamoto
Publikováno v:
Chemical and Pharmaceutical Bulletin. 37:2122-2131
Thiazolo[3,2-a]thieno[3,2-d]-, [3,4-d]- and [2,3-d]pyrimidin-5-one derivatives (6, 11 and 16), and polymethylene condensed thieno[3,2-d]-, [3,4-d]- and [2,3-d]pyrimidin-5-one derivatives (19-21), in which the oxygen atom of the oxazolidine moiety in
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a12c1e89fb74c977cbc3a3b7ea3d4d46
https://doi.org/10.1248/cpb.37.2122
https://doi.org/10.1248/cpb.37.2122
Autor:
Mitsuo Sugiyama, Juichi Koshikawa
Publikováno v:
Sen-ito Kogyo. 2:829-833
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::afbbf66436ef2bd2d997c5e206c87c2c
https://doi.org/10.2115/fiber1968.2.829
https://doi.org/10.2115/fiber1968.2.829